Reaction Details Report a problem with these data
Target
Histone deacetylase 4 [648-1032]
Ligand
BDBM243178
Substrate
n/a
Meas. Tech.
HDAC4 Biochemical Assay
IC50
11.0±n/a nM
Citation
Maillard, MC; Breccia, P; Dominguez, C; Haughan, AF; Van de Poël, A; Stott, AJ; Luckhurst, CA; Saville-Stones, EA; Wishart, G; Wall, M; Jarvis, RE Histone deacetylase inhibitors and compositions and methods of use thereof US Patent US10053434 Publication Date 8/21/2018
More Info.:
Target
Name:
Histone deacetylase 4 [648-1032]
Synonyms:
HDAC4 | HDAC4_HUMAN | Histone deacetylase 4 | KIAA0288
Type:
Enzyme
Mol. Mass.:
41490.90
Organism:
Homo sapiens (Human)
Description:
P56524[648-1032]
Residue:
385
Sequence:
TKPRFTTGLVYDTLMLKHQCTCGSSSSHPEHAGRIQSIWSRLQETGLRGKCECIRGRKATLEELQTVHSEAHTLLYGTNPLNRQKLDSKKLLGSLASVFVRLPCGGVGVDSDTIWNEVHSAGAARLAVGCVVELVFKVATGELKNGFAVVRPPGHHAEESTPMGFCYFNSVAVAAKLLQQRLSVSKILIVDWDVHHGNGTQQAFYSDPSVLYMSLHRYDDGNFFPGSGAPDEVGTGPGVGFNVNMAFTGGLDPPMGDAEYLAAFRTVVMPIASEFAPDVVLVSSGFDAVEGHPTPLGGYNLSARCFGYLTKQLMGLAGGRIVLALEGGHDLTAICDASEACVSALLGNELDPLPEKVLQQRPNANAVRSMEKVMEIHSKYWRCLQ