Compile Data Set for Download or QSAR
Report error Found 5 Enz. Inhib. hit(s) with all data for entry = 50022224
TargetNuclear factor erythroid 2-related factor 2(Human)
Nanjing University of Chinese Medicine

Curated by ChEMBL
LigandPNGBDBM50649618(Halofuginone | Halofuginona | Halofuginon | Ht-100...)
Affinity DataIC50: 22nMAssay Description:Inhibition of NRF2 in human KYSE-70 cellsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/13/2025
Entry Details
PubMed
TargetNuclear factor erythroid 2-related factor 2(Human)
Nanjing University of Chinese Medicine

Curated by ChEMBL
LigandPNGBDBM50649618(Halofuginone | Halofuginona | Halofuginon | Ht-100...)
Affinity DataIC50: 37nMAssay Description:Inhibition of NRF2 in human A549 cellsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/13/2025
Entry Details
PubMed
TargetNuclear factor erythroid 2-related factor 2(Human)
Nanjing University of Chinese Medicine

Curated by ChEMBL
LigandPNGBDBM50649619(CHEMBL5619820)
Affinity DataKd:  1.20E+3nMAssay Description:Binding affinity to NRF2 (unknown origin) using dsDNA as substrate assessed as dissociation constant incubated for 60 mins by FP assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/13/2025
Entry Details
PubMed
TargetTranscription factor MafG(Homo sapiens)
Nanjing University of Chinese Medicine

Curated by ChEMBL
LigandPNGBDBM50649616(CHEMBL1479098)
Affinity DataIC50: 1.90E+3nMAssay Description:Inhibition of NRF2/MAFG (unknown origin) heterodimerization using fluorescein-labeled ARE DNA duplex as substrate preincubated for 1 hr followed by s...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/13/2025
Entry Details
PubMed
TargetNuclear factor erythroid 2-related factor 2(Human)
Nanjing University of Chinese Medicine

Curated by ChEMBL
LigandPNGBDBM50649617(CHEMBL5619019)
Affinity DataIC50: 2.90E+3nMAssay Description:Inhibition of NRF2 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In Depth
Date in BDB:
10/13/2025
Entry Details
PubMed