Found 25 Enz. Inhib. hit(s) with all data for entry = 50015492 TargetInduced myeloid leukemia cell differentiation protein Mcl-1(Homo sapiens (Human))
University Of California Riverside
Curated by ChEMBL
University Of California Riverside
Curated by ChEMBL
Affinity DataKi: 17nMAssay Description:Inhibition of human Mcl-1 assessed as inhibition constant by DELFIA displacement assayMore data for this Ligand-Target Pair
TargetInduced myeloid leukemia cell differentiation protein Mcl-1(Homo sapiens (Human))
University Of California Riverside
Curated by ChEMBL
University Of California Riverside
Curated by ChEMBL
Affinity DataKi: 37nMAssay Description:Inhibition of human Mcl-1 assessed as inhibition constant by DELFIA displacement assayMore data for this Ligand-Target Pair
TargetBcl-2-related protein A1(Homo sapiens (Human))
University Of California Riverside
Curated by ChEMBL
University Of California Riverside
Curated by ChEMBL
Affinity DataIC50: 18nMAssay Description:Inhibition of human Bfl-1 (1 to 149 residues) expressed in Rosetta-gami (DE3) using biotinylated-BH3 peptide as substrate measured after 2 hrs by DEL...More data for this Ligand-Target Pair
TargetInduced myeloid leukemia cell differentiation protein Mcl-1(Homo sapiens (Human))
University Of California Riverside
Curated by ChEMBL
University Of California Riverside
Curated by ChEMBL
Affinity DataIC50: 19nMAssay Description:Inhibition of human Mcl-1 (179 to 323 residues) expressed in Escherichia coli BL21 using biotinylated-BH3 peptide as substrate measured after 2 hrs b...More data for this Ligand-Target Pair
TargetInduced myeloid leukemia cell differentiation protein Mcl-1(Homo sapiens (Human))
University Of California Riverside
Curated by ChEMBL
University Of California Riverside
Curated by ChEMBL
Affinity DataIC50: 22nMAssay Description:Inhibition of human Mcl-1 (179 to 323 residues) expressed in Escherichia coli BL21 using biotinylated-BH3 peptide as substrate measured after 2 hrs b...More data for this Ligand-Target Pair
TargetInduced myeloid leukemia cell differentiation protein Mcl-1(Homo sapiens (Human))
University Of California Riverside
Curated by ChEMBL
University Of California Riverside
Curated by ChEMBL
Affinity DataIC50: 23nMAssay Description:Inhibition of human Mcl-1 (179 to 323 residues) expressed in Escherichia coli BL21 using biotinylated-BH3 peptide as substrate measured after 2 hrs b...More data for this Ligand-Target Pair
TargetInduced myeloid leukemia cell differentiation protein Mcl-1(Homo sapiens (Human))
University Of California Riverside
Curated by ChEMBL
University Of California Riverside
Curated by ChEMBL
Affinity DataIC50: 24nMAssay Description:Inhibition of human Mcl-1 (179 to 323 residues) expressed in Escherichia coli BL21 using biotinylated-BH3 peptide as substrate measured after 2 hrs b...More data for this Ligand-Target Pair
TargetInduced myeloid leukemia cell differentiation protein Mcl-1(Homo sapiens (Human))
University Of California Riverside
Curated by ChEMBL
University Of California Riverside
Curated by ChEMBL
Affinity DataIC50: 94nMAssay Description:Inhibition of human Mcl-1 (179 to 323 residues) expressed in Escherichia coli BL21 using biotinylated-BH3 peptide as substrate measured after 2 hrs b...More data for this Ligand-Target Pair
TargetBcl-2-related protein A1(Homo sapiens (Human))
University Of California Riverside
Curated by ChEMBL
University Of California Riverside
Curated by ChEMBL
Affinity DataIC50: >250nMAssay Description:Inhibition of human Bfl-1 (1 to 149 residues) expressed in Rosetta-gami (DE3) using biotinylated-BH3 peptide as substrate measured after 2 hrs by DEL...More data for this Ligand-Target Pair
TargetInduced myeloid leukemia cell differentiation protein Mcl-1(Homo sapiens (Human))
University Of California Riverside
Curated by ChEMBL
University Of California Riverside
Curated by ChEMBL
Affinity DataIC50: 261nMAssay Description:Inhibition of human Mcl-1 (179 to 323 residues) expressed in Escherichia coli BL21 using biotinylated-BH3 peptide as substrate measured after 2 hrs b...More data for this Ligand-Target Pair
TargetInduced myeloid leukemia cell differentiation protein Mcl-1(Homo sapiens (Human))
University Of California Riverside
Curated by ChEMBL
University Of California Riverside
Curated by ChEMBL
Affinity DataIC50: 313nMAssay Description:Inhibition of human Mcl-1 (179 to 323 residues) expressed in Escherichia coli BL21 using biotinylated-BH3 peptide as substrate measured after 2 hrs b...More data for this Ligand-Target Pair
TargetBcl-2-related protein A1(Homo sapiens (Human))
University Of California Riverside
Curated by ChEMBL
University Of California Riverside
Curated by ChEMBL
Affinity DataIC50: >400nMAssay Description:Inhibition of human Bfl-1 (1 to 149 residues) expressed in Rosetta-gami (DE3) using biotinylated-BH3 peptide as substrate measured after 2 hrs by DEL...More data for this Ligand-Target Pair
TargetInduced myeloid leukemia cell differentiation protein Mcl-1(Homo sapiens (Human))
University Of California Riverside
Curated by ChEMBL
University Of California Riverside
Curated by ChEMBL
Affinity DataIC50: 570nMAssay Description:Inhibition of human Mcl-1 (179 to 323 residues) expressed in Escherichia coli BL21 using biotinylated-BH3 peptide as substrate measured after 2 hrs b...More data for this Ligand-Target Pair
TargetBcl-2-related protein A1(Homo sapiens (Human))
University Of California Riverside
Curated by ChEMBL
University Of California Riverside
Curated by ChEMBL
Affinity DataIC50: >1.00E+3nMAssay Description:Inhibition of human Bfl-1 (1 to 149 residues) expressed in Rosetta-gami (DE3) using biotinylated-BH3 peptide as substrate measured after 2 hrs by DEL...More data for this Ligand-Target Pair
TargetInduced myeloid leukemia cell differentiation protein Mcl-1(Homo sapiens (Human))
University Of California Riverside
Curated by ChEMBL
University Of California Riverside
Curated by ChEMBL
Affinity DataIC50: 1.20E+3nMAssay Description:Inhibition of human Mcl-1 (179 to 323 residues) expressed in Escherichia coli BL21 using biotinylated-BH3 peptide as substrate measured after 2 hrs b...More data for this Ligand-Target Pair
TargetInduced myeloid leukemia cell differentiation protein Mcl-1(Homo sapiens (Human))
University Of California Riverside
Curated by ChEMBL
University Of California Riverside
Curated by ChEMBL
Affinity DataIC50: 1.30E+3nMAssay Description:Inhibition of human Mcl-1 (179 to 323 residues) expressed in Escherichia coli BL21 using biotinylated-BH3 peptide as substrate measured after 2 hrs b...More data for this Ligand-Target Pair
TargetInduced myeloid leukemia cell differentiation protein Mcl-1(Homo sapiens (Human))
University Of California Riverside
Curated by ChEMBL
University Of California Riverside
Curated by ChEMBL
Affinity DataIC50: 1.60E+3nMAssay Description:Inhibition of human Mcl-1 (179 to 323 residues) expressed in Escherichia coli BL21 using biotinylated-BH3 peptide as substrate measured after 2 hrs b...More data for this Ligand-Target Pair
TargetInduced myeloid leukemia cell differentiation protein Mcl-1(Homo sapiens (Human))
University Of California Riverside
Curated by ChEMBL
University Of California Riverside
Curated by ChEMBL
Affinity DataIC50: 1.80E+3nMAssay Description:Inhibition of human Mcl-1 (179 to 323 residues) expressed in Escherichia coli BL21 using biotinylated-BH3 peptide as substrate measured after 2 hrs b...More data for this Ligand-Target Pair
TargetInduced myeloid leukemia cell differentiation protein Mcl-1(Homo sapiens (Human))
University Of California Riverside
Curated by ChEMBL
University Of California Riverside
Curated by ChEMBL
Affinity DataIC50: 1.80E+3nMAssay Description:Inhibition of human Mcl-1 (179 to 323 residues) expressed in Escherichia coli BL21 using biotinylated-BH3 peptide as substrate measured after 2 hrs b...More data for this Ligand-Target Pair
TargetInduced myeloid leukemia cell differentiation protein Mcl-1(Homo sapiens (Human))
University Of California Riverside
Curated by ChEMBL
University Of California Riverside
Curated by ChEMBL
Affinity DataIC50: 2.20E+3nMAssay Description:Inhibition of human Mcl-1 (179 to 323 residues) expressed in Escherichia coli BL21 using biotinylated-BH3 peptide as substrate measured after 2 hrs b...More data for this Ligand-Target Pair
TargetInduced myeloid leukemia cell differentiation protein Mcl-1(Homo sapiens (Human))
University Of California Riverside
Curated by ChEMBL
University Of California Riverside
Curated by ChEMBL
Affinity DataIC50: 3.00E+3nMAssay Description:Inhibition of human Mcl-1 (179 to 323 residues) expressed in Escherichia coli BL21 using biotinylated-BH3 peptide as substrate measured after 2 hrs b...More data for this Ligand-Target Pair
TargetInduced myeloid leukemia cell differentiation protein Mcl-1(Homo sapiens (Human))
University Of California Riverside
Curated by ChEMBL
University Of California Riverside
Curated by ChEMBL
Affinity DataIC50: >3.60E+3nMAssay Description:Inhibition of human Mcl-1 (179 to 323 residues) expressed in Escherichia coli BL21 using biotinylated-BH3 peptide as substrate measured after 2 hrs b...More data for this Ligand-Target Pair
TargetBcl-2-related protein A1(Homo sapiens (Human))
University Of California Riverside
Curated by ChEMBL
University Of California Riverside
Curated by ChEMBL
Affinity DataIC50: >5.00E+3nMAssay Description:Inhibition of human Bfl-1 (1 to 149 residues) expressed in Rosetta-gami (DE3) using biotinylated-BH3 peptide as substrate measured after 2 hrs by DEL...More data for this Ligand-Target Pair
TargetBcl-2-related protein A1(Homo sapiens (Human))
University Of California Riverside
Curated by ChEMBL
University Of California Riverside
Curated by ChEMBL
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of human Bfl-1 (1 to 149 residues) expressed in Rosetta-gami (DE3) using biotinylated-BH3 peptide as substrate measured after 2 hrs by DEL...More data for this Ligand-Target Pair
TargetInduced myeloid leukemia cell differentiation protein Mcl-1(Homo sapiens (Human))
University Of California Riverside
Curated by ChEMBL
University Of California Riverside
Curated by ChEMBL
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of human Mcl-1 (179 to 323 residues) expressed in Escherichia coli BL21 using biotinylated-BH3 peptide as substrate measured after 2 hrs b...More data for this Ligand-Target Pair
