Compile Data Set for Download or QSAR
maximum 50k data
Found 4 Enz. Inhib. hit(s) with all data for entry = 4984
TargetHistamine H1 receptor(Homo sapiens (Human))
University of Cambridge

Curated by PDSP Ki Database
LigandPNGBDBM84646(CAS_86181-42-2 | NSC_55482 | Temelastine)
Affinity DataKi:  3.20nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H1 receptor(Homo sapiens (Human))
University of Cambridge

Curated by PDSP Ki Database
LigandPNGBDBM22567(3H]pyrilamine | CHEMBL511 | Dorantamin | Mepyramin...)
Affinity DataKi:  4.70nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMedDrugBank

TargetHistamine H1 receptor(Homo sapiens (Human))
University of Cambridge

Curated by PDSP Ki Database
LigandPNGBDBM84647(CAS_2830867 | NSC_2830867 | QMDP(+))
In DepthDetails ArticlePubMed
TargetHistamine H1 receptor(Homo sapiens (Human))
University of Cambridge

Curated by PDSP Ki Database
LigandPNGBDBM7966(2-(1H-imidazol-4-yl)ethan-1-amine | CHEMBL544208 |...)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMedDrugBank