Reaction Details
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Target
Tyrosine--tRNA ligase
Ligand
BDBM199148
Substrate
n/a
Meas. Tech.
In vitro Enzyme Inhibition Assay
pH
7.9±n/a
IC50
9.542e+4± 3.1e+2 nM
Comments
extracted
Citation
More Info.:
Target
Name:
Tyrosine--tRNA ligase
Synonyms:
SYY_STAAS | Tyrosyl-tRNA synthetase | tyrS
Type:
Protein
Mol. Mass.:
47586.43
Organism:
Staphylococcus aureus (strain MSSA476)
Description:
n/a
Residue:
420
Sequence:
MTNVLIEDLKWRGLIYQQTDEQGIEDLLNKEQVTLYCGADPTADSLHIGHLLPFLTLRRFQEHGHRPIVLIGGGTGMIGDPSGKSEERVLQTEEQVDKNIEGISKQMHNIFEFGTDHGAVLVNNRDWLGQISLISFLRDYGKHVGVNYMLGKDSIQSRLEHGISYTEFTYTILQAIDFGHLNRELNCKIQVGGSDQWGNITSGIELMRRMYGQTDAYGLTIPLVTKSDGKKFGKSESGAVWLDAEKTSPYEFYQFWINQSDEDVIKFLKYFTFLGKEEIDRLEQSKNEAPHLREAQKTLAEEVTKFIHGEDALNDAIRISQALFSGDLKSLSAKELKDGFKDVPQVTLSNDTTNIVEVLIETGISPSKRQAREDVNNGAIYINGERQQDVNYALAPEDKIDGEFTIIRRGKKKYFMVNYQ