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Found 13 Enz. Inhib. hit(s) with all data for entry = 50029076
TargetPlatelet-activating factor receptor(Cavia porcellus)
TBA

Curated by ChEMBL
LigandPNGBDBM50038774((R)-2-Pyridin-3-yl-thiazolidine-4-carboxylic acid ...)
Affinity DataKi:  5nMAssay Description:Inhibition of [3H]-PAF binding to rabbit platelet membranesMore data for this Ligand-Target Pair
In DepthDetails Article
TargetPlatelet-activating factor receptor(Cavia porcellus)
TBA

Curated by ChEMBL
LigandPNGBDBM50281212((1S,5R,7aR)-3-Oxo-5-pyridin-3-yl-dihydro-thiazolo[...)
Affinity DataKi:  24nMAssay Description:Inhibition of [3H]-PAF binding to rabbit platelet membranesMore data for this Ligand-Target Pair
In DepthDetails Article
TargetPlatelet-activating factor receptor(Cavia porcellus)
TBA

Curated by ChEMBL
LigandPNGBDBM50281213((1S,5S,7aR)-3-Oxo-5-pyridin-3-yl-dihydro-thiazolo[...)
Affinity DataKi:  150nMAssay Description:Inhibition of [3H]-PAF binding to rabbit platelet membranesMore data for this Ligand-Target Pair
In DepthDetails Article
TargetPlatelet-activating factor receptor(Cavia porcellus)
TBA

Curated by ChEMBL
LigandPNGBDBM50281215((3R,7S,7aR)-5-Oxo-3-pyridin-3-yl-tetrahydro-pyrrol...)
Affinity DataKi:  540nMAssay Description:Inhibition of [3H]-PAF binding to rabbit platelet membranesMore data for this Ligand-Target Pair
In DepthDetails Article
TargetPlatelet-activating factor receptor(Cavia porcellus)
TBA

Curated by ChEMBL
LigandPNGBDBM50281209((3S,7S,7aR)-5-Oxo-3-pyridin-3-yl-tetrahydro-pyrrol...)
Affinity DataKi:  600nMAssay Description:Inhibition of [3H]-PAF binding to rabbit platelet membranesMore data for this Ligand-Target Pair
In DepthDetails Article
TargetPlatelet-activating factor receptor(Cavia porcellus)
TBA

Curated by ChEMBL
LigandPNGBDBM50281214((3S,7R,7aR)-5-Oxo-3-pyridin-3-yl-tetrahydro-pyrrol...)
Affinity DataKi:  1.00E+3nMAssay Description:Inhibition of [3H]-PAF binding to rabbit platelet membranesMore data for this Ligand-Target Pair
In DepthDetails Article
TargetPlatelet-activating factor receptor(Cavia porcellus)
TBA

Curated by ChEMBL
LigandPNGBDBM50281216((1R,5R,7aR)-3-Oxo-5-pyridin-3-yl-dihydro-thiazolo[...)
Affinity DataKi:  1.20E+3nMAssay Description:Inhibition of [3H]-PAF binding to rabbit platelet membranesMore data for this Ligand-Target Pair
In DepthDetails Article
TargetPlatelet-activating factor receptor(Cavia porcellus)
TBA

Curated by ChEMBL
LigandPNGBDBM50281210((3R,7S,7aR)-6-Methyl-5-oxo-3-pyridin-3-yl-tetrahyd...)
Affinity DataKi:  1.45E+3nMAssay Description:Inhibition of [3H]-PAF binding to rabbit platelet membranesMore data for this Ligand-Target Pair
In DepthDetails Article
TargetPlatelet-activating factor receptor(Cavia porcellus)
TBA

Curated by ChEMBL
LigandPNGBDBM50281218((3R,7R,7aR)-5-Oxo-3-pyridin-3-yl-tetrahydro-pyrrol...)
Affinity DataKi:  1.80E+3nMAssay Description:Inhibition of [3H]-PAF binding to rabbit platelet membranesMore data for this Ligand-Target Pair
In DepthDetails Article
TargetPlatelet-activating factor receptor(Cavia porcellus)
TBA

Curated by ChEMBL
LigandPNGBDBM50281217((3S,7S,7aR)-6-Methyl-5-oxo-3-pyridin-3-yl-tetrahyd...)
Affinity DataKi:  2.20E+3nMAssay Description:Inhibition of [3H]-PAF binding to rabbit platelet membranesMore data for this Ligand-Target Pair
In DepthDetails Article
TargetPlatelet-activating factor receptor(Cavia porcellus)
TBA

Curated by ChEMBL
LigandPNGBDBM50281219((1R,5S,7aR)-3-Oxo-5-pyridin-3-yl-dihydro-thiazolo[...)
Affinity DataKi:  2.50E+3nMAssay Description:Inhibition of [3H]-PAF binding to rabbit platelet membranesMore data for this Ligand-Target Pair
In DepthDetails Article
TargetPlatelet-activating factor receptor(Cavia porcellus)
TBA

Curated by ChEMBL
LigandPNGBDBM50281220((3S,7R,7aR)-6-Methyl-5-oxo-3-pyridin-3-yl-tetrahyd...)
Affinity DataKi:  1.40E+4nMAssay Description:Inhibition of [3H]-PAF binding to rabbit platelet membranesMore data for this Ligand-Target Pair
In DepthDetails Article
TargetPlatelet-activating factor receptor(Cavia porcellus)
TBA

Curated by ChEMBL
LigandPNGBDBM50281211((3R,7R,7aR)-6-Methyl-5-oxo-3-pyridin-3-yl-tetrahyd...)
Affinity DataKi:  9.50E+4nMAssay Description:Inhibition of [3H]-PAF binding to rabbit platelet membranesMore data for this Ligand-Target Pair
In DepthDetails Article