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Found 3 Enz. Inhib. hit(s) with all data for entry = 50017128
TargetMu-type opioid receptor(Homo sapiens (Human))
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50599918(CHEMBL3736287)
Affinity DataKi:  1nMAssay Description:Binding affinity at MOR (unknown origin) assessed as inhibition constantMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetSubstance-P receptor(Homo sapiens (Human))
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50599918(CHEMBL3736287)
Affinity DataKi:  2.20nMAssay Description:Binding affinity at human NK1R assessed as inhibition constantMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50599918(CHEMBL3736287)
Affinity DataKi:  5nMAssay Description:Binding affinity at DOR (unknown origin) assessed as inhibition constantMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed