Reaction Details Report a problem with these data
Target
Galanin receptor type 3
Ligand
BDBM97156
Substrate
n/a
IC50
203.24±n/a nM
Citation
 PubChem, PC Fluorescence-based cell-based primary high throughput dose response assay to identify antagonists of the Galanin Receptor 3 (GalR3). PubChem Bioassay (2013)[AID] 
Target
Name:
Galanin receptor type 3
Synonyms:
GALNR3 | GALR3 | GALR3_HUMAN | Galanin R3 | Galanin receptor 3 | Galanin receptor type 3
Type:
Enzyme Catalytic Domain
Mol. Mass.:
39599.97
Organism:
Homo sapiens (Human)
Description:
Galanin R3 GALR3 HUMAN::O60755
Residue:
368
Sequence:
MADAQNISLDSPGSVGAVAVPVVFALIFLLGTVGNGLVLAVLLQPGPSAWQEPGSTTDLFILNLAVADLCFILCCVPFQATIYTLDAWLFGALVCKAVHLLIYLTMYASSFTLAAVSVDRYLAVRHPLRSRALRTPRNARAAVGLVWLLAALFSAPYLSYYGTVRYGALELCVPAWEDARRRALDVATFAAGYLLPVAVVSLAYGRTLRFLWAAVGPAGAAAAEARRRATGRAGRAMLAVAALYALCWGPHHALILCFWYGRFAFSPATYACRLASHCLAYANSCLNPLVYALASRHFRARFRRLWPCGRRRRHRARRALRRVRPASSGPPGCPGDARPSGRLLAGGGQGPEPREGPVHGGEAARGPE
  
Inhibitor
Name:
BDBM97156
Synonyms:
1-(4-Chloro-benzyl)-2-methyl-1H-benzoimidazole | 1-(4-chlorobenzyl)-2-methyl-benzimidazole | 1-[(4-chlorophenyl)methyl]-2-methyl-benzimidazole | 1-[(4-chlorophenyl)methyl]-2-methylbenzimidazole | MLS001240197 | SMR000674565 | cid_71821
Type:
Small organic molecule
Emp. Form.:
C15H13ClN2
Mol. Mass.:
256.73
SMILES:
Cc1nc2ccccc2n1Cc1ccc(Cl)cc1
Structure:
Search PDB for entries with ligand similarity: