Compile Data Set for Download or QSAR
maximum 50k data
Found 39 Enz. Inhib. hit(s) with all data for entry = 50029323
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50283398((1-Benzyl-piperidin-4-yl)-(3-phenyl-prop-2-ynyl)-a...)
Affinity DataKi:  2.5nMAssay Description:Inhibiton of [3H]-(+)-SKF-10,047 binding to sigma receptorMore data for this Ligand-Target Pair
In DepthDetails Article
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50283400((1-Benzyl-piperidin-4-yl)-methyl-((E)-3-phenyl-all...)
Affinity DataKi:  2.60nMAssay Description:Inhibiton of [3H]-(+)-SKF-10,047 binding to sigma receptorMore data for this Ligand-Target Pair
In DepthDetails Article
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50283402(3-Phenyl-propynoic acid (1-benzyl-piperidin-4-yl)-...)
Affinity DataKi:  4nMAssay Description:Inhibiton of [3H]-(+)-SKF-10,047 binding to sigma receptorMore data for this Ligand-Target Pair
In DepthDetails Article
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50283395((E)-N-(1-Benzyl-piperidin-4-yl)-N-methyl-3-phenyl-...)
Affinity DataKi:  5nMAssay Description:Inhibiton of [3H]-(+)-SKF-10,047 binding to sigma receptorMore data for this Ligand-Target Pair
In DepthDetails Article
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50283405((1-Benzyl-piperidin-4-yl)-methyl-(3-phenyl-prop-2-...)
Affinity DataKi:  5nMAssay Description:Inhibiton of [3H]-(+)-SKF-10,047 binding to sigma receptorMore data for this Ligand-Target Pair
In DepthDetails Article
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50283399(3-Phenyl-propynoic acid (1-benzyl-piperidin-4-yl)-...)
Affinity DataKi:  6nMAssay Description:Inhibiton of [3H]-(+)-SKF-10,047 binding to sigma receptorMore data for this Ligand-Target Pair
In DepthDetails Article
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50283396((1-Benzyl-piperidin-4-yl)-bis-((E)-3-phenyl-allyl)...)
Affinity DataKi:  7nMAssay Description:Inhibiton of [3H]-(+)-SKF-10,047 binding to sigma receptorMore data for this Ligand-Target Pair
In DepthDetails Article
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50283393(3-Phenyl-propynoic acid (1-benzyl-piperidin-4-yl)-...)
Affinity DataKi:  8nMAssay Description:Inhibiton of [3H]-(+)-SKF-10,047 binding to sigma receptorMore data for this Ligand-Target Pair
In DepthDetails Article
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50283394((E)-N-(1-Benzyl-piperidin-4-yl)-3-phenyl-acrylamid...)
Affinity DataKi:  15nMAssay Description:Inhibiton of [3H]-(+)-SKF-10,047 binding to sigma receptorMore data for this Ligand-Target Pair
In DepthDetails Article
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50283403((1-Benzyl-piperidin-4-yl)-((E)-3-phenyl-allyl)-ami...)
Affinity DataKi:  16nMAssay Description:Inhibiton of [3H]-(+)-SKF-10,047 binding to sigma receptorMore data for this Ligand-Target Pair
In DepthDetails Article
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50283404((1-Benzyl-piperidin-4-yl)-phenyl-(3-phenyl-prop-2-...)
Affinity DataKi:  22nMAssay Description:Inhibiton of [3H]-(+)-SKF-10,047 binding to sigma receptorMore data for this Ligand-Target Pair
In DepthDetails Article
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50283397((E)-N-(1-Benzyl-piperidin-4-yl)-3,N-diphenyl-acryl...)
Affinity DataKi:  58nMAssay Description:Inhibiton of [3H]-(+)-SKF-10,047 binding to sigma receptorMore data for this Ligand-Target Pair
In DepthDetails Article
TargetSerotonin 2 (5-HT2) receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50283394((E)-N-(1-Benzyl-piperidin-4-yl)-3-phenyl-acrylamid...)
Affinity DataKi:  100nMAssay Description:Displacement of [3H]ketanserin from 5-hydroxytryptamine 2 receptorMore data for this Ligand-Target Pair
In DepthDetails Article
TargetSerotonin 2 (5-HT2) receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50283404((1-Benzyl-piperidin-4-yl)-phenyl-(3-phenyl-prop-2-...)
Affinity DataKi:  280nMAssay Description:Displacement of [3H]ketanserin from 5-hydroxytryptamine 2 receptorMore data for this Ligand-Target Pair
In DepthDetails Article
TargetSerotonin 2 (5-HT2) receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50283393(3-Phenyl-propynoic acid (1-benzyl-piperidin-4-yl)-...)
Affinity DataKi:  280nMAssay Description:Displacement of [3H]ketanserin from 5-hydroxytryptamine 2 receptorMore data for this Ligand-Target Pair
In DepthDetails Article
TargetSerotonin 2 (5-HT2) receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50283405((1-Benzyl-piperidin-4-yl)-methyl-(3-phenyl-prop-2-...)
Affinity DataKi:  320nMAssay Description:Displacement of [3H]ketanserin from 5-hydroxytryptamine 2 receptorMore data for this Ligand-Target Pair
In DepthDetails Article
TargetSerotonin 2 (5-HT2) receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50283396((1-Benzyl-piperidin-4-yl)-bis-((E)-3-phenyl-allyl)...)
Affinity DataKi:  550nMAssay Description:Displacement of [3H]ketanserin from 5-hydroxytryptamine 2 receptorMore data for this Ligand-Target Pair
In DepthDetails Article
TargetSerotonin 2 (5-HT2) receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50283400((1-Benzyl-piperidin-4-yl)-methyl-((E)-3-phenyl-all...)
Affinity DataKi:  840nMAssay Description:Displacement of [3H]ketanserin from 5-hydroxytryptamine 2 receptorMore data for this Ligand-Target Pair
In DepthDetails Article
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50283401((1-Benzyl-piperidin-4-yl)-phenyl-((E)-3-phenyl-all...)
Affinity DataKi:  1.50E+3nMAssay Description:Inhibiton of [3H]-(+)-SKF-10,047 binding to sigma receptorMore data for this Ligand-Target Pair
In DepthDetails Article
TargetSerotonin 2 (5-HT2) receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50283395((E)-N-(1-Benzyl-piperidin-4-yl)-N-methyl-3-phenyl-...)
Affinity DataKi:  1.50E+3nMAssay Description:Displacement of [3H]ketanserin from 5-hydroxytryptamine 2 receptorMore data for this Ligand-Target Pair
In DepthDetails Article
TargetSerotonin 2 (5-HT2) receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50283402(3-Phenyl-propynoic acid (1-benzyl-piperidin-4-yl)-...)
Affinity DataKi:  1.70E+3nMAssay Description:Displacement of [3H]ketanserin from 5-hydroxytryptamine 2 receptorMore data for this Ligand-Target Pair
In DepthDetails Article
TargetSerotonin 2 (5-HT2) receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50283399(3-Phenyl-propynoic acid (1-benzyl-piperidin-4-yl)-...)
Affinity DataKi:  3.10E+3nMAssay Description:Displacement of [3H]ketanserin from 5-hydroxytryptamine 2 receptorMore data for this Ligand-Target Pair
In DepthDetails Article
TargetSerotonin 2 (5-HT2) receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50283398((1-Benzyl-piperidin-4-yl)-(3-phenyl-prop-2-ynyl)-a...)
Affinity DataKi:  3.30E+3nMAssay Description:Displacement of [3H]ketanserin from 5-hydroxytryptamine 2 receptorMore data for this Ligand-Target Pair
In DepthDetails Article
TargetSerotonin 2 (5-HT2) receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50283397((E)-N-(1-Benzyl-piperidin-4-yl)-3,N-diphenyl-acryl...)
Affinity DataKi:  4.20E+3nMAssay Description:Displacement of [3H]ketanserin from 5-hydroxytryptamine 2 receptorMore data for this Ligand-Target Pair
In DepthDetails Article
TargetSerotonin 2 (5-HT2) receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50283403((1-Benzyl-piperidin-4-yl)-((E)-3-phenyl-allyl)-ami...)
Affinity DataKi:  4.60E+3nMAssay Description:Displacement of [3H]ketanserin from 5-hydroxytryptamine 2 receptorMore data for this Ligand-Target Pair
In DepthDetails Article
TargetSerotonin 2 (5-HT2) receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50283401((1-Benzyl-piperidin-4-yl)-phenyl-((E)-3-phenyl-all...)
Affinity DataKi: >1.00E+4nMAssay Description:Displacement of [3H]ketanserin from 5-hydroxytryptamine 2 receptorMore data for this Ligand-Target Pair
In DepthDetails Article
TargetD(2) dopamine receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50283404((1-Benzyl-piperidin-4-yl)-phenyl-(3-phenyl-prop-2-...)
Affinity DataIC50:  890nMAssay Description:Displacement of [3H]-spiperone from dopamine D2 receptorMore data for this Ligand-Target Pair
In DepthDetails Article
TargetD(2) dopamine receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50283399(3-Phenyl-propynoic acid (1-benzyl-piperidin-4-yl)-...)
Affinity DataIC50:  1.50E+3nMAssay Description:Displacement of [3H]-spiperone from dopamine D2 receptorMore data for this Ligand-Target Pair
In DepthDetails Article
TargetD(2) dopamine receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50283393(3-Phenyl-propynoic acid (1-benzyl-piperidin-4-yl)-...)
Affinity DataIC50:  2.50E+3nMAssay Description:Displacement of [3H]-spiperone from dopamine D2 receptorMore data for this Ligand-Target Pair
In DepthDetails Article
TargetD(2) dopamine receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50283405((1-Benzyl-piperidin-4-yl)-methyl-(3-phenyl-prop-2-...)
Affinity DataIC50:  4.10E+3nMAssay Description:Displacement of [3H]-spiperone from dopamine D2 receptorMore data for this Ligand-Target Pair
In DepthDetails Article
TargetD(2) dopamine receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50283394((E)-N-(1-Benzyl-piperidin-4-yl)-3-phenyl-acrylamid...)
Affinity DataIC50:  4.70E+3nMAssay Description:Displacement of [3H]-spiperone from dopamine D2 receptorMore data for this Ligand-Target Pair
In DepthDetails Article
TargetD(2) dopamine receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50283402(3-Phenyl-propynoic acid (1-benzyl-piperidin-4-yl)-...)
Affinity DataIC50:  4.90E+3nMAssay Description:Displacement of [3H]-spiperone from dopamine D2 receptorMore data for this Ligand-Target Pair
In DepthDetails Article
TargetD(2) dopamine receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50283395((E)-N-(1-Benzyl-piperidin-4-yl)-N-methyl-3-phenyl-...)
Affinity DataIC50:  7.10E+3nMAssay Description:Displacement of [3H]-spiperone from dopamine D2 receptorMore data for this Ligand-Target Pair
In DepthDetails Article
TargetD(2) dopamine receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50283397((E)-N-(1-Benzyl-piperidin-4-yl)-3,N-diphenyl-acryl...)
Affinity DataIC50: >1.00E+4nMAssay Description:Displacement of [3H]-spiperone from dopamine D2 receptorMore data for this Ligand-Target Pair
In DepthDetails Article
TargetD(2) dopamine receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50283400((1-Benzyl-piperidin-4-yl)-methyl-((E)-3-phenyl-all...)
Affinity DataIC50: >1.00E+4nMAssay Description:Displacement of [3H]-spiperone from dopamine D2 receptorMore data for this Ligand-Target Pair
In DepthDetails Article
TargetD(2) dopamine receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50283396((1-Benzyl-piperidin-4-yl)-bis-((E)-3-phenyl-allyl)...)
Affinity DataIC50: >1.00E+4nMAssay Description:Displacement of [3H]-spiperone from dopamine D2 receptorMore data for this Ligand-Target Pair
In DepthDetails Article
TargetD(2) dopamine receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50283403((1-Benzyl-piperidin-4-yl)-((E)-3-phenyl-allyl)-ami...)
Affinity DataIC50: >1.00E+4nMAssay Description:Displacement of [3H]-spiperone from dopamine D2 receptorMore data for this Ligand-Target Pair
In DepthDetails Article
TargetD(2) dopamine receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50283398((1-Benzyl-piperidin-4-yl)-(3-phenyl-prop-2-ynyl)-a...)
Affinity DataIC50: >1.00E+4nMAssay Description:Displacement of [3H]-spiperone from dopamine D2 receptorMore data for this Ligand-Target Pair
In DepthDetails Article
TargetD(2) dopamine receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50283401((1-Benzyl-piperidin-4-yl)-phenyl-((E)-3-phenyl-all...)
Affinity DataIC50: >1.00E+4nMAssay Description:Displacement of [3H]-spiperone from dopamine D2 receptorMore data for this Ligand-Target Pair
In DepthDetails Article