TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Hunan University Of Science And Technology
Curated by ChEMBL
Hunan University Of Science And Technology
Curated by ChEMBL
Affinity DataKi: 0.0160nMAssay Description:Binding affinity to Src (unknown origin) assessed as inhibition constantMore data for this Ligand-Target Pair
TargetSphingosine kinase 2(Homo sapiens (Human))
Hunan University Of Science And Technology
Curated by ChEMBL
Hunan University Of Science And Technology
Curated by ChEMBL
Affinity DataKi: 7.90E+3nMAssay Description:Binding affinity to Sphk2 (unknown origin) assessed as inhibition constantMore data for this Ligand-Target Pair
TargetSphingosine kinase 1(Homo sapiens (Human))
Hunan University Of Science And Technology
Curated by ChEMBL
Hunan University Of Science And Technology
Curated by ChEMBL
Affinity DataKi: 1.60E+4nMAssay Description:Binding affinity to Sphk1 (unknown origin) assessed as inhibition constantMore data for this Ligand-Target Pair
TargetHistone deacetylase(Homo sapiens (Human))
Hunan University Of Science And Technology
Curated by ChEMBL
Hunan University Of Science And Technology
Curated by ChEMBL
Affinity DataIC50: 120nMAssay Description:Inhibition of HDAC in human HeLa nuclear extract measured after 30 mins by fluorescence based assayMore data for this Ligand-Target Pair
TargetHistone deacetylase(Homo sapiens (Human))
Hunan University Of Science And Technology
Curated by ChEMBL
Hunan University Of Science And Technology
Curated by ChEMBL
Affinity DataIC50: 250nMAssay Description:Inhibition of HDAC in human HeLa nuclear extract measured after 30 mins by fluorescence based assayMore data for this Ligand-Target Pair
TargetCyclin-dependent kinase 2(Homo sapiens (Human))
Hunan University Of Science And Technology
Curated by ChEMBL
Hunan University Of Science And Technology
Curated by ChEMBL
Affinity DataIC50: 780nMAssay Description:Inhibition of CDK2 in human A549 cellsMore data for this Ligand-Target Pair
TargetCyclin-dependent kinase 3(Homo sapiens (Human))
Hunan University Of Science And Technology
Curated by ChEMBL
Hunan University Of Science And Technology
Curated by ChEMBL
Affinity DataIC50: 870nMAssay Description:Inhibition of CDK3 in human A549 cellsMore data for this Ligand-Target Pair
TargetCyclin-dependent kinase 1(Homo sapiens (Human))
Hunan University Of Science And Technology
Curated by ChEMBL
Hunan University Of Science And Technology
Curated by ChEMBL
Affinity DataIC50: 1.47E+3nMAssay Description:Inhibition of CDK1 in human A549 cellsMore data for this Ligand-Target Pair