Reaction Details
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Target
Glucocorticoid receptor
Ligand
BDBM50265673
Substrate
n/a
Meas. Tech.
ChEMBL_1700185 (CHEMBL4051167)
Ki
>10000±n/a nM
Citation
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More Info.:
Target
Name:
Glucocorticoid receptor
Synonyms:
Glucocorticoid receptor isoform alpha variant 1 | Glucocorticoid receptor isoform alpha variant 2 | NR3C1 | Nuclear receptor subfamily 3 group C member 1
Type:
PROTEIN
Mol. Mass.:
86027.98
Organism:
Canis lupus familiaris
Description:
ChEMBL_117571
Residue:
781
Sequence:
MDSKESLSPPSKEEISSSVLGRERGNVMDFYKTLRGGATVKVSASSPSLAAASQSDSKQQRLLVDFPKGSGSHAQQPDLSKAVSLSMGLYMGETETKVMGNDLGFPQQGQISLSSGETDFRLLEESIANLNRSTSVPENPKSSVSAVSAAPTEKEFAQTLSDVSSEQQHLKGQTGTNGGNVKLYTTDQSTFDVWRKKLQDLDFTSGSPEKEASESPWRSDLLIDENCLLSPLAGEDDPFLLEGNSNEDCKPLVLPDTKPKIKDNGDLILASPNSVPLPQVKTEKEDFIELCTPGVIKQEKLGPVYCQASFSGANIIGNKMSAISVHGVSTSGGQMYHYDMNTASLSQQQDQKPIFNVIPPIPVGSENWNRCQGSGDDNLASLGTLNFPGRSVFSNGYSSPGMRPDVSSPPSSSSAATGPPPKLCLVCSDEASGCHYGVLTCGSCKVFFKRAVEGRQHNYLCAGRNDCIIDKIRRKNCPACRYRKCLQAGMNLEARKTKKKIKGIQQATPGASQETSENPANKTIVPATLPQLTPTLVSLLEVIEPEVLYAGYDSSVPDSTWRIMTTLNMLGGRQVIAAVKWAKAIPGFRNLHLDDQMTLLQYSWMFLMAFALGWRSYRQSSGSMLCFAPDLIINEQRMTLPCMYDQCKHMLFVSSELQRLQVSYEEYLCMKTLLLLSSVPKEGLKSQELFDEIRMTYIKELGKAIVKREGNSSQNWQRFYQLTKLLDSMHDVVENLLNFCFQTFLDKTMSIEFPEMLAEIITNQIPKYSSGNIKKLLFHQK