Compile Data Set for Download or QSAR
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Found 35 Enz. Inhib. hit(s) with all data for entry = 50029656
TargetMu-type opioid receptor(Rattus norvegicus (rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50286589((S)-5-{(S)-2-[Bis-((R)-sec-butyl)-amino]-1-hydroxy...)
Affinity DataKi:  0.25nMAssay Description:Inhibition of [3H]-dihydromorphine (1 nM) binding to mu opioid receptor of rat brain homogenateMore data for this Ligand-Target Pair
In DepthDetails Article
TargetMu-type opioid receptor(Rattus norvegicus (rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50000092((-)-(etorphine) | (-)-morphine | (1S,5R,13R,14S)-1...)
Affinity DataKi:  3nMAssay Description:Inhibition of [3H]-dihydromorphine (1 nM) binding to mu opioid receptor of rat brain homogenateMore data for this Ligand-Target Pair
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50000092((-)-(etorphine) | (-)-morphine | (1S,5R,13R,14S)-1...)
Affinity DataKi:  15nMAssay Description:Inhibition of [3H]-[D-Pen2, D-Pen5]-enkephalin (2 nM) to Opioid receptor delta 1 of male Sprague-Dawley rat brain homogenateMore data for this Ligand-Target Pair
In DepthDetails Article
TargetKappa-type opioid receptor(Rattus norvegicus (rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50000092((-)-(etorphine) | (-)-morphine | (1S,5R,13R,14S)-1...)
Affinity DataKi:  27nMAssay Description:Inhibition of 9 (2nM) binding to Opioid receptor kappa 1 of rat brain homogenateMore data for this Ligand-Target Pair
In DepthDetails Article
TargetMu-type opioid receptor(Rattus norvegicus (rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50286584((S)-5-{(S)-2-[((R)-sec-Butyl)-((S)-sec-butyl)-amin...)
Affinity DataKi:  32nMAssay Description:Inhibition of [3H]-dihydromorphine (1 nM) binding to mu opioid receptor of rat brain homogenateMore data for this Ligand-Target Pair
In DepthDetails Article
TargetMu-type opioid receptor(Rattus norvegicus (rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50286586((R)-5-{(R)-2-[Bis-((R)-sec-butyl)-amino]-1-hydroxy...)
Affinity DataKi:  35nMAssay Description:Inhibition of [3H]-dihydromorphine (1 nM) binding to mu opioid receptor of rat brain homogenateMore data for this Ligand-Target Pair
In DepthDetails Article
TargetKappa-type opioid receptor(Rattus norvegicus (rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50286589((S)-5-{(S)-2-[Bis-((R)-sec-butyl)-amino]-1-hydroxy...)
Affinity DataKi:  63nMAssay Description:Inhibition of 9 (2nM) binding to Opioid receptor kappa 1 of rat brain homogenateMore data for this Ligand-Target Pair
In DepthDetails Article
TargetMu-type opioid receptor(Rattus norvegicus (rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50286587((R)-5-{(R)-2-[((R)-sec-Butyl)-((S)-sec-butyl)-amin...)
Affinity DataKi:  87nMAssay Description:Inhibition of [3H]-dihydromorphine (1 nM) binding to mu opioid receptor of rat brain homogenateMore data for this Ligand-Target Pair
In DepthDetails Article
TargetMu-type opioid receptor(Rattus norvegicus (rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50286580((R)-5-{(S)-2-[Bis-((R)-sec-butyl)-amino]-1-hydroxy...)
Affinity DataKi:  100nMAssay Description:Inhibition of [3H]-dihydromorphine (1 nM) binding to mu opioid receptor of rat brain homogenateMore data for this Ligand-Target Pair
In DepthDetails Article
TargetMu-type opioid receptor(Rattus norvegicus (rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50286585((S)-5-{(R)-2-[Bis-((S)-sec-butyl)-amino]-1-hydroxy...)
Affinity DataKi:  145nMAssay Description:Inhibition of [3H]-dihydromorphine (1 nM) binding to mu opioid receptor of rat brain homogenateMore data for this Ligand-Target Pair
In DepthDetails Article
TargetKappa-type opioid receptor(Rattus norvegicus (rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50286591((R)-5-{(S)-2-[((R)-sec-Butyl)-((S)-sec-butyl)-amin...)
Affinity DataKi:  198nMAssay Description:Inhibition of 9 (2nM) binding to Opioid receptor kappa 1 of rat brain homogenateMore data for this Ligand-Target Pair
In DepthDetails Article
TargetKappa-type opioid receptor(Rattus norvegicus (rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50286587((R)-5-{(R)-2-[((R)-sec-Butyl)-((S)-sec-butyl)-amin...)
Affinity DataKi:  260nMAssay Description:Inhibition of 9 (2nM) binding to Opioid receptor kappa 1 of rat brain homogenateMore data for this Ligand-Target Pair
In DepthDetails Article
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50286589((S)-5-{(S)-2-[Bis-((R)-sec-butyl)-amino]-1-hydroxy...)
Affinity DataKi:  265nMAssay Description:Inhibition of [3H]-[D-Pen2, D-Pen5]-enkephalin (2 nM) to Opioid receptor delta 1 of male Sprague-Dawley rat brain homogenateMore data for this Ligand-Target Pair
In DepthDetails Article
TargetKappa-type opioid receptor(Rattus norvegicus (rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50286583((R)-5-{(S)-2-[Bis-((S)-sec-butyl)-amino]-1-hydroxy...)
Affinity DataKi:  270nMAssay Description:Inhibition of 9 (2nM) binding to Opioid receptor kappa 1 of rat brain homogenateMore data for this Ligand-Target Pair
In DepthDetails Article
TargetMu-type opioid receptor(Rattus norvegicus (rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50286588((S)-5-{(R)-2-[((R)-sec-Butyl)-((S)-sec-butyl)-amin...)
Affinity DataKi:  340nMAssay Description:Inhibition of [3H]-dihydromorphine (1 nM) binding to mu opioid receptor of rat brain homogenateMore data for this Ligand-Target Pair
In DepthDetails Article
TargetMu-type opioid receptor(Rattus norvegicus (rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50286581((S)-5-{(R)-2-[Bis-((R)-sec-butyl)-amino]-1-hydroxy...)
Affinity DataKi:  390nMAssay Description:Inhibition of [3H]-dihydromorphine (1 nM) binding to mu opioid receptor of rat brain homogenateMore data for this Ligand-Target Pair
In DepthDetails Article
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50286581((S)-5-{(R)-2-[Bis-((R)-sec-butyl)-amino]-1-hydroxy...)
Affinity DataKi:  550nMAssay Description:Inhibition of [3H]-[D-Pen2, D-Pen5]-enkephalin (2 nM) to Opioid receptor delta 1 of male Sprague-Dawley rat brain homogenateMore data for this Ligand-Target Pair
In DepthDetails Article
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50286587((R)-5-{(R)-2-[((R)-sec-Butyl)-((S)-sec-butyl)-amin...)
Affinity DataKi:  1.78E+3nMAssay Description:Inhibition of [3H]-[D-Pen2, D-Pen5]-enkephalin (2 nM) to Opioid receptor delta 1 of male Sprague-Dawley rat brain homogenateMore data for this Ligand-Target Pair
In DepthDetails Article
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50286580((R)-5-{(S)-2-[Bis-((R)-sec-butyl)-amino]-1-hydroxy...)
Affinity DataKi:  1.85E+3nMAssay Description:Inhibition of [3H]-[D-Pen2, D-Pen5]-enkephalin (2 nM) to Opioid receptor delta 1 of male Sprague-Dawley rat brain homogenateMore data for this Ligand-Target Pair
In DepthDetails Article
TargetMu-type opioid receptor(Rattus norvegicus (rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50286582((S)-5-{(S)-2-[Bis-((S)-sec-butyl)-amino]-1-hydroxy...)
Affinity DataKi:  2.25E+3nMAssay Description:Inhibition of [3H]-dihydromorphine (1 nM) binding to mu opioid receptor of rat brain homogenateMore data for this Ligand-Target Pair
In DepthDetails Article
TargetKappa-type opioid receptor(Rattus norvegicus (rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50286588((S)-5-{(R)-2-[((R)-sec-Butyl)-((S)-sec-butyl)-amin...)
Affinity DataKi:  3.65E+3nMAssay Description:Inhibition of 9 (2nM) binding to Opioid receptor kappa 1 of rat brain homogenateMore data for this Ligand-Target Pair
In DepthDetails Article
TargetKappa-type opioid receptor(Rattus norvegicus (rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50286586((R)-5-{(R)-2-[Bis-((R)-sec-butyl)-amino]-1-hydroxy...)
Affinity DataKi:  4.85E+3nMAssay Description:Inhibition of 9 (2nM) binding to Opioid receptor kappa 1 of rat brain homogenateMore data for this Ligand-Target Pair
In DepthDetails Article
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50286583((R)-5-{(S)-2-[Bis-((S)-sec-butyl)-amino]-1-hydroxy...)
Affinity DataKi: >5.00E+3nMAssay Description:Inhibition of [3H]-[D-Pen2, D-Pen5]-enkephalin (2 nM) to Opioid receptor delta 1 of male Sprague-Dawley rat brain homogenateMore data for this Ligand-Target Pair
In DepthDetails Article
TargetKappa-type opioid receptor(Rattus norvegicus (rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50286585((S)-5-{(R)-2-[Bis-((S)-sec-butyl)-amino]-1-hydroxy...)
Affinity DataKi: >5.00E+3nMAssay Description:Inhibition of 9 (2nM) binding to Opioid receptor kappa 1 of rat brain homogenateMore data for this Ligand-Target Pair
In DepthDetails Article
TargetMu-type opioid receptor(Rattus norvegicus (rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50286591((R)-5-{(S)-2-[((R)-sec-Butyl)-((S)-sec-butyl)-amin...)
Affinity DataKi: >5.00E+3nMAssay Description:Inhibition of [3H]-dihydromorphine (1 nM) binding to mu opioid receptor of rat brain homogenateMore data for this Ligand-Target Pair
In DepthDetails Article
TargetKappa-type opioid receptor(Rattus norvegicus (rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50286581((S)-5-{(R)-2-[Bis-((R)-sec-butyl)-amino]-1-hydroxy...)
Affinity DataKi: >5.00E+3nMAssay Description:Inhibition of 9 (2nM) binding to Opioid receptor kappa 1 of rat brain homogenateMore data for this Ligand-Target Pair
In DepthDetails Article
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50286586((R)-5-{(R)-2-[Bis-((R)-sec-butyl)-amino]-1-hydroxy...)
Affinity DataKi: >5.00E+3nMAssay Description:Inhibition of [3H]-[D-Pen2, D-Pen5]-enkephalin (2 nM) to Opioid receptor delta 1 of male Sprague-Dawley rat brain homogenateMore data for this Ligand-Target Pair
In DepthDetails Article
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50286584((S)-5-{(S)-2-[((R)-sec-Butyl)-((S)-sec-butyl)-amin...)
Affinity DataKi: >5.00E+3nMAssay Description:Inhibition of [3H]-[D-Pen2, D-Pen5]-enkephalin (2 nM) to Opioid receptor delta 1 of male Sprague-Dawley rat brain homogenateMore data for this Ligand-Target Pair
In DepthDetails Article
TargetKappa-type opioid receptor(Rattus norvegicus (rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50286580((R)-5-{(S)-2-[Bis-((R)-sec-butyl)-amino]-1-hydroxy...)
Affinity DataKi: >5.00E+3nMAssay Description:Inhibition of 9 (2nM) binding to Opioid receptor kappa 1 of rat brain homogenateMore data for this Ligand-Target Pair
In DepthDetails Article
TargetMu-type opioid receptor(Rattus norvegicus (rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50286583((R)-5-{(S)-2-[Bis-((S)-sec-butyl)-amino]-1-hydroxy...)
Affinity DataKi: >5.00E+3nMAssay Description:Inhibition of [3H]-dihydromorphine (1 nM) binding to mu opioid receptor of rat brain homogenateMore data for this Ligand-Target Pair
In DepthDetails Article
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50286588((S)-5-{(R)-2-[((R)-sec-Butyl)-((S)-sec-butyl)-amin...)
Affinity DataKi: >5.00E+3nMAssay Description:Inhibition of [3H]-[D-Pen2, D-Pen5]-enkephalin (2 nM) to Opioid receptor delta 1 of male Sprague-Dawley rat brain homogenateMore data for this Ligand-Target Pair
In DepthDetails Article
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50286582((S)-5-{(S)-2-[Bis-((S)-sec-butyl)-amino]-1-hydroxy...)
Affinity DataKi: >5.00E+3nMAssay Description:Inhibition of [3H]-[D-Pen2, D-Pen5]-enkephalin (2 nM) to Opioid receptor delta 1 of male Sprague-Dawley rat brain homogenateMore data for this Ligand-Target Pair
In DepthDetails Article
TargetMu-type opioid receptor(Rattus norvegicus (rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50286590((R)-5-{(R)-2-[Bis-((S)-sec-butyl)-amino]-1-hydroxy...)
Affinity DataKi: >5.00E+3nMAssay Description:Inhibition of [3H]-dihydromorphine (1 nM) binding to mu opioid receptor of rat brain homogenateMore data for this Ligand-Target Pair
In DepthDetails Article
TargetKappa-type opioid receptor(Rattus norvegicus (rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50286582((S)-5-{(S)-2-[Bis-((S)-sec-butyl)-amino]-1-hydroxy...)
Affinity DataKi: >5.00E+3nMAssay Description:Inhibition of 9 (2nM) binding to Opioid receptor kappa 1 of rat brain homogenateMore data for this Ligand-Target Pair
In DepthDetails Article
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
TBA

Curated by ChEMBL
LigandPNGBDBM50286585((S)-5-{(R)-2-[Bis-((S)-sec-butyl)-amino]-1-hydroxy...)
Affinity DataKi: >5.00E+3nMAssay Description:Inhibition of [3H]-[D-Pen2, D-Pen5]-enkephalin (2 nM) to Opioid receptor delta 1 of male Sprague-Dawley rat brain homogenateMore data for this Ligand-Target Pair
In DepthDetails Article