Reaction Details Report a problem with these data
Target
Galanin receptor type 3
Ligand
BDBM64723
Substrate
n/a
IC50
128.42±n/a nM
Citation
 PubChem, PC Fluorescence-based cell-based primary high throughput dose response assay to identify antagonists of the Galanin Receptor 3 (GalR3). PubChem Bioassay (2013)[AID] 
Target
Name:
Galanin receptor type 3
Synonyms:
GALNR3 | GALR3 | GALR3_HUMAN | Galanin R3 | Galanin receptor 3 | Galanin receptor type 3
Type:
Enzyme Catalytic Domain
Mol. Mass.:
39599.97
Organism:
Homo sapiens (Human)
Description:
Galanin R3 GALR3 HUMAN::O60755
Residue:
368
Sequence:
MADAQNISLDSPGSVGAVAVPVVFALIFLLGTVGNGLVLAVLLQPGPSAWQEPGSTTDLFILNLAVADLCFILCCVPFQATIYTLDAWLFGALVCKAVHLLIYLTMYASSFTLAAVSVDRYLAVRHPLRSRALRTPRNARAAVGLVWLLAALFSAPYLSYYGTVRYGALELCVPAWEDARRRALDVATFAAGYLLPVAVVSLAYGRTLRFLWAAVGPAGAAAAEARRRATGRAGRAMLAVAALYALCWGPHHALILCFWYGRFAFSPATYACRLASHCLAYANSCLNPLVYALASRHFRARFRRLWPCGRRRRHRARRALRRVRPASSGPPGCPGDARPSGRLLAGGGQGPEPREGPVHGGEAARGPE
  
Inhibitor
Name:
BDBM64723
Synonyms:
(1-Phenyl-ethyl)-quinazolin-4-yl-amine | 1-phenylethyl(quinazolin-4-yl)amine | MLS001206299 | N-(1-phenylethyl)-4-quinazolinamine | N-(1-phenylethyl)quinazolin-4-amine | SMR000518519 | cid_3146673
Type:
Small organic molecule
Emp. Form.:
C16H15N3
Mol. Mass.:
249.3104
SMILES:
CC(Nc1ncnc2ccccc12)c1ccccc1
Structure:
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