Reaction Details
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Target
Acid-sensing ion channel 2
Ligand
BDBM50510050
Substrate
n/a
Meas. Tech.
ChEMBL_1840001 (CHEMBL4340216)
IC50
>30000±n/a nM
Citation
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More Info.:
Target
Name:
Acid-sensing ion channel 2
Synonyms:
ASIC2_MOUSE | Accn1 | Acid-sensing ion channel 2 | Amiloride-sensitive brain sodium channel | Amiloride-sensitive cation channel 1, neuronal | Asic2 | BNC1 | Bnac1 | Brain sodium channel 1
Type:
PROTEIN
Mol. Mass.:
57721.82
Organism:
Mus musculus
Description:
ChEMBL_119368
Residue:
512
Sequence:
MDLKESPSEGSLQPSSIQIFANTSTLHGIRHIFVYGPLTIRRVLWAVAFVGSLGLLLVESSERVSYYFSYQHVTKVDEVVAQSLVFPAVTLCNLNGFRFSRLTTNDLYHAGELLALLDVNLQIPDPHLADPTVLEALRQKANFKHYKPKQFSMLEFLHRVGHDLKDMMLYCKFKGQECGHQDFTTVFTKYGKCYMFNSGEDGKPLLTTVKGGTGNGLEIMLDIQQDEYLPIWGETEETTFEAGVKVQIHSQSEPPFIQELGFGVAPGFQTFVATQEQRLTYLPPPWGECRSSEMGLDFFPVYSITACRIDCETRYIVENCNCRMVHMPGDAPFCTPEQHKECAEPALGLLAEKDSNYCLCRTPCNLTRYNKELSMVKIPSKTSAKYLEKKFNKSEKYISENILVLDIFFEALNYETIEQKKAYEVAALLGDIGGQMGLFIGASILTILELFDYIYELIKEKLLDLLGKEEEEGSHDENMSTCDTMPNHSETISHTVNVPLQTALGTLEEIAC