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Found 12 Enz. Inhib. hit(s) with all data for entry = 50000505
TargetSerine/threonine-protein kinase pim-1(Homo sapiens (Human))
Ain Shams University

Curated by ChEMBL
LigandPNGBDBM50251746(CHEMBL4079516)
Affinity DataIC50:  940nMAssay Description:Inhibition of human PIM1 measured after 5 mins by ELISA relative to controlMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase pim-1(Homo sapiens (Human))
Ain Shams University

Curated by ChEMBL
LigandPNGBDBM50251734(CHEMBL4096022)
Affinity DataIC50:  1.16E+3nMAssay Description:Inhibition of human PIM1 measured after 5 mins by ELISA relative to controlMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase pim-1(Homo sapiens (Human))
Ain Shams University

Curated by ChEMBL
LigandPNGBDBM50251735(CHEMBL4103770)
Affinity DataIC50:  1.47E+3nMAssay Description:Inhibition of human PIM1 measured after 5 mins by ELISA relative to controlMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase pim-1(Homo sapiens (Human))
Ain Shams University

Curated by ChEMBL
LigandPNGBDBM50251752(CHEMBL1306213)
Affinity DataIC50:  3.16E+3nMAssay Description:Inhibition of human PIM1 measured after 5 mins by ELISA relative to controlMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase pim-1(Homo sapiens (Human))
Ain Shams University

Curated by ChEMBL
LigandPNGBDBM50014846((S)-N-(5,6,7,9-tetrahydro-1,2,3,10-tetramethoxy-9-...)
Affinity DataIC50:  4.30E+3nMAssay Description:Inhibition of human PIM1 measured after 5 mins by ELISA relative to controlMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase pim-1(Homo sapiens (Human))
Ain Shams University

Curated by ChEMBL
LigandPNGBDBM50251760(CHEMBL4087394)
Affinity DataIC50:  4.80E+3nMAssay Description:Inhibition of human PIM1 measured after 5 mins by ELISA relative to controlMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase pim-1(Homo sapiens (Human))
Ain Shams University

Curated by ChEMBL
LigandPNGBDBM50251747(CHEMBL2235178)
Affinity DataIC50:  6.70E+3nMAssay Description:Inhibition of human PIM1 measured after 5 mins by ELISA relative to controlMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase pim-1(Homo sapiens (Human))
Ain Shams University

Curated by ChEMBL
LigandPNGBDBM50262435(2-Amino-4,6-di-thiophen-2-yl-nicotinonitrile | CHE...)
Affinity DataIC50:  7.52E+3nMAssay Description:Inhibition of human PIM1 measured after 5 mins by ELISA relative to controlMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase pim-1(Homo sapiens (Human))
Ain Shams University

Curated by ChEMBL
LigandPNGBDBM50251753(CHEMBL4095080)
Affinity DataIC50:  1.00E+4nMAssay Description:Inhibition of human PIM1 measured after 5 mins by ELISA relative to controlMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase pim-1(Homo sapiens (Human))
Ain Shams University

Curated by ChEMBL
LigandPNGBDBM50251759(CHEMBL4068706)
Affinity DataIC50:  1.06E+4nMAssay Description:Inhibition of human PIM1 measured after 5 mins by ELISA relative to controlMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase pim-1(Homo sapiens (Human))
Ain Shams University

Curated by ChEMBL
LigandPNGBDBM50251754(CHEMBL4074899)
Affinity DataIC50:  1.93E+4nMAssay Description:Inhibition of human PIM1 measured after 5 mins by ELISA relative to controlMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase pim-1(Homo sapiens (Human))
Ain Shams University

Curated by ChEMBL
LigandPNGBDBM50251733(CHEMBL4063523)
Affinity DataIC50:  2.55E+4nMAssay Description:Inhibition of human PIM1 measured after 5 mins by ELISA relative to controlMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed