Compile Data Set for Download or QSAR
maximum 50k data
Found 63 Enz. Inhib. hit(s) with all data for entry = 50016113
TargetCytochrome P450 2D6(Homo sapiens (Human))
University Of Sharjah

Curated by ChEMBL
LigandPNGBDBM8610(1-[4-(4-{[(2R,4S)-2-(2,4-dichlorophenyl)-2-(1H-imi...)
Affinity DataIC50:  1.90nMAssay Description:Inhibition of CYP2D6 (unknown origin) using EOMCC as a substrateMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
University Of Sharjah

Curated by ChEMBL
LigandPNGBDBM50117930((4-{1-[2-(6-Methyl-pyridin-2-yl)-ethyl]-piperidine...)
Affinity DataIC50:  43nMAssay Description:Inhibition of hERG measured by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetCytochrome P450 3A4(Homo sapiens (Human))
University Of Sharjah

Curated by ChEMBL
LigandPNGBDBM8610(1-[4-(4-{[(2R,4S)-2-(2,4-dichlorophenyl)-2-(1H-imi...)
Affinity DataIC50:  55nMAssay Description:Inhibition of CYP3A4 (unknown origin) using BOMCC as a substrateMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetMitogen-activated protein kinase 10(Homo sapiens (Human))
University Of Sharjah

Curated by ChEMBL
LigandPNGBDBM16018(14,15-diazatetracyclo[7.6.1.0^{2,7}.0^{13,16}]hexa...)
Affinity DataIC50:  91nMAssay Description:Inhibition of JNK3 (unknown origin)More data for this Ligand-Target Pair
TargetMitogen-activated protein kinase 10(Homo sapiens (Human))
University Of Sharjah

Curated by ChEMBL
LigandPNGBDBM50592452(CHEMBL5191468)
Affinity DataIC50:  97nMAssay Description:Inhibition of JNK3 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetMitogen-activated protein kinase 10(Homo sapiens (Human))
University Of Sharjah

Curated by ChEMBL
LigandPNGBDBM50592452(CHEMBL5191468)
Affinity DataIC50:  98nMAssay Description:Inhibition of JNK3 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetMitogen-activated protein kinase 10(Homo sapiens (Human))
University Of Sharjah

Curated by ChEMBL
LigandPNGBDBM50592449(CHEMBL5201911)
Affinity DataIC50:  99nMAssay Description:Inhibition of JNK3 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetMitogen-activated protein kinase 10(Homo sapiens (Human))
University Of Sharjah

Curated by ChEMBL
LigandPNGBDBM50592449(CHEMBL5201911)
Affinity DataIC50:  100nMAssay Description:Inhibition of JNK3 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetMitogen-activated protein kinase 10(Homo sapiens (Human))
University Of Sharjah

Curated by ChEMBL
LigandPNGBDBM50592447(CHEMBL5196004)
Affinity DataIC50:  190nMAssay Description:Inhibition of JNK3 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetMitogen-activated protein kinase 10(Homo sapiens (Human))
University Of Sharjah

Curated by ChEMBL
LigandPNGBDBM50592447(CHEMBL5196004)
Affinity DataIC50:  191nMAssay Description:Inhibition of JNK3 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetMitogen-activated protein kinase 10(Homo sapiens (Human))
University Of Sharjah

Curated by ChEMBL
LigandPNGBDBM50592470(CHEMBL5189795 | US20240002365, Compound CTx-029488...)
Affinity DataIC50:  370nMAssay Description:Inhibition of JNK3 in human HEK293 cells transfected with JNK3-NanoLuc fusion vector measured after 1 hr by NanoBRET assayMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetMitogen-activated protein kinase 10(Homo sapiens (Human))
University Of Sharjah

Curated by ChEMBL
LigandPNGBDBM50592454(CHEMBL5205920)
Affinity DataIC50:  474nMAssay Description:Inhibition of JNK3 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetMitogen-activated protein kinase 10(Homo sapiens (Human))
University Of Sharjah

Curated by ChEMBL
LigandPNGBDBM50592454(CHEMBL5205920)
Affinity DataIC50:  479nMAssay Description:Inhibition of JNK3 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetMitogen-activated protein kinase 10(Homo sapiens (Human))
University Of Sharjah

Curated by ChEMBL
LigandPNGBDBM50592448(CHEMBL5183673)
Affinity DataIC50:  525nMAssay Description:Inhibition of JNK3 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetMitogen-activated protein kinase 10(Homo sapiens (Human))
University Of Sharjah

Curated by ChEMBL
LigandPNGBDBM50592448(CHEMBL5183673)
Affinity DataIC50:  526nMAssay Description:Inhibition of JNK3 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetMitogen-activated protein kinase 10(Homo sapiens (Human))
University Of Sharjah

Curated by ChEMBL
LigandPNGBDBM50592455(CHEMBL5179126)
Affinity DataIC50:  614nMAssay Description:Inhibition of JNK3 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetMitogen-activated protein kinase 10(Homo sapiens (Human))
University Of Sharjah

Curated by ChEMBL
LigandPNGBDBM50592455(CHEMBL5179126)
Affinity DataIC50:  617nMAssay Description:Inhibition of JNK3 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetVascular endothelial growth factor receptor 3(Homo sapiens (Human))
University Of Sharjah

Curated by ChEMBL
LigandPNGBDBM50592452(CHEMBL5191468)
Affinity DataIC50:  791nMAssay Description:Inhibition of FLT4 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetMitogen-activated protein kinase 10(Homo sapiens (Human))
University Of Sharjah

Curated by ChEMBL
LigandPNGBDBM50592464(CHEMBL5199545)
Affinity DataIC50: >1.00E+3nMAssay Description:Inhibition of JNK3 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetMitogen-activated protein kinase 10(Homo sapiens (Human))
University Of Sharjah

Curated by ChEMBL
LigandPNGBDBM50592465(CHEMBL5171564)
Affinity DataIC50: >1.00E+3nMAssay Description:Inhibition of JNK3 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetMitogen-activated protein kinase 10(Homo sapiens (Human))
University Of Sharjah

Curated by ChEMBL
LigandPNGBDBM50592466(CHEMBL5197538)
Affinity DataIC50: >1.00E+3nMAssay Description:Inhibition of JNK3 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetMitogen-activated protein kinase 10(Homo sapiens (Human))
University Of Sharjah

Curated by ChEMBL
LigandPNGBDBM50592467(CHEMBL5174880)
Affinity DataIC50: >1.00E+3nMAssay Description:Inhibition of JNK3 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetMitogen-activated protein kinase 10(Homo sapiens (Human))
University Of Sharjah

Curated by ChEMBL
LigandPNGBDBM50592468(CHEMBL5179338)
Affinity DataIC50: >1.00E+3nMAssay Description:Inhibition of JNK3 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetMitogen-activated protein kinase 10(Homo sapiens (Human))
University Of Sharjah

Curated by ChEMBL
LigandPNGBDBM50592469(CHEMBL5178484)
Affinity DataIC50: >1.00E+3nMAssay Description:Inhibition of JNK3 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetMitogen-activated protein kinase 10(Homo sapiens (Human))
University Of Sharjah

Curated by ChEMBL
LigandPNGBDBM50592457(CHEMBL5182819)
Affinity DataIC50: >1.00E+3nMAssay Description:Inhibition of JNK3 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetMitogen-activated protein kinase 10(Homo sapiens (Human))
University Of Sharjah

Curated by ChEMBL
LigandPNGBDBM50592456(CHEMBL5206891)
Affinity DataIC50: >1.00E+3nMAssay Description:Inhibition of JNK3 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetMitogen-activated protein kinase 10(Homo sapiens (Human))
University Of Sharjah

Curated by ChEMBL
LigandPNGBDBM50592450(CHEMBL5190930)
Affinity DataIC50:  1.00E+3nMAssay Description:Inhibition of JNK3 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetMitogen-activated protein kinase 10(Homo sapiens (Human))
University Of Sharjah

Curated by ChEMBL
LigandPNGBDBM50592451(CHEMBL5190777)
Affinity DataIC50:  1.00E+3nMAssay Description:Inhibition of JNK3 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetMitogen-activated protein kinase 10(Homo sapiens (Human))
University Of Sharjah

Curated by ChEMBL
LigandPNGBDBM50592453(CHEMBL5177988)
Affinity DataIC50:  1.00E+3nMAssay Description:Inhibition of JNK3 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetMitogen-activated protein kinase 10(Homo sapiens (Human))
University Of Sharjah

Curated by ChEMBL
LigandPNGBDBM50592453(CHEMBL5177988)
Affinity DataIC50: >1.00E+3nMAssay Description:Inhibition of JNK3 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetMitogen-activated protein kinase 10(Homo sapiens (Human))
University Of Sharjah

Curated by ChEMBL
LigandPNGBDBM50592456(CHEMBL5206891)
Affinity DataIC50:  1.00E+3nMAssay Description:Inhibition of JNK3 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetMitogen-activated protein kinase 10(Homo sapiens (Human))
University Of Sharjah

Curated by ChEMBL
LigandPNGBDBM50592457(CHEMBL5182819)
Affinity DataIC50:  1.00E+3nMAssay Description:Inhibition of JNK3 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetMitogen-activated protein kinase 10(Homo sapiens (Human))
University Of Sharjah

Curated by ChEMBL
LigandPNGBDBM50592458(CHEMBL5173811)
Affinity DataIC50:  1.00E+3nMAssay Description:Inhibition of JNK3 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetMitogen-activated protein kinase 10(Homo sapiens (Human))
University Of Sharjah

Curated by ChEMBL
LigandPNGBDBM50592459(CHEMBL5190656)
Affinity DataIC50:  1.00E+3nMAssay Description:Inhibition of JNK3 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetMitogen-activated protein kinase 10(Homo sapiens (Human))
University Of Sharjah

Curated by ChEMBL
LigandPNGBDBM50592460(CHEMBL5206209)
Affinity DataIC50:  1.00E+3nMAssay Description:Inhibition of JNK3 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetMitogen-activated protein kinase 10(Homo sapiens (Human))
University Of Sharjah

Curated by ChEMBL
LigandPNGBDBM50592461(CHEMBL5180621)
Affinity DataIC50:  1.00E+3nMAssay Description:Inhibition of JNK3 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetMitogen-activated protein kinase 10(Homo sapiens (Human))
University Of Sharjah

Curated by ChEMBL
LigandPNGBDBM50592462(CHEMBL5176396)
Affinity DataIC50:  1.00E+3nMAssay Description:Inhibition of JNK3 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetMitogen-activated protein kinase 10(Homo sapiens (Human))
University Of Sharjah

Curated by ChEMBL
LigandPNGBDBM50592463(CHEMBL5175285)
Affinity DataIC50:  1.00E+3nMAssay Description:Inhibition of JNK3 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetMitogen-activated protein kinase 10(Homo sapiens (Human))
University Of Sharjah

Curated by ChEMBL
LigandPNGBDBM50592464(CHEMBL5199545)
Affinity DataIC50:  1.00E+3nMAssay Description:Inhibition of JNK3 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetMitogen-activated protein kinase 10(Homo sapiens (Human))
University Of Sharjah

Curated by ChEMBL
LigandPNGBDBM50592465(CHEMBL5171564)
Affinity DataIC50:  1.00E+3nMAssay Description:Inhibition of JNK3 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetMitogen-activated protein kinase 10(Homo sapiens (Human))
University Of Sharjah

Curated by ChEMBL
LigandPNGBDBM50592466(CHEMBL5197538)
Affinity DataIC50:  1.00E+3nMAssay Description:Inhibition of JNK3 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetMitogen-activated protein kinase 10(Homo sapiens (Human))
University Of Sharjah

Curated by ChEMBL
LigandPNGBDBM50592467(CHEMBL5174880)
Affinity DataIC50:  1.00E+3nMAssay Description:Inhibition of JNK3 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetMitogen-activated protein kinase 10(Homo sapiens (Human))
University Of Sharjah

Curated by ChEMBL
LigandPNGBDBM50592468(CHEMBL5179338)
Affinity DataIC50:  1.00E+3nMAssay Description:Inhibition of JNK3 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetMitogen-activated protein kinase 10(Homo sapiens (Human))
University Of Sharjah

Curated by ChEMBL
LigandPNGBDBM50592469(CHEMBL5178484)
Affinity DataIC50:  1.00E+3nMAssay Description:Inhibition of JNK3 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetMitogen-activated protein kinase 8(Homo sapiens (Human))
University Of Sharjah

Curated by ChEMBL
LigandPNGBDBM50592452(CHEMBL5191468)
Affinity DataIC50:  1.00E+3nMAssay Description:Inhibition of JNK1-alpha-1 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetMitogen-activated protein kinase 9(Homo sapiens (Human))
University Of Sharjah

Curated by ChEMBL
LigandPNGBDBM50592452(CHEMBL5191468)
Affinity DataIC50:  1.00E+3nMAssay Description:Inhibition of JNK2-alpha-2 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetPlatelet-derived growth factor receptor alpha(Homo sapiens (Human))
University Of Sharjah

Curated by ChEMBL
LigandPNGBDBM50592449(CHEMBL5201911)
Affinity DataIC50:  1.00E+3nMAssay Description:Inhibition of PDGFRalpha (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetMitogen-activated protein kinase 10(Homo sapiens (Human))
University Of Sharjah

Curated by ChEMBL
LigandPNGBDBM50592463(CHEMBL5175285)
Affinity DataIC50: >1.00E+3nMAssay Description:Inhibition of JNK3 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetMitogen-activated protein kinase 10(Homo sapiens (Human))
University Of Sharjah

Curated by ChEMBL
LigandPNGBDBM50592462(CHEMBL5176396)
Affinity DataIC50: >1.00E+3nMAssay Description:Inhibition of JNK3 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetMitogen-activated protein kinase 10(Homo sapiens (Human))
University Of Sharjah

Curated by ChEMBL
LigandPNGBDBM50592461(CHEMBL5180621)
Affinity DataIC50: >1.00E+3nMAssay Description:Inhibition of JNK3 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
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