Compile Data Set for Download or QSAR
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Found 10 Enz. Inhib. hit(s) with all data for entry = 50005716
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Oregon State University

Curated by ChEMBL
LigandPNGBDBM50002184(CHEMBL415330 | H-Tyr-Gly-Gly-Phe-Leu-Arg-Arg-Ile-A...)
Affinity DataKi:  0.150nMAssay Description:Compound was tested for binding affinity towards kappa opioid receptor in guinea pig cerebellar membrane using [3H]-bremazocineMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Oregon State University

Curated by ChEMBL
LigandPNGBDBM50002184(CHEMBL415330 | H-Tyr-Gly-Gly-Phe-Leu-Arg-Arg-Ile-A...)
Affinity DataKi:  0.190nMAssay Description:Compound was tested for binding affinity towards mu-opioid receptor in rat forebrain membrane using [3H]-DAMGOMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
Oregon State University

Curated by ChEMBL
LigandPNGBDBM50002184(CHEMBL415330 | H-Tyr-Gly-Gly-Phe-Leu-Arg-Arg-Ile-A...)
Affinity DataKi:  3.90nMAssay Description:Compound was tested for binding affinity towards delta-opioid receptor in rat forebrain membrane using [3H]-DPDPEMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Oregon State University

Curated by ChEMBL
LigandPNGBDBM50040187(CHEMBL404976 | Tyr-Aib-Gly-Phe-Leu-Arg-Arg-Ile-Arg...)
Affinity DataKi:  10nMAssay Description:Compound was tested for binding affinity towards mu-opioid receptor in rat forebrain membrane using [3H]-DAMGOMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Oregon State University

Curated by ChEMBL
LigandPNGBDBM50040188((cis)Tyr-1-Amino-CycloHexylcarbonyl-Phe-Leu-Arg-Ar...)
Affinity DataKi:  13nMAssay Description:Compound was tested for binding affinity towards kappa opioid receptor in guinea pig cerebellar membrane using [3H]-bremazocineMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Oregon State University

Curated by ChEMBL
LigandPNGBDBM50040188((cis)Tyr-1-Amino-CycloHexylcarbonyl-Phe-Leu-Arg-Ar...)
Affinity DataKi:  13nMAssay Description:Compound was tested for binding affinity towards kappa opioid receptor in guinea pig cerebellar membrane using [3H]-bremazocineMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Oregon State University

Curated by ChEMBL
LigandPNGBDBM50040187(CHEMBL404976 | Tyr-Aib-Gly-Phe-Leu-Arg-Arg-Ile-Arg...)
Affinity DataKi:  50nMAssay Description:Compound was tested for binding affinity towards kappa opioid receptor in guinea pig cerebellar membrane using [3H]-bremazocineMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
Oregon State University

Curated by ChEMBL
LigandPNGBDBM50040188((cis)Tyr-1-Amino-CycloHexylcarbonyl-Phe-Leu-Arg-Ar...)
Affinity DataKi:  117nMAssay Description:Compound was tested for binding affinity towards delta-opioid receptor in rat forebrain membrane using [3H]-DPDPEMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Oregon State University

Curated by ChEMBL
LigandPNGBDBM50040188((cis)Tyr-1-Amino-CycloHexylcarbonyl-Phe-Leu-Arg-Ar...)
Affinity DataKi:  275nMAssay Description:Compound was tested for binding affinity towards mu-opioid receptor in rat forebrain membrane using [3H]-DAMGOMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
Oregon State University

Curated by ChEMBL
LigandPNGBDBM50040188((cis)Tyr-1-Amino-CycloHexylcarbonyl-Phe-Leu-Arg-Ar...)
Affinity DataKi:  1.37E+3nMAssay Description:Compound was tested for binding affinity towards delta-opioid receptor in rat forebrain membrane using [3H]-DPDPEMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed