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Found 11 Enz. Inhib. hit(s) with all data for entry = 50029412
TargetAcyl-CoA:cholesterol acyltransferase(Oryctolagus cuniculus)
TBA

Curated by ChEMBL
LigandPNGBDBM50284231(1-Benzhydryl-3-(2,6-diisopropyl-phenyl)-imidazolid...)
Affinity DataIC50:  1.30E+3nMAssay Description:In vitro Acyl coenzyme A:cholesterol acyltransferase inhibition by incubation with [14C]-oleolyl-CoA and intestinal microsomes isolated from choleste...More data for this Ligand-Target Pair
In DepthDetails Article
TargetAcyl-CoA:cholesterol acyltransferase(Oryctolagus cuniculus)
TBA

Curated by ChEMBL
LigandPNGBDBM50284230(5-Benzhydryl-3-(2,6-diisopropyl-phenyl)-imidazolid...)
Affinity DataIC50:  3.90E+3nMAssay Description:In vitro Acyl coenzyme A:cholesterol acyltransferase inhibition by incubation with [14C]-oleolyl-CoA and intestinal microsomes isolated from choleste...More data for this Ligand-Target Pair
In DepthDetails Article
TargetAcyl-CoA:cholesterol acyltransferase(Oryctolagus cuniculus)
TBA

Curated by ChEMBL
LigandPNGBDBM50284229(3-(2,6-Diisopropyl-phenyl)-1-(2,2-diphenyl-ethyl)-...)
Affinity DataIC50:  5.00E+3nMAssay Description:In vitro Acyl coenzyme A:cholesterol acyltransferase inhibition by incubation with [14C]-oleolyl-CoA and intestinal microsomes isolated from choleste...More data for this Ligand-Target Pair
In DepthDetails Article
TargetAcyl-CoA:cholesterol acyltransferase(Oryctolagus cuniculus)
TBA

Curated by ChEMBL
LigandPNGBDBM50284227(5-Decyl-2-(2,6-dimethyl-phenyl)-2,4-dihydro-pyrazo...)
Affinity DataIC50:  5.00E+3nMAssay Description:In vitro Acyl coenzyme A:cholesterol acyltransferase inhibition by incubation with [14C]-oleolyl-CoA and intestinal microsomes isolated from choleste...More data for this Ligand-Target Pair
In DepthDetails Article
TargetAcyl-CoA:cholesterol acyltransferase(Oryctolagus cuniculus)
TBA

Curated by ChEMBL
LigandPNGBDBM50284228(2-(2,4-Dimethyl-phenyl)-5-((Z)-heptadec-8-enyl)-2,...)
Affinity DataIC50:  5.00E+3nMAssay Description:In vitro Acyl coenzyme A:cholesterol acyltransferase inhibition by incubation with [14C]-oleolyl-CoA and intestinal microsomes isolated from choleste...More data for this Ligand-Target Pair
In DepthDetails Article
TargetAcyl-CoA:cholesterol acyltransferase(Oryctolagus cuniculus)
TBA

Curated by ChEMBL
LigandPNGBDBM50284233(2-(2,4-Dinitro-phenyl)-5-((Z)-heptadec-8-enyl)-2,4...)
Affinity DataIC50:  5.00E+3nMAssay Description:In vitro Acyl coenzyme A:cholesterol acyltransferase inhibition by incubation with [14C]-oleolyl-CoA and intestinal microsomes isolated from choleste...More data for this Ligand-Target Pair
In DepthDetails Article
TargetAcyl-CoA:cholesterol acyltransferase(Oryctolagus cuniculus)
TBA

Curated by ChEMBL
LigandPNGBDBM50284235(2-(2,4-Difluoro-phenyl)-5-((Z)-heptadec-8-enyl)-2,...)
Affinity DataIC50:  5.00E+3nMAssay Description:In vitro Acyl coenzyme A:cholesterol acyltransferase inhibition by incubation with [14C]-oleolyl-CoA and intestinal microsomes isolated from choleste...More data for this Ligand-Target Pair
In DepthDetails Article
TargetAcyl-CoA:cholesterol acyltransferase(Oryctolagus cuniculus)
TBA

Curated by ChEMBL
LigandPNGBDBM50284225(5-Benzyl-3-(2,6-diisopropyl-phenyl)-imidazolidin-4...)
Affinity DataIC50:  5.50E+3nMAssay Description:In vitro Acyl coenzyme A:cholesterol acyltransferase inhibition by incubation with [14C]-oleolyl-CoA and intestinal microsomes isolated from choleste...More data for this Ligand-Target Pair
In DepthDetails Article
TargetAcyl-CoA:cholesterol acyltransferase(Oryctolagus cuniculus)
TBA

Curated by ChEMBL
LigandPNGBDBM50284226(2-(2,4-Dichloro-phenyl)-5-((Z)-heptadec-8-enyl)-2,...)
Affinity DataIC50:  9.90E+3nMAssay Description:In vitro Acyl coenzyme A:cholesterol acyltransferase inhibition by incubation with [14C]-oleolyl-CoA and intestinal microsomes isolated from choleste...More data for this Ligand-Target Pair
In DepthDetails Article
TargetAcyl-CoA:cholesterol acyltransferase(Oryctolagus cuniculus)
TBA

Curated by ChEMBL
LigandPNGBDBM50284232(2-(2,6-Dichloro-phenyl)-5-((Z)-heptadec-8-enyl)-2,...)
Affinity DataIC50:  2.29E+4nMAssay Description:In vitro Acyl coenzyme A:cholesterol acyltransferase inhibition by incubation with [14C]-oleolyl-CoA and intestinal microsomes isolated from choleste...More data for this Ligand-Target Pair
In DepthDetails Article
TargetAcyl-CoA:cholesterol acyltransferase(Oryctolagus cuniculus)
TBA

Curated by ChEMBL
LigandPNGBDBM50284234(2-(2,6-Dimethyl-phenyl)-5-(2,2-diphenyl-ethyl)-2,4...)
Affinity DataIC50:  5.08E+4nMAssay Description:In vitro Acyl coenzyme A:cholesterol acyltransferase inhibition by incubation with [14C]-oleolyl-CoA and intestinal microsomes isolated from choleste...More data for this Ligand-Target Pair
In DepthDetails Article