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Target
Inward rectifier potassium channel 13
Ligand
BDBM600745
Substrate
n/a
Meas. Tech.
thallium-flux assay
IC50
>30000±n/a nM
Citation
 Swale, DR; Foil, LD Method for controlling hematophagous or sap-feeding arthropods US Patent  US11632953 Publication Date 4/25/2023 
Target
Name:
Inward rectifier potassium channel 13
Synonyms:
Inward rectifier K(+) channel Kir7.1 | KCJ13_HUMAN | KCNJ13 | Potassium channel, inwardly rectifying subfamily J member 13
Type:
PROTEIN
Mol. Mass.:
40527.12
Organism:
Homo sapiens (Human)
Description:
ChEMBL_105176
Residue:
360
Sequence:
MDSSNCKVIAPLLSQRYRRMVTKDGHSTLQMDGAQRGLAYLRDAWGILMDMRWRWMMLVFSASFVVHWLVFAVLWYVLAEMNGDLELDHDAPPENHTICVKYITSFTAAFSFSLETQLTIGYGTMFPSGDCPSAIALLAIQMLLGLMLEAFITGAFVAKIARPKNRAFSIRFTDTAVVAHMDGKPNLIFQVANTRPSPLTSVRVSAVLYQERENGKLYQTSVDFHLDGISSDECPFFIFPLTYYHSITPSSPLATLLQHENPSHFELVVFLSAMQEGTGEICQRRTSYLPSEIMLHHCFASLLTRGSKGEYQIKMENFDKTVPEFPTPLVSKSPNRTDLDIHINGQSIDNFQISETGLTE
  
Inhibitor
Name:
BDBM600745
Synonyms:
US11632953, Compound 1 | US11632953, Compound VU041
Type:
Small organic molecule
Emp. Form.:
C19H20F3N3O
Mol. Mass.:
363.3768
SMILES:
FC(F)(F)c1nn(CC(=O)N2CCCc3ccccc23)c2CCCCc12
Structure:
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