TargetTyrosine-protein kinase BTK(Homo sapiens (Human))
The First Affiliated Hospital Of Dalian Medical University
Curated by ChEMBL
The First Affiliated Hospital Of Dalian Medical University
Curated by ChEMBL
Affinity DataIC50: 0.300nMAssay Description:Inhibition of recombinant full-length N-terminal His-tagged human BTK expressed in baculovirus infected Sf9 insect cells using Poly(4:1 Glu,Tyr) pept...More data for this Ligand-Target Pair
TargetTyrosine-protein kinase BTK(Homo sapiens (Human))
The First Affiliated Hospital Of Dalian Medical University
Curated by ChEMBL
The First Affiliated Hospital Of Dalian Medical University
Curated by ChEMBL
Affinity DataIC50: 0.5nMAssay Description:Inhibition of recombinant full-length N-terminal His-tagged human BTK expressed in baculovirus infected Sf9 insect cells using Poly(4:1 Glu,Tyr) pept...More data for this Ligand-Target Pair
TargetTyrosine-protein kinase BTK(Homo sapiens (Human))
The First Affiliated Hospital Of Dalian Medical University
Curated by ChEMBL
The First Affiliated Hospital Of Dalian Medical University
Curated by ChEMBL
Affinity DataIC50: 0.600nMAssay Description:Inhibition of recombinant full-length N-terminal His-tagged human BTK expressed in baculovirus infected Sf9 insect cells using Poly(4:1 Glu,Tyr) pept...More data for this Ligand-Target Pair
TargetTyrosine-protein kinase BTK(Homo sapiens (Human))
The First Affiliated Hospital Of Dalian Medical University
Curated by ChEMBL
The First Affiliated Hospital Of Dalian Medical University
Curated by ChEMBL
Affinity DataIC50: 0.600nMAssay Description:Inhibition of recombinant full-length N-terminal His-tagged human BTK expressed in baculovirus infected Sf9 insect cells using Poly(4:1 Glu,Tyr) pept...More data for this Ligand-Target Pair
TargetTyrosine-protein kinase JAK3(Homo sapiens (Human))
The First Affiliated Hospital Of Dalian Medical University
Curated by ChEMBL
The First Affiliated Hospital Of Dalian Medical University
Curated by ChEMBL
Affinity DataIC50: 0.690nMAssay Description:Inhibition of recombinant N-terminal GST-tagged human JAK3 (781 to end residues) expressed in baculovirus infected Sf9 insect cells using Poly(4:1 Gl...More data for this Ligand-Target Pair
TargetTyrosine-protein kinase BTK(Homo sapiens (Human))
The First Affiliated Hospital Of Dalian Medical University
Curated by ChEMBL
The First Affiliated Hospital Of Dalian Medical University
Curated by ChEMBL
Affinity DataIC50: 0.700nMAssay Description:Inhibition of recombinant full-length N-terminal His-tagged human BTK expressed in baculovirus infected Sf9 insect cells using Poly(4:1 Glu,Tyr) pept...More data for this Ligand-Target Pair
TargetTyrosine-protein kinase BTK(Homo sapiens (Human))
The First Affiliated Hospital Of Dalian Medical University
Curated by ChEMBL
The First Affiliated Hospital Of Dalian Medical University
Curated by ChEMBL
Affinity DataIC50: 0.700nMAssay Description:Inhibition of recombinant full-length N-terminal His-tagged human BTK expressed in baculovirus infected Sf9 insect cells using Poly(4:1 Glu,Tyr) pept...More data for this Ligand-Target Pair
TargetTyrosine-protein kinase BTK(Homo sapiens (Human))
The First Affiliated Hospital Of Dalian Medical University
Curated by ChEMBL
The First Affiliated Hospital Of Dalian Medical University
Curated by ChEMBL
Affinity DataIC50: 0.800nMAssay Description:Inhibition of recombinant full-length N-terminal His-tagged human BTK expressed in baculovirus infected Sf9 insect cells using Poly(4:1 Glu,Tyr) pept...More data for this Ligand-Target Pair
TargetTyrosine-protein kinase BTK(Homo sapiens (Human))
The First Affiliated Hospital Of Dalian Medical University
Curated by ChEMBL
The First Affiliated Hospital Of Dalian Medical University
Curated by ChEMBL
Affinity DataIC50: 0.800nMAssay Description:Inhibition of recombinant full-length N-terminal His-tagged human BTK expressed in baculovirus infected Sf9 insect cells using Poly(4:1 Glu,Tyr) pept...More data for this Ligand-Target Pair
TargetTyrosine-protein kinase JAK3(Homo sapiens (Human))
The First Affiliated Hospital Of Dalian Medical University
Curated by ChEMBL
The First Affiliated Hospital Of Dalian Medical University
Curated by ChEMBL
Affinity DataIC50: 0.830nMAssay Description:Inhibition of recombinant N-terminal GST-tagged human JAK3 (781 to end residues) expressed in baculovirus infected Sf9 insect cells using Poly(4:1 Gl...More data for this Ligand-Target Pair
TargetTyrosine-protein kinase JAK3(Homo sapiens (Human))
The First Affiliated Hospital Of Dalian Medical University
Curated by ChEMBL
The First Affiliated Hospital Of Dalian Medical University
Curated by ChEMBL
Affinity DataIC50: 0.910nMAssay Description:Inhibition of recombinant N-terminal GST-tagged human JAK3 (781 to end residues) expressed in baculovirus infected Sf9 insect cells using Poly(4:1 Gl...More data for this Ligand-Target Pair
TargetTyrosine-protein kinase JAK3(Homo sapiens (Human))
The First Affiliated Hospital Of Dalian Medical University
Curated by ChEMBL
The First Affiliated Hospital Of Dalian Medical University
Curated by ChEMBL
Affinity DataIC50: 0.950nMAssay Description:Inhibition of recombinant N-terminal GST-tagged human JAK3 (781 to end residues) expressed in baculovirus infected Sf9 insect cells using Poly(4:1 Gl...More data for this Ligand-Target Pair
TargetTyrosine-protein kinase BTK(Homo sapiens (Human))
The First Affiliated Hospital Of Dalian Medical University
Curated by ChEMBL
The First Affiliated Hospital Of Dalian Medical University
Curated by ChEMBL
Affinity DataIC50: 1nMAssay Description:Inhibition of recombinant full-length N-terminal His-tagged human BTK expressed in baculovirus infected Sf9 insect cells using Poly(4:1 Glu,Tyr) pept...More data for this Ligand-Target Pair
TargetTyrosine-protein kinase JAK3(Homo sapiens (Human))
The First Affiliated Hospital Of Dalian Medical University
Curated by ChEMBL
The First Affiliated Hospital Of Dalian Medical University
Curated by ChEMBL
Affinity DataIC50: 1.10nMAssay Description:Inhibition of recombinant N-terminal GST-tagged human JAK3 (781 to end residues) expressed in baculovirus infected Sf9 insect cells using Poly(4:1 Gl...More data for this Ligand-Target Pair
TargetTyrosine-protein kinase JAK3(Homo sapiens (Human))
The First Affiliated Hospital Of Dalian Medical University
Curated by ChEMBL
The First Affiliated Hospital Of Dalian Medical University
Curated by ChEMBL
Affinity DataIC50: 1.40nMAssay Description:Inhibition of recombinant N-terminal GST-tagged human JAK3 (781 to end residues) expressed in baculovirus infected Sf9 insect cells using Poly(4:1 Gl...More data for this Ligand-Target Pair
TargetTyrosine-protein kinase JAK3(Homo sapiens (Human))
The First Affiliated Hospital Of Dalian Medical University
Curated by ChEMBL
The First Affiliated Hospital Of Dalian Medical University
Curated by ChEMBL
Affinity DataIC50: 6.80nMAssay Description:Inhibition of recombinant N-terminal GST-tagged human JAK3 (781 to end residues) expressed in baculovirus infected Sf9 insect cells using Poly(4:1 Gl...More data for this Ligand-Target Pair
TargetTyrosine-protein kinase JAK3(Homo sapiens (Human))
The First Affiliated Hospital Of Dalian Medical University
Curated by ChEMBL
The First Affiliated Hospital Of Dalian Medical University
Curated by ChEMBL
Affinity DataIC50: 8.30nMAssay Description:Inhibition of recombinant N-terminal GST-tagged human JAK3 (781 to end residues) expressed in baculovirus infected Sf9 insect cells using Poly(4:1 Gl...More data for this Ligand-Target Pair
TargetTyrosine-protein kinase JAK3(Homo sapiens (Human))
The First Affiliated Hospital Of Dalian Medical University
Curated by ChEMBL
The First Affiliated Hospital Of Dalian Medical University
Curated by ChEMBL
Affinity DataIC50: 11nMAssay Description:Inhibition of recombinant N-terminal GST-tagged human JAK3 (781 to end residues) expressed in baculovirus infected Sf9 insect cells using Poly(4:1 Gl...More data for this Ligand-Target Pair
TargetTyrosine-protein kinase BTK(Homo sapiens (Human))
The First Affiliated Hospital Of Dalian Medical University
Curated by ChEMBL
The First Affiliated Hospital Of Dalian Medical University
Curated by ChEMBL
Affinity DataIC50: 11nMAssay Description:Inhibition of recombinant full-length N-terminal His-tagged human BTK expressed in baculovirus infected Sf9 insect cells using Poly(4:1 Glu,Tyr) pept...More data for this Ligand-Target Pair
TargetTyrosine-protein kinase JAK3(Homo sapiens (Human))
The First Affiliated Hospital Of Dalian Medical University
Curated by ChEMBL
The First Affiliated Hospital Of Dalian Medical University
Curated by ChEMBL
Affinity DataIC50: 16nMAssay Description:Inhibition of recombinant N-terminal GST-tagged human JAK3 (781 to end residues) expressed in baculovirus infected Sf9 insect cells using Poly(4:1 Gl...More data for this Ligand-Target Pair
TargetTyrosine-protein kinase BTK(Homo sapiens (Human))
The First Affiliated Hospital Of Dalian Medical University
Curated by ChEMBL
The First Affiliated Hospital Of Dalian Medical University
Curated by ChEMBL
Affinity DataIC50: 17nMAssay Description:Inhibition of recombinant full-length N-terminal His-tagged human BTK expressed in baculovirus infected Sf9 insect cells using Poly(4:1 Glu,Tyr) pept...More data for this Ligand-Target Pair
TargetTyrosine-protein kinase JAK3(Homo sapiens (Human))
The First Affiliated Hospital Of Dalian Medical University
Curated by ChEMBL
The First Affiliated Hospital Of Dalian Medical University
Curated by ChEMBL
Affinity DataIC50: 22nMAssay Description:Inhibition of recombinant N-terminal GST-tagged human JAK3 (781 to end residues) expressed in baculovirus infected Sf9 insect cells using Poly(4:1 Gl...More data for this Ligand-Target Pair
TargetTyrosine-protein kinase JAK3(Homo sapiens (Human))
The First Affiliated Hospital Of Dalian Medical University
Curated by ChEMBL
The First Affiliated Hospital Of Dalian Medical University
Curated by ChEMBL
Affinity DataIC50: 23nMAssay Description:Inhibition of recombinant N-terminal GST-tagged human JAK3 (781 to end residues) expressed in baculovirus infected Sf9 insect cells using Poly(4:1 Gl...More data for this Ligand-Target Pair
TargetTyrosine-protein kinase BTK(Homo sapiens (Human))
The First Affiliated Hospital Of Dalian Medical University
Curated by ChEMBL
The First Affiliated Hospital Of Dalian Medical University
Curated by ChEMBL
Affinity DataIC50: 31nMAssay Description:Inhibition of recombinant full-length N-terminal His-tagged human BTK expressed in baculovirus infected Sf9 insect cells using Poly(4:1 Glu,Tyr) pept...More data for this Ligand-Target Pair
TargetTyrosine-protein kinase BTK(Homo sapiens (Human))
The First Affiliated Hospital Of Dalian Medical University
Curated by ChEMBL
The First Affiliated Hospital Of Dalian Medical University
Curated by ChEMBL
Affinity DataIC50: 82nMAssay Description:Inhibition of recombinant full-length N-terminal His-tagged human BTK expressed in baculovirus infected Sf9 insect cells using Poly(4:1 Glu,Tyr) pept...More data for this Ligand-Target Pair
TargetTyrosine-protein kinase BTK(Homo sapiens (Human))
The First Affiliated Hospital Of Dalian Medical University
Curated by ChEMBL
The First Affiliated Hospital Of Dalian Medical University
Curated by ChEMBL
Affinity DataIC50: 89nMAssay Description:Inhibition of recombinant full-length N-terminal His-tagged human BTK expressed in baculovirus infected Sf9 insect cells using Poly(4:1 Glu,Tyr) pept...More data for this Ligand-Target Pair
TargetTyrosine-protein kinase BTK(Homo sapiens (Human))
The First Affiliated Hospital Of Dalian Medical University
Curated by ChEMBL
The First Affiliated Hospital Of Dalian Medical University
Curated by ChEMBL
Affinity DataIC50: 90nMAssay Description:Inhibition of recombinant full-length N-terminal His-tagged human BTK expressed in baculovirus infected Sf9 insect cells using Poly(4:1 Glu,Tyr) pept...More data for this Ligand-Target Pair
TargetTyrosine-protein kinase JAK3(Homo sapiens (Human))
The First Affiliated Hospital Of Dalian Medical University
Curated by ChEMBL
The First Affiliated Hospital Of Dalian Medical University
Curated by ChEMBL
Affinity DataIC50: 91nMAssay Description:Inhibition of recombinant N-terminal GST-tagged human JAK3 (781 to end residues) expressed in baculovirus infected Sf9 insect cells using Poly(4:1 Gl...More data for this Ligand-Target Pair
TargetTyrosine-protein kinase JAK3(Homo sapiens (Human))
The First Affiliated Hospital Of Dalian Medical University
Curated by ChEMBL
The First Affiliated Hospital Of Dalian Medical University
Curated by ChEMBL
Affinity DataIC50: >100nMAssay Description:Inhibition of recombinant N-terminal GST-tagged human JAK3 (781 to end residues) expressed in baculovirus infected Sf9 insect cells using Poly(4:1 Gl...More data for this Ligand-Target Pair
TargetTyrosine-protein kinase JAK3(Homo sapiens (Human))
The First Affiliated Hospital Of Dalian Medical University
Curated by ChEMBL
The First Affiliated Hospital Of Dalian Medical University
Curated by ChEMBL
Affinity DataIC50: >100nMAssay Description:Inhibition of recombinant N-terminal GST-tagged human JAK3 (781 to end residues) expressed in baculovirus infected Sf9 insect cells using Poly(4:1 Gl...More data for this Ligand-Target Pair
TargetTyrosine-protein kinase JAK3(Homo sapiens (Human))
The First Affiliated Hospital Of Dalian Medical University
Curated by ChEMBL
The First Affiliated Hospital Of Dalian Medical University
Curated by ChEMBL
Affinity DataIC50: >100nMAssay Description:Inhibition of recombinant N-terminal GST-tagged human JAK3 (781 to end residues) expressed in baculovirus infected Sf9 insect cells using Poly(4:1 Gl...More data for this Ligand-Target Pair
TargetTyrosine-protein kinase BTK(Homo sapiens (Human))
The First Affiliated Hospital Of Dalian Medical University
Curated by ChEMBL
The First Affiliated Hospital Of Dalian Medical University
Curated by ChEMBL
Affinity DataIC50: >100nMAssay Description:Inhibition of recombinant full-length N-terminal His-tagged human BTK expressed in baculovirus infected Sf9 insect cells using Poly(4:1 Glu,Tyr) pept...More data for this Ligand-Target Pair