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Found 14 Enz. Inhib. hit(s) with all data for entry = 50015663
TargetAmine oxidase [flavin-containing] A(Homo sapiens (Human))
Taipei Medical University

Curated by ChEMBL
LigandPNGBDBM15581(CHEMBL8706 | CLG | CLORGILINE | Clorgyline | N-[3-...)
Affinity DataIC50:  0.610nMAssay Description:Inhibition of human full length recombinant MAO-A expressed in insect cells using kynuramine as substrateMore data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))
Taipei Medical University

Curated by ChEMBL
LigandPNGBDBM50588335(CHEMBL5170163)
Affinity DataIC50:  6.70nMAssay Description:Inhibition of human full length recombinant MAO-B expressed in insect cells using kynuramine as substrateMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
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TargetHistone deacetylase 6(Homo sapiens (Human))
Taipei Medical University

Curated by ChEMBL
LigandPNGBDBM50588334(CHEMBL5171489)
Affinity DataIC50:  20nMAssay Description:Inhibition of human HDAC6 (379 to 382 residues) using RHKKAc as flurogenic substrateMore data for this Ligand-Target Pair
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TargetHistone deacetylase 3(Homo sapiens (Human))
Taipei Medical University

Curated by ChEMBL
LigandPNGBDBM50588334(CHEMBL5171489)
Affinity DataIC50:  133nMAssay Description:Inhibition of human HDAC3 (379 to 382 residues) using RHKKAc as flurogenic substrateMore data for this Ligand-Target Pair
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TargetHistone deacetylase 8(Homo sapiens (Human))
Taipei Medical University

Curated by ChEMBL
LigandPNGBDBM50588334(CHEMBL5171489)
Affinity DataIC50:  210nMAssay Description:Inhibition of human HDAC8 (379 to 382 residues) using RHKAcKAc as flurogenic substrateMore data for this Ligand-Target Pair
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TargetPolyamine deacetylase HDAC10(Homo sapiens (Human))
Taipei Medical University

Curated by ChEMBL
LigandPNGBDBM50588334(CHEMBL5171489)
Affinity DataIC50:  374nMAssay Description:Inhibition of human HDAC10 using Ac-Spermidine-AMC as flurogenic substrateMore data for this Ligand-Target Pair
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TargetHistone deacetylase 1(Homo sapiens (Human))
Taipei Medical University

Curated by ChEMBL
LigandPNGBDBM50588334(CHEMBL5171489)
Affinity DataIC50:  673nMAssay Description:Inhibition of human HDAC1 (379 to 382 residues) using RHKKAc as flurogenic substrateMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetAmine oxidase [flavin-containing] A(Homo sapiens (Human))
Taipei Medical University

Curated by ChEMBL
LigandPNGBDBM50588334(CHEMBL5171489)
Affinity DataIC50:  790nMAssay Description:Inhibition of human full length recombinant MAO-A expressed in insect cells using kynuramine as substrateMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetHistone deacetylase 2(Homo sapiens (Human))
Taipei Medical University

Curated by ChEMBL
LigandPNGBDBM50588334(CHEMBL5171489)
Affinity DataIC50:  1.54E+3nMAssay Description:Inhibition of human HDAC2 (379 to 382 residues) using RHKKAc as flurogenic substrateMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetHistone deacetylase 9(Homo sapiens (Human))
Taipei Medical University

Curated by ChEMBL
LigandPNGBDBM50588334(CHEMBL5171489)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of human HDAC9 using Boc-Lys(trifluoroacetyl)-AMC as flurogenic substrateMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetHistone deacetylase 4(Homo sapiens (Human))
Taipei Medical University

Curated by ChEMBL
LigandPNGBDBM50588334(CHEMBL5171489)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of human HDAC4 using Boc-Lys(trifluoroacetyl)-AMC as flurogenic substrateMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetHistone deacetylase 7(Homo sapiens (Human))
Taipei Medical University

Curated by ChEMBL
LigandPNGBDBM50588334(CHEMBL5171489)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of human HDAC7 using Boc-Lys(trifluoroacetyl)-AMC as flurogenic substrateMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetHistone deacetylase 5(Homo sapiens (Human))
Taipei Medical University

Curated by ChEMBL
LigandPNGBDBM50588334(CHEMBL5171489)
Affinity DataIC50:  1.34E+4nMAssay Description:Inhibition of human HDAC5 using Boc-Lys(trifluoroacetyl)-AMC as flurogenic substrateMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))
Taipei Medical University

Curated by ChEMBL
LigandPNGBDBM50588334(CHEMBL5171489)
Affinity DataIC50:  6.70E+4nMAssay Description:Inhibition of human full length recombinant MAO-B expressed in insect cells using kynuramine as substrateMore data for this Ligand-Target Pair
In DepthDetails PubMed