Compile Data Set for Download or QSAR
maximum 50k data
Found 74 Enz. Inhib. hit(s) with all data for entry = 50016967
TargetTyrosine-protein kinase JAK3(Homo sapiens (Human))
Jinan University

Curated by ChEMBL
LigandPNGBDBM50598717(CHEMBL5193702 | US20230348487, Example LS 6-45)
Affinity DataIC50:  1.20nMAssay Description:Inhibition of GST tagged recombinant human JAK3 expressed in baculovirus infection system by FRET assayMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetTyrosine-protein kinase JAK3(Homo sapiens (Human))
Jinan University

Curated by ChEMBL
LigandPNGBDBM50598708(CHEMBL5189603 | US20230348487, Example LS 5-77)
Affinity DataIC50:  1.20nMAssay Description:Inhibition of GST tagged recombinant human JAK3 expressed in baculovirus infection system by FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetTyrosine-protein kinase JAK3(Homo sapiens (Human))
Jinan University

Curated by ChEMBL
LigandPNGBDBM50598722(CHEMBL5192736 | US20230348487, Example LS 6-105)
Affinity DataIC50:  1.20nMAssay Description:Inhibition of GST tagged recombinant human JAK3 expressed in baculovirus infection system by FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetTyrosine-protein kinase JAK3(Homo sapiens (Human))
Jinan University

Curated by ChEMBL
LigandPNGBDBM50598720(CHEMBL5201705 | US20230348487, Example LS 6-77)
Affinity DataIC50:  1.30nMAssay Description:Inhibition of GST tagged recombinant human JAK3 expressed in baculovirus infection system by FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetTyrosine-protein kinase JAK3(Homo sapiens (Human))
Jinan University

Curated by ChEMBL
LigandPNGBDBM50598721(CHEMBL5180117 | US20230348487, Example LS 6-88)
Affinity DataIC50:  1.30nMAssay Description:Inhibition of GST tagged recombinant human JAK3 expressed in baculovirus infection system by FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetTyrosine-protein kinase JAK3(Homo sapiens (Human))
Jinan University

Curated by ChEMBL
LigandPNGBDBM50598719(CHEMBL5186937 | US20230348487, Example LS 7-18)
Affinity DataIC50:  1.30nMAssay Description:Inhibition of GST tagged recombinant human JAK3 expressed in baculovirus infection system by FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetTyrosine-protein kinase JAK3(Homo sapiens (Human))
Jinan University

Curated by ChEMBL
LigandPNGBDBM50598718(CHEMBL5176661 | US20230348487, Example LS 7-13)
Affinity DataIC50:  1.30nMAssay Description:Inhibition of GST tagged recombinant human JAK3 expressed in baculovirus infection system by FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetTyrosine-protein kinase JAK3(Homo sapiens (Human))
Jinan University

Curated by ChEMBL
LigandPNGBDBM50598711(CHEMBL5205480 | US20230348487, Example LS 5-152)
Affinity DataIC50:  1.5nMAssay Description:Inhibition of GST tagged recombinant human JAK3 expressed in baculovirus infection system by FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetTyrosine-protein kinase JAK3(Homo sapiens (Human))
Jinan University

Curated by ChEMBL
LigandPNGBDBM50598710(CHEMBL5184187 | US20230348487, Example LS 5-154)
Affinity DataIC50:  1.5nMAssay Description:Inhibition of GST tagged recombinant human JAK3 expressed in baculovirus infection system by FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetTyrosine-protein kinase JAK3(Homo sapiens (Human))
Jinan University

Curated by ChEMBL
LigandPNGBDBM50598712(CHEMBL5182065 | US20230348487, Example LS 5-66)
Affinity DataIC50:  1.60nMAssay Description:Inhibition of GST tagged recombinant human JAK3 expressed in baculovirus infection system by FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetTyrosine-protein kinase JAK3(Homo sapiens (Human))
Jinan University

Curated by ChEMBL
LigandPNGBDBM50598723(CHEMBL5208026)
Affinity DataIC50:  1.70nMAssay Description:Inhibition of GST tagged recombinant human JAK3 expressed in baculovirus infection system by FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetTyrosine-protein kinase JAK3(Homo sapiens (Human))
Jinan University

Curated by ChEMBL
LigandPNGBDBM50598707(CHEMBL5191734 | US20230348487, Example LS 5-12)
Affinity DataIC50:  1.80nMAssay Description:Inhibition of GST tagged recombinant human JAK3 expressed in baculovirus infection system by FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetTyrosine-protein kinase JAK3(Homo sapiens (Human))
Jinan University

Curated by ChEMBL
LigandPNGBDBM50598716(CHEMBL5174210 | US20230348487, Example LS 5-88)
Affinity DataIC50:  1.90nMAssay Description:Inhibition of GST tagged recombinant human JAK3 expressed in baculovirus infection system by FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetTyrosine-protein kinase JAK3(Homo sapiens (Human))
Jinan University

Curated by ChEMBL
LigandPNGBDBM50598715(CHEMBL5190599 | US20230348487, Example LS 5-150)
Affinity DataIC50:  1.90nMAssay Description:Inhibition of GST tagged recombinant human JAK3 expressed in baculovirus infection system by FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetTyrosine-protein kinase JAK1(Homo sapiens (Human))
Jinan University

Curated by ChEMBL
LigandPNGBDBM50193995(3-((3R,4R)-4-methyl-3-(methyl(7H-pyrrolo[2,3-d]pyr...)
Affinity DataIC50:  2.20nMAssay Description:Inhibition of GST-tagged recombinant human JAK1 (866 to 1154 residues) expressed in baculovirus infection system by FRET assayMore data for this Ligand-Target Pair
TargetTyrosine-protein kinase JAK3(Homo sapiens (Human))
Jinan University

Curated by ChEMBL
LigandPNGBDBM50598714(CHEMBL5184019 | US20230348487, Example LS 5-143)
Affinity DataIC50:  2.20nMAssay Description:Inhibition of GST tagged recombinant human JAK3 expressed in baculovirus infection system by FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetTyrosine-protein kinase JAK3(Homo sapiens (Human))
Jinan University

Curated by ChEMBL
LigandPNGBDBM209866(PF-06651600 | US11111242, Example 5 | US2023034848...)
Affinity DataIC50:  2.30nMAssay Description:Inhibition of GST tagged recombinant human JAK3 expressed in baculovirus infection system by FRET assayMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetTyrosine-protein kinase JAK3(Homo sapiens (Human))
Jinan University

Curated by ChEMBL
LigandPNGBDBM50598713(CHEMBL5185016 | US20230348487, Example LS 5-102)
Affinity DataIC50:  2.5nMAssay Description:Inhibition of GST tagged recombinant human JAK3 expressed in baculovirus infection system by FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetTyrosine-protein kinase JAK3(Homo sapiens (Human))
Jinan University

Curated by ChEMBL
LigandPNGBDBM50598709(CHEMBL5207354 | US20230348487, Example LS 5-91)
Affinity DataIC50:  5.5nMAssay Description:Inhibition of GST tagged recombinant human JAK3 expressed in baculovirus infection system by FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetTyrosine-protein kinase JAK3(Homo sapiens (Human))
Jinan University

Curated by ChEMBL
LigandPNGBDBM50193995(3-((3R,4R)-4-methyl-3-(methyl(7H-pyrrolo[2,3-d]pyr...)
Affinity DataIC50:  6.70nMAssay Description:Inhibition of GST tagged recombinant human JAK3 expressed in baculovirus infection system by FRET assayMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetTyrosine-protein kinase JAK3(Homo sapiens (Human))
Jinan University

Curated by ChEMBL
LigandPNGBDBM50598717(CHEMBL5193702 | US20230348487, Example LS 6-45)
Affinity DataIC50:  8nMAssay Description:Inhibition of human JAK3More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetTyrosine-protein kinase JAK3(Homo sapiens (Human))
Jinan University

Curated by ChEMBL
LigandPNGBDBM50598706(CHEMBL5185440 | US20230348487, Example LS 4-104)
Affinity DataIC50:  18nMAssay Description:Inhibition of GST tagged recombinant human JAK3 expressed in baculovirus infection system by FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetNUAK family SNF1-like kinase 1(Homo sapiens (Human))
Jinan University

Curated by ChEMBL
LigandPNGBDBM50598717(CHEMBL5193702 | US20230348487, Example LS 6-45)
Affinity DataIC50:  25nMAssay Description:Inhibition of human ARK5More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetTyrosine-protein kinase JAK2(Homo sapiens (Human))
Jinan University

Curated by ChEMBL
LigandPNGBDBM50193995(3-((3R,4R)-4-methyl-3-(methyl(7H-pyrrolo[2,3-d]pyr...)
Affinity DataIC50:  26nMAssay Description:Inhibition of GST tagged recombinant human JAK2 expressed in baculovirus infection system by FRET assayMore data for this Ligand-Target Pair
TargetTyrosine-protein kinase JAK3(Homo sapiens (Human))
Jinan University

Curated by ChEMBL
LigandPNGBDBM50598705(CHEMBL5182374)
Affinity DataIC50:  32nMAssay Description:Inhibition of GST tagged recombinant human JAK3 expressed in baculovirus infection system by FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetNon-receptor tyrosine-protein kinase TYK2(Homo sapiens (Human))
Jinan University

Curated by ChEMBL
LigandPNGBDBM50598708(CHEMBL5189603 | US20230348487, Example LS 5-77)
Affinity DataIC50:  94nMAssay Description:Inhibition of human TYK2 by FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetNon-receptor tyrosine-protein kinase TYK2(Homo sapiens (Human))
Jinan University

Curated by ChEMBL
LigandPNGBDBM50193995(3-((3R,4R)-4-methyl-3-(methyl(7H-pyrrolo[2,3-d]pyr...)
Affinity DataIC50:  112nMAssay Description:Inhibition of human TYK2 by FRET assayMore data for this Ligand-Target Pair
TargetReceptor-type tyrosine-protein kinase FLT3(Homo sapiens (Human))
Jinan University

Curated by ChEMBL
LigandPNGBDBM50598717(CHEMBL5193702 | US20230348487, Example LS 6-45)
Affinity DataIC50:  132nMAssay Description:Inhibition of human FLT3More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetCyclin-Y/Cyclin-dependent kinase 16(Homo sapiens (Human))
Jinan University

Curated by ChEMBL
LigandPNGBDBM50598717(CHEMBL5193702 | US20230348487, Example LS 6-45)
Affinity DataIC50:  135nMAssay Description:Inhibition of human CDK16/cyclin-Y protein-protein complexMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetNon-receptor tyrosine-protein kinase TYK2(Homo sapiens (Human))
Jinan University

Curated by ChEMBL
LigandPNGBDBM50598711(CHEMBL5205480 | US20230348487, Example LS 5-152)
Affinity DataIC50:  148nMAssay Description:Inhibition of human TYK2 by FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetNon-receptor tyrosine-protein kinase TYK2(Homo sapiens (Human))
Jinan University

Curated by ChEMBL
LigandPNGBDBM50598706(CHEMBL5185440 | US20230348487, Example LS 4-104)
Affinity DataIC50:  150nMAssay Description:Inhibition of human TYK2 by FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetNon-receptor tyrosine-protein kinase TYK2(Homo sapiens (Human))
Jinan University

Curated by ChEMBL
LigandPNGBDBM50598714(CHEMBL5184019 | US20230348487, Example LS 5-143)
Affinity DataIC50:  166nMAssay Description:Inhibition of human TYK2 by FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetNon-receptor tyrosine-protein kinase TYK2(Homo sapiens (Human))
Jinan University

Curated by ChEMBL
LigandPNGBDBM50598705(CHEMBL5182374)
Affinity DataIC50:  170nMAssay Description:Inhibition of human TYK2 by FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetNon-receptor tyrosine-protein kinase TYK2(Homo sapiens (Human))
Jinan University

Curated by ChEMBL
LigandPNGBDBM50598715(CHEMBL5190599 | US20230348487, Example LS 5-150)
Affinity DataIC50:  186nMAssay Description:Inhibition of human TYK2 by FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetNon-receptor tyrosine-protein kinase TYK2(Homo sapiens (Human))
Jinan University

Curated by ChEMBL
LigandPNGBDBM50598710(CHEMBL5184187 | US20230348487, Example LS 5-154)
Affinity DataIC50:  187nMAssay Description:Inhibition of human TYK2 by FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetTyrosine-protein kinase JAK1(Homo sapiens (Human))
Jinan University

Curated by ChEMBL
LigandPNGBDBM50598711(CHEMBL5205480 | US20230348487, Example LS 5-152)
Affinity DataIC50:  190nMAssay Description:Inhibition of GST-tagged recombinant human JAK1 (866 to 1154 residues) expressed in baculovirus infection system by FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetNon-receptor tyrosine-protein kinase TYK2(Homo sapiens (Human))
Jinan University

Curated by ChEMBL
LigandPNGBDBM50598709(CHEMBL5207354 | US20230348487, Example LS 5-91)
Affinity DataIC50:  233nMAssay Description:Inhibition of human TYK2 by FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetNon-receptor tyrosine-protein kinase TYK2(Homo sapiens (Human))
Jinan University

Curated by ChEMBL
LigandPNGBDBM50598713(CHEMBL5185016 | US20230348487, Example LS 5-102)
Affinity DataIC50:  241nMAssay Description:Inhibition of human TYK2 by FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetTyrosine-protein kinase JAK3(Homo sapiens (Human))
Jinan University

Curated by ChEMBL
LigandPNGBDBM50598704(CHEMBL5203904 | US20230348487, Example LS 3-96)
Affinity DataIC50:  268nMAssay Description:Inhibition of GST tagged recombinant human JAK3 expressed in baculovirus infection system by FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetTyrosine-protein kinase JAK1(Homo sapiens (Human))
Jinan University

Curated by ChEMBL
LigandPNGBDBM50598715(CHEMBL5190599 | US20230348487, Example LS 5-150)
Affinity DataIC50:  270nMAssay Description:Inhibition of GST-tagged recombinant human JAK1 (866 to 1154 residues) expressed in baculovirus infection system by FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetTyrosine-protein kinase JAK2(Homo sapiens (Human))
Jinan University

Curated by ChEMBL
LigandPNGBDBM50598706(CHEMBL5185440 | US20230348487, Example LS 4-104)
Affinity DataIC50:  290nMAssay Description:Inhibition of GST tagged recombinant human JAK2 expressed in baculovirus infection system by FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetNon-receptor tyrosine-protein kinase TYK2(Homo sapiens (Human))
Jinan University

Curated by ChEMBL
LigandPNGBDBM50598712(CHEMBL5182065 | US20230348487, Example LS 5-66)
Affinity DataIC50:  335nMAssay Description:Inhibition of human TYK2 by FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetTyrosine-protein kinase JAK2(Homo sapiens (Human))
Jinan University

Curated by ChEMBL
LigandPNGBDBM50598711(CHEMBL5205480 | US20230348487, Example LS 5-152)
Affinity DataIC50:  357nMAssay Description:Inhibition of GST tagged recombinant human JAK2 expressed in baculovirus infection system by FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetTyrosine-protein kinase JAK2(Homo sapiens (Human))
Jinan University

Curated by ChEMBL
LigandPNGBDBM50598714(CHEMBL5184019 | US20230348487, Example LS 5-143)
Affinity DataIC50:  362nMAssay Description:Inhibition of GST tagged recombinant human JAK2 expressed in baculovirus infection system by FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetNon-receptor tyrosine-protein kinase TYK2(Homo sapiens (Human))
Jinan University

Curated by ChEMBL
LigandPNGBDBM50598717(CHEMBL5193702 | US20230348487, Example LS 6-45)
Affinity DataIC50:  365nMAssay Description:Inhibition of human TYK2More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetNon-receptor tyrosine-protein kinase TYK2(Homo sapiens (Human))
Jinan University

Curated by ChEMBL
LigandPNGBDBM50598707(CHEMBL5191734 | US20230348487, Example LS 5-12)
Affinity DataIC50:  369nMAssay Description:Inhibition of human TYK2 by FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetTyrosine-protein kinase JAK2(Homo sapiens (Human))
Jinan University

Curated by ChEMBL
LigandPNGBDBM50598705(CHEMBL5182374)
Affinity DataIC50:  410nMAssay Description:Inhibition of GST tagged recombinant human JAK2 expressed in baculovirus infection system by FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetNon-receptor tyrosine-protein kinase TYK2(Homo sapiens (Human))
Jinan University

Curated by ChEMBL
LigandPNGBDBM50598716(CHEMBL5174210 | US20230348487, Example LS 5-88)
Affinity DataIC50:  424nMAssay Description:Inhibition of human TYK2 by FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetTyrosine-protein kinase JAK2(Homo sapiens (Human))
Jinan University

Curated by ChEMBL
LigandPNGBDBM50598713(CHEMBL5185016 | US20230348487, Example LS 5-102)
Affinity DataIC50:  437nMAssay Description:Inhibition of GST tagged recombinant human JAK2 expressed in baculovirus infection system by FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetTyrosine-protein kinase JAK1(Homo sapiens (Human))
Jinan University

Curated by ChEMBL
LigandPNGBDBM50598714(CHEMBL5184019 | US20230348487, Example LS 5-143)
Affinity DataIC50:  481nMAssay Description:Inhibition of GST-tagged recombinant human JAK1 (866 to 1154 residues) expressed in baculovirus infection system by FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
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