Reaction Details Report a problem with these data
Target
Interleukin 1 receptor associated kinase 4
Ligand
BDBM50204290
Substrate
n/a
Meas. Tech.
Radiometric Protein Kinase Assay
IC50
17.7±n/a nM
Citation
Griebenow, N; Mottier, MD; Beddies, G; Cramer, J; Bömer, U; Heisler, I Use of fused heteroaromatic pyrrolidones for treatment and prevention of diseases in animals US Patent US11077111 Publication Date 8/3/2021
More Info.:
Target
Name:
Interleukin 1 receptor associated kinase 4
Synonyms:
Interleukin-1 receptor-associated kinase 4
Type:
Protein
Mol. Mass.:
51392.15
Organism:
Dog
Description:
A0A8I3Q059
Residue:
466
Sequence:
MLCGRGPGGSFVVWAGRGRGLTGRPRPTPVPFGAPGSLRQPAQRGGASVPRCSGFPLLARRFEALLQTGKSPTCELLFDWGTTNCTVGDLVDLLIQNEFFAPASLLLPDAIPKTPNTVPSEEAVTVQQQQMPLNGKDRTFVLPVQNFEQNYMPPDSSSPENTSLEGSDTRFHSFSFYELKNVTNNFDERPISLGGNKMGEGGFGVVYKGYVNNKTVAVKKLAAMVDISTEELKQQFDQEIKVMAKCQHENLVELLGFSSDGDDLCLVYVYMPNGSLLDRLSCLDGTPPLSWHMRCKIAQGAANGISFLHENHHIHRDIKSANILLDEDFTAKVSDFGLARASEKFAQTVMTSRIVGTTAYMAPEALRGEITPKSDIYSFGVVLLEIITGLPAVDEHREPQLLLDIKEEIEDEEKTIEDYIDPKMNDTDPTSIETMYSVASQCLHEKKNKRPDIEKVQQLLQDLTAS