Reaction Details Report a problem with these data
Target
Bromodomain testis-specific protein [22-138]
Ligand
BDBM562599
Substrate
n/a
Meas. Tech.
Acetyl-Histone Binding Assay
IC50
61.0±n/a nM
Citation
 Bradner, JE; Qi, J; Tanaka, M Acetamide thienotriazolodiazepines and uses thereof US Patent  US11406645 Publication Date 8/9/2022 
Target
Name:
Bromodomain testis-specific protein [22-138]
Synonyms:
BRDT | BRDT_HUMAN | Bromodomain testis-specific protein (BRDT)(BD1)
Type:
n/a
Mol. Mass.:
13948.58
Organism:
Homo sapiens (Human)
Description:
Q58F21[22-138]
Residue:
117
Sequence:
TKKNGRLTNQLQYLQKVVLKDLWKHSFSWPFQRPVDAVKLQLPDYYTIIKNPMDLNTIKKRLENKYYAKASECIEDFNTMFSNCYLYNKPGDDIVLMAQALEKLFMQKLSQMPQEEQ
  
Inhibitor
Name:
BDBM562599
Synonyms:
US11406645, Compound 502
Type:
Small organic molecule
Emp. Form.:
C22H24ClN5O2S
Mol. Mass.:
457.976
SMILES:
C[C@@H](O)CNC(=O)C[C@@H]1N=C(c2c(C)c(C)sc2-n2c(C)nnc12)c1ccc(Cl)cc1 |r,c:9|
Structure:
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