Reaction Details Report a problem with these data
Target
Calmodulin-1
Ligand
BDBM588489
Substrate
n/a
Meas. Tech.
Fluorescence Polarization Assay
IC50
2970±n/a nM
Citation
Bumcrot, DA; Sehgal, A; Hertzog, DL Phenothiazine derivatives and uses thereof US Patent US11542290 Publication Date 1/3/2023
More Info.:
Target
Name:
Calmodulin-1
Synonyms:
CALM | CALM1 | CALM1_HUMAN | CALM2 | CAM | CAM1 | CAM2 | CAMB | Calmodulin-2
Type:
Protein
Mol. Mass.:
16813.73
Organism:
Human
Description:
P0DP23
Residue:
149
Sequence:
MADQLTEEQIAEFKEAFSLFDKDGDGTITTKELGTVMRSLGQNPTEAELQDMINEVDADGNGTIDFPEFLTMMARKMKDTDSEEEIREAFRVFDKDGNGYISAAELRHVMTNLGEKLTDEEVDEMIREADIDGDGQVNYEEFVQMMTAK