Compile Data Set for Download or QSAR
maximum 50k data
Found 8 Enz. Inhib. hit(s) with all data for entry = 50005309
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
University Of Minnesota

Curated by ChEMBL
LigandPNGBDBM50035476(CHEMBL413530 | N-[(S)-1-(3-Amino-phenyl)-2-pyrroli...)
Affinity DataIC50:  0.000320nMAssay Description:Binding affinity kappa opioid receptor in guinea pig brain membranes; using 1 nM [3H]-U69,593 as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
University Of Minnesota

Curated by ChEMBL
LigandPNGBDBM50035471(2-(3,4-Dichloro-phenyl)-N-[(S)-1-(3-isothiocyanato...)
Affinity DataIC50:  2.20nMAssay Description:Binding affinity kappa opioid receptor in guinea pig brain membranes, using 1 nM [3H]-U69,593 as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(GUINEA PIG)
University Of Minnesota

Curated by ChEMBL
LigandPNGBDBM50035476(CHEMBL413530 | N-[(S)-1-(3-Amino-phenyl)-2-pyrroli...)
Affinity DataIC50:  31nMAssay Description:Binding affinity for mu opioid receptor in guinea pig brain membranes; using 2 nM [3H]-DAMGO as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
University Of Minnesota

Curated by ChEMBL
LigandPNGBDBM50035476(CHEMBL413530 | N-[(S)-1-(3-Amino-phenyl)-2-pyrroli...)
Affinity DataIC50:  89nMAssay Description:Binding affinity for delta opioid receptor in guinea pig brain membranes; using 2 nM [3H]-DPDPE as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
University Of Minnesota

Curated by ChEMBL
LigandPNGBDBM50035471(2-(3,4-Dichloro-phenyl)-N-[(S)-1-(3-isothiocyanato...)
Affinity DataIC50: >1.00E+3nMAssay Description:Binding affinity for delta opioid receptor in guinea pig brain membranes, using 2 nM [3H]-DPDPE as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(GUINEA PIG)
University Of Minnesota

Curated by ChEMBL
LigandPNGBDBM50035471(2-(3,4-Dichloro-phenyl)-N-[(S)-1-(3-isothiocyanato...)
Affinity DataIC50:  1.80E+3nMAssay Description:Binding affinity for mu opioid receptor in guinea pig brain membranes, using 2 nM [3H]-DAMGO as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
University Of Minnesota

Curated by ChEMBL
LigandPNGBDBM50035471(2-(3,4-Dichloro-phenyl)-N-[(S)-1-(3-isothiocyanato...)
Affinity DataKd:  2.40nMAssay Description:Tested for competitive covalent binding of compound against k opioid receptor in guinea pig brain membrane using [3H]-U-69,593 as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
University Of Minnesota

Curated by ChEMBL
LigandPNGBDBM50035476(CHEMBL413530 | N-[(S)-1-(3-Amino-phenyl)-2-pyrroli...)
Affinity DataKd:  3.40nMAssay Description:Tested for competitive covalent binding of compound against k opioid receptor in guinea pig brain membrane; using [3H]-U-69,593 as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed