Compile Data Set for Download or QSAR
maximum 50k data
Found 21 Enz. Inhib. hit(s) with all data for entry = 10884
TargetNon-receptor tyrosine-protein kinase TYK2 [556-871](Homo sapiens (Human))
Janssen Pharmaceutica

WIPO
LigandPNGBDBM576244(WO2022109580, Example 3)
Affinity DataIC50:  1nMAssay Description:The probe displacement assay is conducted as follows: In a 384-well plate, test compound along with recombinantly expressed His-tagged protein corres...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetNon-receptor tyrosine-protein kinase TYK2 [556-871](Homo sapiens (Human))
Janssen Pharmaceutica

WIPO
LigandPNGBDBM576242(WO2022109580, Example 1)
Affinity DataIC50:  2nMAssay Description:The probe displacement assay is conducted as follows: In a 384-well plate, test compound along with recombinantly expressed His-tagged protein corres...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetNon-receptor tyrosine-protein kinase TYK2 [556-871](Homo sapiens (Human))
Janssen Pharmaceutica

WIPO
LigandPNGBDBM576262(WO2022109580, Example 25)
Affinity DataIC50:  2nMAssay Description:The probe displacement assay is conducted as follows: In a 384-well plate, test compound along with recombinantly expressed His-tagged protein corres...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetNon-receptor tyrosine-protein kinase TYK2 [556-871](Homo sapiens (Human))
Janssen Pharmaceutica

WIPO
LigandPNGBDBM576245(WO2022109580, Example 4)
Affinity DataIC50:  2nMAssay Description:The probe displacement assay is conducted as follows: In a 384-well plate, test compound along with recombinantly expressed His-tagged protein corres...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetNon-receptor tyrosine-protein kinase TYK2 [556-871](Homo sapiens (Human))
Janssen Pharmaceutica

WIPO
LigandPNGBDBM576250(WO2022109580, Example 11)
Affinity DataIC50:  2nMAssay Description:The probe displacement assay is conducted as follows: In a 384-well plate, test compound along with recombinantly expressed His-tagged protein corres...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetNon-receptor tyrosine-protein kinase TYK2 [556-871](Homo sapiens (Human))
Janssen Pharmaceutica

WIPO
LigandPNGBDBM576257(WO2022109580, Example 19)
Affinity DataIC50:  2nMAssay Description:The probe displacement assay is conducted as follows: In a 384-well plate, test compound along with recombinantly expressed His-tagged protein corres...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetNon-receptor tyrosine-protein kinase TYK2 [556-871](Homo sapiens (Human))
Janssen Pharmaceutica

WIPO
LigandPNGBDBM576248(WO2022109580, Example 9)
Affinity DataIC50:  2nMAssay Description:The probe displacement assay is conducted as follows: In a 384-well plate, test compound along with recombinantly expressed His-tagged protein corres...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetNon-receptor tyrosine-protein kinase TYK2 [556-871](Homo sapiens (Human))
Janssen Pharmaceutica

WIPO
LigandPNGBDBM576252(WO2022109580, Example 13)
Affinity DataIC50:  2nMAssay Description:The probe displacement assay is conducted as follows: In a 384-well plate, test compound along with recombinantly expressed His-tagged protein corres...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetNon-receptor tyrosine-protein kinase TYK2 [556-871](Homo sapiens (Human))
Janssen Pharmaceutica

WIPO
LigandPNGBDBM576246(WO2022109580, Example 5)
Affinity DataIC50:  3nMAssay Description:The probe displacement assay is conducted as follows: In a 384-well plate, test compound along with recombinantly expressed His-tagged protein corres...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetNon-receptor tyrosine-protein kinase TYK2 [556-871](Homo sapiens (Human))
Janssen Pharmaceutica

WIPO
LigandPNGBDBM576243(WO2022109580, Example 2)
Affinity DataIC50:  4nMAssay Description:The probe displacement assay is conducted as follows: In a 384-well plate, test compound along with recombinantly expressed His-tagged protein corres...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetNon-receptor tyrosine-protein kinase TYK2 [556-871](Homo sapiens (Human))
Janssen Pharmaceutica

WIPO
LigandPNGBDBM576255(WO2022109580, Example 17)
Affinity DataIC50:  4nMAssay Description:The probe displacement assay is conducted as follows: In a 384-well plate, test compound along with recombinantly expressed His-tagged protein corres...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetNon-receptor tyrosine-protein kinase TYK2 [556-871](Homo sapiens (Human))
Janssen Pharmaceutica

WIPO
LigandPNGBDBM576253(WO2022109580, Example 14)
Affinity DataIC50:  4nMAssay Description:The probe displacement assay is conducted as follows: In a 384-well plate, test compound along with recombinantly expressed His-tagged protein corres...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetNon-receptor tyrosine-protein kinase TYK2 [556-871](Homo sapiens (Human))
Janssen Pharmaceutica

WIPO
LigandPNGBDBM576260(WO2022109580, Example 23)
Affinity DataIC50:  5nMAssay Description:The probe displacement assay is conducted as follows: In a 384-well plate, test compound along with recombinantly expressed His-tagged protein corres...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetNon-receptor tyrosine-protein kinase TYK2 [556-871](Homo sapiens (Human))
Janssen Pharmaceutica

WIPO
LigandPNGBDBM576249(WO2022109580, Example 10)
Affinity DataIC50:  6nMAssay Description:The probe displacement assay is conducted as follows: In a 384-well plate, test compound along with recombinantly expressed His-tagged protein corres...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetNon-receptor tyrosine-protein kinase TYK2 [556-871](Homo sapiens (Human))
Janssen Pharmaceutica

WIPO
LigandPNGBDBM576251(WO2022109580, Example 12)
Affinity DataIC50:  6nMAssay Description:The probe displacement assay is conducted as follows: In a 384-well plate, test compound along with recombinantly expressed His-tagged protein corres...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetNon-receptor tyrosine-protein kinase TYK2 [556-871](Homo sapiens (Human))
Janssen Pharmaceutica

WIPO
LigandPNGBDBM576254(WO2022109580, Example 16)
Affinity DataIC50:  7nMAssay Description:The probe displacement assay is conducted as follows: In a 384-well plate, test compound along with recombinantly expressed His-tagged protein corres...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetNon-receptor tyrosine-protein kinase TYK2 [556-871](Homo sapiens (Human))
Janssen Pharmaceutica

WIPO
LigandPNGBDBM576256(WO2022109580, Example 18)
Affinity DataIC50:  8nMAssay Description:The probe displacement assay is conducted as follows: In a 384-well plate, test compound along with recombinantly expressed His-tagged protein corres...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetNon-receptor tyrosine-protein kinase TYK2 [556-871](Homo sapiens (Human))
Janssen Pharmaceutica

WIPO
LigandPNGBDBM576247(WO2022109580, Example 6)
Affinity DataIC50:  8nMAssay Description:The probe displacement assay is conducted as follows: In a 384-well plate, test compound along with recombinantly expressed His-tagged protein corres...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetNon-receptor tyrosine-protein kinase TYK2 [556-871](Homo sapiens (Human))
Janssen Pharmaceutica

WIPO
LigandPNGBDBM576258(WO2022109580, Example 20)
Affinity DataIC50:  11nMAssay Description:The probe displacement assay is conducted as follows: In a 384-well plate, test compound along with recombinantly expressed His-tagged protein corres...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetNon-receptor tyrosine-protein kinase TYK2 [556-871](Homo sapiens (Human))
Janssen Pharmaceutica

WIPO
LigandPNGBDBM576259(WO2022109580, Example 22)
Affinity DataIC50:  14nMAssay Description:The probe displacement assay is conducted as follows: In a 384-well plate, test compound along with recombinantly expressed His-tagged protein corres...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetNon-receptor tyrosine-protein kinase TYK2 [556-871](Homo sapiens (Human))
Janssen Pharmaceutica

WIPO
LigandPNGBDBM576261(WO2022109580, Example 24)
Affinity DataIC50:  42nMAssay Description:The probe displacement assay is conducted as follows: In a 384-well plate, test compound along with recombinantly expressed His-tagged protein corres...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed