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Found 12 Enz. Inhib. hit(s) with all data for entry = 50000648
TargetMu-type opioid receptor(Rattus norvegicus (rat))
The Reproductive Medicine Special Hospital Of The First Hospital Of Lanzhou University

Curated by ChEMBL
LigandPNGBDBM50256911(CHEMBL4095621)
Affinity DataKi:  0.350nMAssay Description:Displacement of [3H]DAMGO from mu-opioid receptor in Wistar rat brain membrane after 1 hr by microbeta scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
The Reproductive Medicine Special Hospital Of The First Hospital Of Lanzhou University

Curated by ChEMBL
LigandPNGBDBM50256914(CHEMBL4061665)
Affinity DataKi:  0.420nMAssay Description:Displacement of [3H]DAMGO from mu-opioid receptor in Wistar rat brain membrane after 1 hr by microbeta scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
The Reproductive Medicine Special Hospital Of The First Hospital Of Lanzhou University

Curated by ChEMBL
LigandPNGBDBM50256915(CHEMBL4068851)
Affinity DataKi:  1.20nMAssay Description:Displacement of [3H]DAMGO from mu-opioid receptor in Wistar rat brain membrane after 1 hr by microbeta scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
The Reproductive Medicine Special Hospital Of The First Hospital Of Lanzhou University

Curated by ChEMBL
LigandPNGBDBM21123((2S)-2-{2-[(2R)-2-[(2S)-2-amino-3-(4-hydroxyphenyl...)
Affinity DataKi:  2.10nMAssay Description:Displacement of [3H]DAMGO from mu-opioid receptor in Wistar rat brain membrane after 1 hr by microbeta scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
The Reproductive Medicine Special Hospital Of The First Hospital Of Lanzhou University

Curated by ChEMBL
LigandPNGBDBM50095155((S)-1-[(S)-2-Amino-3-(4-hydroxy-phenyl)-propionyl]...)
Affinity DataKi:  6.20nMAssay Description:Displacement of [3H]DAMGO from mu-opioid receptor in Wistar rat brain membrane after 1 hr by microbeta scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
The Reproductive Medicine Special Hospital Of The First Hospital Of Lanzhou University

Curated by ChEMBL
LigandPNGBDBM50256911(CHEMBL4095621)
Affinity DataKi:  101nMAssay Description:Displacement of [3H]DPDPE from delta-opioid receptor in Wistar rat brain membrane after 3 hrs by microbeta scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
The Reproductive Medicine Special Hospital Of The First Hospital Of Lanzhou University

Curated by ChEMBL
LigandPNGBDBM50256916(CHEMBL4096142)
Affinity DataKi:  247nMAssay Description:Displacement of [3H]DAMGO from mu-opioid receptor in Wistar rat brain membrane after 1 hr by microbeta scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
The Reproductive Medicine Special Hospital Of The First Hospital Of Lanzhou University

Curated by ChEMBL
LigandPNGBDBM50256914(CHEMBL4061665)
Affinity DataKi:  840nMAssay Description:Displacement of [3H]DPDPE from delta-opioid receptor in Wistar rat brain membrane after 3 hrs by microbeta scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
The Reproductive Medicine Special Hospital Of The First Hospital Of Lanzhou University

Curated by ChEMBL
LigandPNGBDBM50256915(CHEMBL4068851)
Affinity DataKi: >1.00E+3nMAssay Description:Displacement of [3H]DPDPE from delta-opioid receptor in Wistar rat brain membrane after 3 hrs by microbeta scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
The Reproductive Medicine Special Hospital Of The First Hospital Of Lanzhou University

Curated by ChEMBL
LigandPNGBDBM21123((2S)-2-{2-[(2R)-2-[(2S)-2-amino-3-(4-hydroxyphenyl...)
Affinity DataKi:  3.80E+3nMAssay Description:Displacement of [3H]DPDPE from delta-opioid receptor in Wistar rat brain membrane after 3 hrs by microbeta scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
The Reproductive Medicine Special Hospital Of The First Hospital Of Lanzhou University

Curated by ChEMBL
LigandPNGBDBM50256916(CHEMBL4096142)
Affinity DataKi:  4.55E+3nMAssay Description:Displacement of [3H]DPDPE from delta-opioid receptor in Wistar rat brain membrane after 3 hrs by microbeta scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
The Reproductive Medicine Special Hospital Of The First Hospital Of Lanzhou University

Curated by ChEMBL
LigandPNGBDBM50095155((S)-1-[(S)-2-Amino-3-(4-hydroxy-phenyl)-propionyl]...)
Affinity DataKi:  5.78E+3nMAssay Description:Displacement of [3H]DPDPE from delta-opioid receptor in Wistar rat brain membrane after 3 hrs by microbeta scintillation counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed