Compile Data Set for Download or QSAR
maximum 50k data
Found 10 Enz. Inhib. hit(s) with all data for entry = 50029978
TargetSubstance-P receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50346332(2-Oxo-5-phenyl-1,2,3,5-tetrahydro-benzo[e][1,4]dia...)
Affinity DataKi:  10nMAssay Description:Tested for affinity against NK-1(Neurokinin-1) receptor expressed as pKiMore data for this Ligand-Target Pair
In DepthDetails Article
TargetSubstance-P receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50214736(CHEMBL304638)
Affinity DataKi:  32nMAssay Description:Tested for affinity against NK-1(Neurokinin-1) receptor expressed as pKiMore data for this Ligand-Target Pair
In DepthDetails Article
TargetSubstance-P receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50214732(CHEMBL64839)
Affinity DataKi:  40nMAssay Description:Tested for affinity against NK-1(Neurokinin-1) receptor expressed as pKiMore data for this Ligand-Target Pair
In DepthDetails Article
TargetSubstance-P receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50214733(CHEMBL62597)
Affinity DataKi:  316nMAssay Description:Tested for affinity against NK-1(Neurokinin-1) receptor expressed as pKiMore data for this Ligand-Target Pair
In DepthDetails Article
TargetSubstance-P receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50214734(CHEMBL302163)
Affinity DataKi:  631nMAssay Description:Tested for affinity against NK-1(Neurokinin-1) receptor expressed as pKiMore data for this Ligand-Target Pair
In DepthDetails Article
TargetSubstance-P receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50214641(CHEMBL291650)
Affinity DataKi:  794nMAssay Description:Tested for affinity against NK-1(Neurokinin-1) receptor expressed as pKiMore data for this Ligand-Target Pair
In DepthDetails Article
TargetSubstance-P receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50214735(CHEMBL64698)
Affinity DataKi:  1.00E+3nMAssay Description:Tested for affinity against NK-1(Neurokinin-1) receptor expressed as pKiMore data for this Ligand-Target Pair
In DepthDetails Article
TargetSubstance-P receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50214640(CHEMBL64862)
Affinity DataKi:  1.00E+3nMAssay Description:Tested for affinity against NK-1(Neurokinin-1) receptor expressed as pKiMore data for this Ligand-Target Pair
In DepthDetails Article
TargetCholecystokinin receptor type A(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50008634((S)-3,4-Dichloro-N-[1-dipentylcarbamoyl-2-(1H-indo...)
Affinity DataIC50:  190nMAssay Description:Concentration required for 50% inhibition of cholecystokinin A(CCK A)More data for this Ligand-Target Pair
In DepthDetails Article
TargetSubstance-P receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50289925(2-Acetylamino-N-benzyl-3-(1H-indol-3-yl)-N-methyl-...)
Affinity DataIC50:  750nMAssay Description:Concentration required for 50% inhibition of neurokinin-1 receptorMore data for this Ligand-Target Pair
In DepthDetails Article