Compile Data Set for Download or QSAR
maximum 50k data
Found 16 Enz. Inhib. hit(s) with all data for entry = 50010836
TargetHistone deacetylase 2(Homo sapiens (Human))
Khon Kaen University

Curated by ChEMBL
LigandPNGBDBM50542410(CHEMBL4636333)
Affinity DataKi:  550nMAssay Description:Inhibition of HDAC2 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetHistone deacetylase 8(Homo sapiens (Human))
Khon Kaen University

Curated by ChEMBL
LigandPNGBDBM50542410(CHEMBL4636333)
Affinity DataKi:  880nMAssay Description:Inhibition of HDAC8 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetHistone deacetylase 1(Homo sapiens (Human))
Khon Kaen University

Curated by ChEMBL
LigandPNGBDBM50542410(CHEMBL4636333)
Affinity DataKi:  936nMAssay Description:Inhibition of HDAC1 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetHistone deacetylase 2(Homo sapiens (Human))
Khon Kaen University

Curated by ChEMBL
LigandPNGBDBM50542411(CHEMBL4634461)
Affinity DataKi:  1.06E+3nMAssay Description:Inhibition of HDAC2 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetHistone deacetylase 1(Homo sapiens (Human))
Khon Kaen University

Curated by ChEMBL
LigandPNGBDBM50542409(CHEMBL3402858)
Affinity DataKi:  1.96E+3nMAssay Description:Inhibition of HDAC1 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetHistone deacetylase 1(Homo sapiens (Human))
Khon Kaen University

Curated by ChEMBL
LigandPNGBDBM50542411(CHEMBL4634461)
Affinity DataKi:  2.50E+3nMAssay Description:Inhibition of HDAC1 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetHistone deacetylase 8(Homo sapiens (Human))
Khon Kaen University

Curated by ChEMBL
LigandPNGBDBM50542411(CHEMBL4634461)
Affinity DataKi:  3.60E+3nMAssay Description:Inhibition of HDAC8 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetHistone deacetylase 2(Homo sapiens (Human))
Khon Kaen University

Curated by ChEMBL
LigandPNGBDBM50542409(CHEMBL3402858)
Affinity DataKi:  3.99E+3nMAssay Description:Inhibition of HDAC2 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetHistone deacetylase 2(Homo sapiens (Human))
Khon Kaen University

Curated by ChEMBL
LigandPNGBDBM50542408(CHEMBL4634564)
Affinity DataKi:  7.47E+3nMAssay Description:Inhibition of HDAC2 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetHistone deacetylase 8(Homo sapiens (Human))
Khon Kaen University

Curated by ChEMBL
LigandPNGBDBM50542408(CHEMBL4634564)
Affinity DataKi:  1.02E+4nMAssay Description:Inhibition of HDAC8 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetHistone deacetylase 8(Homo sapiens (Human))
Khon Kaen University

Curated by ChEMBL
LigandPNGBDBM50542409(CHEMBL3402858)
Affinity DataKi:  1.42E+4nMAssay Description:Inhibition of HDAC8 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetHistone deacetylase 1(Homo sapiens (Human))
Khon Kaen University

Curated by ChEMBL
LigandPNGBDBM50542408(CHEMBL4634564)
Affinity DataKi:  2.07E+4nMAssay Description:Inhibition of HDAC1 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetHistone deacetylase 1(Homo sapiens (Human))
Khon Kaen University

Curated by ChEMBL
LigandPNGBDBM50140172(CHEBI:3962 | CHEMBL140 | Curcumin | US9409845, Tab...)
Affinity DataKi:  5.08E+4nMAssay Description:Inhibition of HDAC1 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 8(Homo sapiens (Human))
Khon Kaen University

Curated by ChEMBL
LigandPNGBDBM50140172(CHEBI:3962 | CHEMBL140 | Curcumin | US9409845, Tab...)
Affinity DataKi:  6.50E+4nMAssay Description:Inhibition of HDAC8 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase 2(Homo sapiens (Human))
Khon Kaen University

Curated by ChEMBL
LigandPNGBDBM50140172(CHEBI:3962 | CHEMBL140 | Curcumin | US9409845, Tab...)
Affinity DataKi:  9.77E+4nMAssay Description:Inhibition of HDAC2 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone deacetylase(Homo sapiens (Human))
Khon Kaen University

Curated by ChEMBL
LigandPNGBDBM50542407(CHEMBL4634699)
Affinity DataIC50:  7.20E+4nMAssay Description:Inhibition of HDAC in human HeLa cell nuclear extract using fluor-de-lys as substrate by spectrofluorometric analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed