Compile Data Set for Download or QSAR
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Found 15 Enz. Inhib. hit(s) with all data for entry = 50007922
TargetProthrombin(Homo sapiens (Human))
Biotech Research Institute

Curated by ChEMBL
LigandPNGBDBM50069294((S)-3-[4-(carbohydrazonamidol)-phenyl]-N-cyclopent...)
Affinity DataKi:  0.380nMAssay Description:Compound was tested for inhibitory activity against human thrombinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Bos taurus (Bovine))
Biotech Research Institute

Curated by ChEMBL
LigandPNGBDBM50069294((S)-3-[4-(carbohydrazonamidol)-phenyl]-N-cyclopent...)
Affinity DataKi:  1.10nMAssay Description:Compound was tested for inhibitory activity against bovine thrombinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Bos taurus (Bovine))
Biotech Research Institute

Curated by ChEMBL
LigandPNGBDBM50069292(CHEMBL156082 | N-ethyl-N-cyclopentyl-3-(4-hydrazon...)
Affinity DataKi:  4nMAssay Description:Compound was tested for inhibitory activity against bovine thrombinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Bos taurus (Bovine))
Biotech Research Institute

Curated by ChEMBL
LigandPNGBDBM50069293(CHEMBL440188 | N-methyl-N-n-butyl-3-(4-hydrazonofo...)
Affinity DataKi:  41nMAssay Description:Compound was tested for inhibitory activity against bovine thrombinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Bos taurus (Bovine))
Biotech Research Institute

Curated by ChEMBL
LigandPNGBDBM50069296(CHEMBL347371 | N-(n-propyl)-N-cyclopentyl-3-(4-hyd...)
Affinity DataKi:  93nMAssay Description:Compound was tested for inhibitory activity against bovine thrombinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Bos taurus (Bovine))
Biotech Research Institute

Curated by ChEMBL
LigandPNGBDBM50069298(CHEMBL434678 | N-methyl-N-cyclohexyl-3-(4-hydrazon...)
Affinity DataKi:  152nMAssay Description:Compound was tested for inhibitory activity against bovine thrombinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Bos taurus (Bovine))
Biotech Research Institute

Curated by ChEMBL
LigandPNGBDBM50069299(CHEMBL155317 | N-(n-butyl)-N-cyclopentyl-3-(4-hydr...)
Affinity DataKi:  231nMAssay Description:Compound was tested for inhibitory activity against bovine thrombinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Bos taurus (Bovine))
Biotech Research Institute

Curated by ChEMBL
LigandPNGBDBM50069295(CHEMBL348175 | N-methyl-N-cyclopropyl-3-(4-hydrazo...)
Affinity DataKi:  247nMAssay Description:Compound was tested for inhibitory activity against bovine thrombinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Bos taurus (Bovine))
Biotech Research Institute

Curated by ChEMBL
LigandPNGBDBM50069300(CHEMBL350901 | N-hydroxy-N-cyclopentyl-3-(4-hydraz...)
Affinity DataKi:  367nMAssay Description:Compound was tested for inhibitory activity against bovine thrombinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
Biotech Research Institute

Curated by ChEMBL
LigandPNGBDBM50069294((S)-3-[4-(carbohydrazonamidol)-phenyl]-N-cyclopent...)
Affinity DataKi:  1.10E+3nMAssay Description:The compound was tested for inhibitory activity against Coagulation factor XMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Bos taurus (Bovine))
Biotech Research Institute

Curated by ChEMBL
LigandPNGBDBM50069297(1-[3-[4-amino(amineimino)methylphenyl]-2-(2-naphth...)
Affinity DataKi:  1.47E+3nMAssay Description:Compound was tested for inhibitory activity against bovine thrombinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTrypsin(Homo sapiens (Human))
Biotech Research Institute

Curated by ChEMBL
LigandPNGBDBM50069294((S)-3-[4-(carbohydrazonamidol)-phenyl]-N-cyclopent...)
Affinity DataKi:  3.29E+3nMAssay Description:Compound was tested for inhibitory activity against bovine trypsinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Bos taurus (Bovine))
Biotech Research Institute

Curated by ChEMBL
LigandPNGBDBM50069301(CHEMBL155311 | N-hydroxyethyl-N-cyclopentyl-3-(4-h...)
Affinity DataKi:  7.04E+3nMAssay Description:Compound was tested for inhibitory activity against bovine thrombinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTissue-type plasminogen activator(Homo sapiens (Human))
Biotech Research Institute

Curated by ChEMBL
LigandPNGBDBM50069294((S)-3-[4-(carbohydrazonamidol)-phenyl]-N-cyclopent...)
Affinity DataKi:  2.72E+4nMAssay Description:The compound was tested for inhibitory activity against tissue plasminogen activatorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlasminogen(Homo sapiens (Human))
Biotech Research Institute

Curated by ChEMBL
LigandPNGBDBM50069294((S)-3-[4-(carbohydrazonamidol)-phenyl]-N-cyclopent...)
Affinity DataKi:  4.79E+4nMAssay Description:The compound was tested for inhibitory activity against human plasminMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed