Compile Data Set for Download or QSAR
maximum 50k data
Found 32 Enz. Inhib. hit(s) with all data for entry = 50002896
TargetTyrosine-protein kinase BTK(Homo sapiens (Human))
The First Affiliated Hospital Of Dalian Medical University

Curated by ChEMBL
LigandPNGBDBM50357312(IBRUTINIB | PCI-32765 | US10124003, Ref. Ex. Compo...)
Affinity DataIC50:  0.300nMAssay Description:Inhibition of recombinant full-length N-terminal His-tagged human BTK expressed in baculovirus infected Sf9 insect cells using Poly(4:1 Glu,Tyr) pept...More data for this Ligand-Target Pair
TargetTyrosine-protein kinase BTK(Homo sapiens (Human))
The First Affiliated Hospital Of Dalian Medical University

Curated by ChEMBL
LigandPNGBDBM50464517(CHEMBL4294772)
Affinity DataIC50:  0.5nMAssay Description:Inhibition of recombinant full-length N-terminal His-tagged human BTK expressed in baculovirus infected Sf9 insect cells using Poly(4:1 Glu,Tyr) pept...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase BTK(Homo sapiens (Human))
The First Affiliated Hospital Of Dalian Medical University

Curated by ChEMBL
LigandPNGBDBM50161162(AVL-292 | CC-292 | Spebrutinib | US10596172, Compo...)
Affinity DataIC50:  0.600nMAssay Description:Inhibition of recombinant full-length N-terminal His-tagged human BTK expressed in baculovirus infected Sf9 insect cells using Poly(4:1 Glu,Tyr) pept...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase BTK(Homo sapiens (Human))
The First Affiliated Hospital Of Dalian Medical University

Curated by ChEMBL
LigandPNGBDBM50464516(CHEMBL4290692)
Affinity DataIC50:  0.600nMAssay Description:Inhibition of recombinant full-length N-terminal His-tagged human BTK expressed in baculovirus infected Sf9 insect cells using Poly(4:1 Glu,Tyr) pept...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase JAK3(Homo sapiens (Human))
The First Affiliated Hospital Of Dalian Medical University

Curated by ChEMBL
LigandPNGBDBM50464521(CHEMBL4289281)
Affinity DataIC50:  0.690nMAssay Description:Inhibition of recombinant N-terminal GST-tagged human JAK3 (781 to end residues) expressed in baculovirus infected Sf9 insect cells using Poly(4:1 Gl...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase BTK(Homo sapiens (Human))
The First Affiliated Hospital Of Dalian Medical University

Curated by ChEMBL
LigandPNGBDBM50464524(CHEMBL4290449)
Affinity DataIC50:  0.700nMAssay Description:Inhibition of recombinant full-length N-terminal His-tagged human BTK expressed in baculovirus infected Sf9 insect cells using Poly(4:1 Glu,Tyr) pept...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase BTK(Homo sapiens (Human))
The First Affiliated Hospital Of Dalian Medical University

Curated by ChEMBL
LigandPNGBDBM50464526(CHEMBL4284156)
Affinity DataIC50:  0.700nMAssay Description:Inhibition of recombinant full-length N-terminal His-tagged human BTK expressed in baculovirus infected Sf9 insect cells using Poly(4:1 Glu,Tyr) pept...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase BTK(Homo sapiens (Human))
The First Affiliated Hospital Of Dalian Medical University

Curated by ChEMBL
LigandPNGBDBM50464513(CHEMBL4286900)
Affinity DataIC50:  0.800nMAssay Description:Inhibition of recombinant full-length N-terminal His-tagged human BTK expressed in baculovirus infected Sf9 insect cells using Poly(4:1 Glu,Tyr) pept...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase BTK(Homo sapiens (Human))
The First Affiliated Hospital Of Dalian Medical University

Curated by ChEMBL
LigandPNGBDBM50464521(CHEMBL4289281)
Affinity DataIC50:  0.800nMAssay Description:Inhibition of recombinant full-length N-terminal His-tagged human BTK expressed in baculovirus infected Sf9 insect cells using Poly(4:1 Glu,Tyr) pept...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase JAK3(Homo sapiens (Human))
The First Affiliated Hospital Of Dalian Medical University

Curated by ChEMBL
LigandPNGBDBM50464516(CHEMBL4290692)
Affinity DataIC50:  0.830nMAssay Description:Inhibition of recombinant N-terminal GST-tagged human JAK3 (781 to end residues) expressed in baculovirus infected Sf9 insect cells using Poly(4:1 Gl...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase JAK3(Homo sapiens (Human))
The First Affiliated Hospital Of Dalian Medical University

Curated by ChEMBL
LigandPNGBDBM50464517(CHEMBL4294772)
Affinity DataIC50:  0.910nMAssay Description:Inhibition of recombinant N-terminal GST-tagged human JAK3 (781 to end residues) expressed in baculovirus infected Sf9 insect cells using Poly(4:1 Gl...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase JAK3(Homo sapiens (Human))
The First Affiliated Hospital Of Dalian Medical University

Curated by ChEMBL
LigandPNGBDBM50464524(CHEMBL4290449)
Affinity DataIC50:  0.950nMAssay Description:Inhibition of recombinant N-terminal GST-tagged human JAK3 (781 to end residues) expressed in baculovirus infected Sf9 insect cells using Poly(4:1 Gl...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase BTK(Homo sapiens (Human))
The First Affiliated Hospital Of Dalian Medical University

Curated by ChEMBL
LigandPNGBDBM50464515(CHEMBL4289688)
Affinity DataIC50:  1nMAssay Description:Inhibition of recombinant full-length N-terminal His-tagged human BTK expressed in baculovirus infected Sf9 insect cells using Poly(4:1 Glu,Tyr) pept...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase JAK3(Homo sapiens (Human))
The First Affiliated Hospital Of Dalian Medical University

Curated by ChEMBL
LigandPNGBDBM50464526(CHEMBL4284156)
Affinity DataIC50:  1.10nMAssay Description:Inhibition of recombinant N-terminal GST-tagged human JAK3 (781 to end residues) expressed in baculovirus infected Sf9 insect cells using Poly(4:1 Gl...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase JAK3(Homo sapiens (Human))
The First Affiliated Hospital Of Dalian Medical University

Curated by ChEMBL
LigandPNGBDBM50464515(CHEMBL4289688)
Affinity DataIC50:  1.40nMAssay Description:Inhibition of recombinant N-terminal GST-tagged human JAK3 (781 to end residues) expressed in baculovirus infected Sf9 insect cells using Poly(4:1 Gl...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase JAK3(Homo sapiens (Human))
The First Affiliated Hospital Of Dalian Medical University

Curated by ChEMBL
LigandPNGBDBM50464518(CHEMBL4292468)
Affinity DataIC50:  6.80nMAssay Description:Inhibition of recombinant N-terminal GST-tagged human JAK3 (781 to end residues) expressed in baculovirus infected Sf9 insect cells using Poly(4:1 Gl...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase JAK3(Homo sapiens (Human))
The First Affiliated Hospital Of Dalian Medical University

Curated by ChEMBL
LigandPNGBDBM50464513(CHEMBL4286900)
Affinity DataIC50:  8.30nMAssay Description:Inhibition of recombinant N-terminal GST-tagged human JAK3 (781 to end residues) expressed in baculovirus infected Sf9 insect cells using Poly(4:1 Gl...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase JAK3(Homo sapiens (Human))
The First Affiliated Hospital Of Dalian Medical University

Curated by ChEMBL
LigandPNGBDBM50464522(CHEMBL4280709)
Affinity DataIC50:  11nMAssay Description:Inhibition of recombinant N-terminal GST-tagged human JAK3 (781 to end residues) expressed in baculovirus infected Sf9 insect cells using Poly(4:1 Gl...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase BTK(Homo sapiens (Human))
The First Affiliated Hospital Of Dalian Medical University

Curated by ChEMBL
LigandPNGBDBM50464514(CHEMBL4278652)
Affinity DataIC50:  11nMAssay Description:Inhibition of recombinant full-length N-terminal His-tagged human BTK expressed in baculovirus infected Sf9 insect cells using Poly(4:1 Glu,Tyr) pept...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase JAK3(Homo sapiens (Human))
The First Affiliated Hospital Of Dalian Medical University

Curated by ChEMBL
LigandPNGBDBM50357312(IBRUTINIB | PCI-32765 | US10124003, Ref. Ex. Compo...)
Affinity DataIC50:  16nMAssay Description:Inhibition of recombinant N-terminal GST-tagged human JAK3 (781 to end residues) expressed in baculovirus infected Sf9 insect cells using Poly(4:1 Gl...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase BTK(Homo sapiens (Human))
The First Affiliated Hospital Of Dalian Medical University

Curated by ChEMBL
LigandPNGBDBM50464522(CHEMBL4280709)
Affinity DataIC50:  17nMAssay Description:Inhibition of recombinant full-length N-terminal His-tagged human BTK expressed in baculovirus infected Sf9 insect cells using Poly(4:1 Glu,Tyr) pept...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase JAK3(Homo sapiens (Human))
The First Affiliated Hospital Of Dalian Medical University

Curated by ChEMBL
LigandPNGBDBM50464514(CHEMBL4278652)
Affinity DataIC50:  22nMAssay Description:Inhibition of recombinant N-terminal GST-tagged human JAK3 (781 to end residues) expressed in baculovirus infected Sf9 insect cells using Poly(4:1 Gl...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase JAK3(Homo sapiens (Human))
The First Affiliated Hospital Of Dalian Medical University

Curated by ChEMBL
LigandPNGBDBM50161162(AVL-292 | CC-292 | Spebrutinib | US10596172, Compo...)
Affinity DataIC50:  23nMAssay Description:Inhibition of recombinant N-terminal GST-tagged human JAK3 (781 to end residues) expressed in baculovirus infected Sf9 insect cells using Poly(4:1 Gl...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase BTK(Homo sapiens (Human))
The First Affiliated Hospital Of Dalian Medical University

Curated by ChEMBL
LigandPNGBDBM50464518(CHEMBL4292468)
Affinity DataIC50:  31nMAssay Description:Inhibition of recombinant full-length N-terminal His-tagged human BTK expressed in baculovirus infected Sf9 insect cells using Poly(4:1 Glu,Tyr) pept...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase BTK(Homo sapiens (Human))
The First Affiliated Hospital Of Dalian Medical University

Curated by ChEMBL
LigandPNGBDBM50464520(CHEMBL4287960)
Affinity DataIC50:  82nMAssay Description:Inhibition of recombinant full-length N-terminal His-tagged human BTK expressed in baculovirus infected Sf9 insect cells using Poly(4:1 Glu,Tyr) pept...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase BTK(Homo sapiens (Human))
The First Affiliated Hospital Of Dalian Medical University

Curated by ChEMBL
LigandPNGBDBM50464525(CHEMBL4279066)
Affinity DataIC50:  89nMAssay Description:Inhibition of recombinant full-length N-terminal His-tagged human BTK expressed in baculovirus infected Sf9 insect cells using Poly(4:1 Glu,Tyr) pept...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase BTK(Homo sapiens (Human))
The First Affiliated Hospital Of Dalian Medical University

Curated by ChEMBL
LigandPNGBDBM50464523(CHEMBL4277319)
Affinity DataIC50:  90nMAssay Description:Inhibition of recombinant full-length N-terminal His-tagged human BTK expressed in baculovirus infected Sf9 insect cells using Poly(4:1 Glu,Tyr) pept...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase JAK3(Homo sapiens (Human))
The First Affiliated Hospital Of Dalian Medical University

Curated by ChEMBL
LigandPNGBDBM50464520(CHEMBL4287960)
Affinity DataIC50:  91nMAssay Description:Inhibition of recombinant N-terminal GST-tagged human JAK3 (781 to end residues) expressed in baculovirus infected Sf9 insect cells using Poly(4:1 Gl...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase JAK3(Homo sapiens (Human))
The First Affiliated Hospital Of Dalian Medical University

Curated by ChEMBL
LigandPNGBDBM50464525(CHEMBL4279066)
Affinity DataIC50: >100nMAssay Description:Inhibition of recombinant N-terminal GST-tagged human JAK3 (781 to end residues) expressed in baculovirus infected Sf9 insect cells using Poly(4:1 Gl...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase JAK3(Homo sapiens (Human))
The First Affiliated Hospital Of Dalian Medical University

Curated by ChEMBL
LigandPNGBDBM50464523(CHEMBL4277319)
Affinity DataIC50: >100nMAssay Description:Inhibition of recombinant N-terminal GST-tagged human JAK3 (781 to end residues) expressed in baculovirus infected Sf9 insect cells using Poly(4:1 Gl...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase JAK3(Homo sapiens (Human))
The First Affiliated Hospital Of Dalian Medical University

Curated by ChEMBL
LigandPNGBDBM50464519(CHEMBL4284578)
Affinity DataIC50: >100nMAssay Description:Inhibition of recombinant N-terminal GST-tagged human JAK3 (781 to end residues) expressed in baculovirus infected Sf9 insect cells using Poly(4:1 Gl...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase BTK(Homo sapiens (Human))
The First Affiliated Hospital Of Dalian Medical University

Curated by ChEMBL
LigandPNGBDBM50464519(CHEMBL4284578)
Affinity DataIC50: >100nMAssay Description:Inhibition of recombinant full-length N-terminal His-tagged human BTK expressed in baculovirus infected Sf9 insect cells using Poly(4:1 Glu,Tyr) pept...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed