Compile Data Set for Download or QSAR
maximum 50k data
Found 27 Enz. Inhib. hit(s) with all data for entry = 50036233
TargetDelta-type opioid receptor(MOUSE)
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50041669(2-Amino-N-(7-benzyl-4-dihydroxymethyl-3,3,10,14,14...)
Affinity DataIC50:  12nMAssay Description:Inhibitory activity of the electrically induced smooth muscle contraction of mouse vas deferensMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50041669(2-Amino-N-(7-benzyl-4-dihydroxymethyl-3,3,10,14,14...)
Affinity DataIC50:  18nMAssay Description:Evaluation for the binding affinity by competitive inhibition of [3H]- p-chloro DPDPE bindingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50041663(2-Amino-N-(7-benzyl-4-dihydroxymethyl-10-hydroxyme...)
Affinity DataIC50:  42nMAssay Description:Evaluation for the binding affinity by competitive inhibition of [3H]- p-chloro DPDPE bindingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50453339(CHEMBL2372412)
Affinity DataIC50:  66nMAssay Description:Evaluation for the binding affinity by competitive inhibition of [3H]- p-chloro DPDPE bindingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(MOUSE)
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50453339(CHEMBL2372412)
Affinity DataIC50:  85nMAssay Description:Inhibitory activity of the electrically induced smooth muscle contraction of mouse vas deferensMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(MOUSE)
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50041663(2-Amino-N-(7-benzyl-4-dihydroxymethyl-10-hydroxyme...)
Affinity DataIC50:  250nMAssay Description:Inhibitory activity of the electrically induced smooth muscle contraction of mouse vas deferensMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(MOUSE)
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50001683(13-[2-Amino-3-(4-hydroxy-phenyl)-propionylamino]-7...)
Affinity DataIC50:  570nMAssay Description:Inhibitory activity of the electrically induced smooth muscle contraction of mouse vas deferensMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50001683(13-[2-Amino-3-(4-hydroxy-phenyl)-propionylamino]-7...)
Affinity DataIC50:  620nMAssay Description:Evaluation for the binding affinity by competitive inhibition of [3H]- p-chloro DPDPE bindingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(MOUSE)
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50041666(2-Amino-N-((S)-7-benzyl-4-dihydroxymethyl-10-hydro...)
Affinity DataIC50:  760nMAssay Description:Inhibitory activity of the electrically induced smooth muscle contraction of mouse vas deferensMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50041666(2-Amino-N-((S)-7-benzyl-4-dihydroxymethyl-10-hydro...)
Affinity DataIC50:  760nMAssay Description:Evaluation for the binding affinity by competitive inhibition of [3H]- p-chloro DPDPE bindingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(GUINEA PIG)
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50453339(CHEMBL2372412)
Affinity DataIC50:  4.90E+3nMAssay Description:Inhibitory activity of the electrically induced guinea pig ileum longitudal muscle-myenteric plexusMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(GUINEA PIG)
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50001683(13-[2-Amino-3-(4-hydroxy-phenyl)-propionylamino]-7...)
Affinity DataIC50:  7.30E+3nMAssay Description:Inhibitory activity of the electrically induced guinea pig ileum longitudal muscle-myenteric plexusMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50041669(2-Amino-N-(7-benzyl-4-dihydroxymethyl-3,3,10,14,14...)
Affinity DataIC50:  1.10E+4nMAssay Description:Evaluation for the binding affinity by competitive inhibition of [3H]- CTOP bindingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50453339(CHEMBL2372412)
Affinity DataIC50:  1.20E+4nMAssay Description:Evaluation for the binding affinity by competitive inhibition of [3H]- CTOP bindingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50041663(2-Amino-N-(7-benzyl-4-dihydroxymethyl-10-hydroxyme...)
Affinity DataIC50: >2.25E+4nMAssay Description:Evaluation for the binding affinity by competitive inhibition of [3H]- CTOP bindingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50041668(2-Amino-N-((S)-7-benzyl-4-dihydroxymethyl-10-ethyl...)
Affinity DataIC50:  3.00E+4nMAssay Description:Evaluation for the binding affinity by competitive inhibition of [3H]- p-chloro DPDPE bindingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(MOUSE)
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50041668(2-Amino-N-((S)-7-benzyl-4-dihydroxymethyl-10-ethyl...)
Affinity DataIC50:  3.00E+4nMAssay Description:Inhibitory activity of the electrically induced smooth muscle contraction of mouse vas deferensMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(GUINEA PIG)
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50041668(2-Amino-N-((S)-7-benzyl-4-dihydroxymethyl-10-ethyl...)
Affinity DataIC50:  3.00E+4nMAssay Description:Inhibitory activity of the electrically induced guinea pig ileum longitudal muscle-myenteric plexusMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50041665(2-Amino-N-(7-benzyl-4-dihydroxymethyl-10-ethyl-3,3...)
Affinity DataIC50:  3.30E+4nMAssay Description:Evaluation for the binding affinity by competitive inhibition of [3H]- CTOP bindingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50041665(2-Amino-N-(7-benzyl-4-dihydroxymethyl-10-ethyl-3,3...)
Affinity DataIC50:  3.30E+4nMAssay Description:Evaluation for the binding affinity by competitive inhibition of [3H]- p-chloro DPDPE bindingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(MOUSE)
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50041665(2-Amino-N-(7-benzyl-4-dihydroxymethyl-10-ethyl-3,3...)
Affinity DataIC50:  3.30E+4nMAssay Description:Inhibitory activity of the electrically induced smooth muscle contraction of mouse vas deferensMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(GUINEA PIG)
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50041665(2-Amino-N-(7-benzyl-4-dihydroxymethyl-10-ethyl-3,3...)
Affinity DataIC50:  3.30E+4nMAssay Description:Inhibitory activity of the electrically induced guinea pig ileum longitudal muscle-myenteric plexusMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50001683(13-[2-Amino-3-(4-hydroxy-phenyl)-propionylamino]-7...)
Affinity DataIC50: >3.50E+4nMAssay Description:Evaluation for the binding affinity by competitive inhibition of [3H]- CTOP bindingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(GUINEA PIG)
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50041663(2-Amino-N-(7-benzyl-4-dihydroxymethyl-10-hydroxyme...)
Affinity DataIC50:  3.90E+4nMAssay Description:Inhibitory activity of the electrically induced guinea pig ileum longitudal muscle-myenteric plexusMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50041666(2-Amino-N-((S)-7-benzyl-4-dihydroxymethyl-10-hydro...)
Affinity DataIC50: >5.00E+4nMAssay Description:Evaluation for the binding affinity by competitive inhibition of [3H]- CTOP bindingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50041668(2-Amino-N-((S)-7-benzyl-4-dihydroxymethyl-10-ethyl...)
Affinity DataIC50: >5.00E+4nMAssay Description:Evaluation for the binding affinity by competitive inhibition of [3H]- CTOP bindingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(GUINEA PIG)
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50041669(2-Amino-N-(7-benzyl-4-dihydroxymethyl-3,3,10,14,14...)
Affinity DataIC50:  5.40E+4nMAssay Description:Inhibitory activity of the electrically induced guinea pig ileum longitudal muscle-myenteric plexusMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed