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Target
fMet-Leu-Phe receptor
Ligand
BDBM37754
Substrate
n/a
Meas. Tech.
Dose Response Assay for Formylpeptide Receptor (FPR) Ligands and Dose Response Counter-Screen Assay for Formylpeptide-Like-1 (FPRL1) Ligands
Ki
>43700±n/a nM
Citation
 PubChem, PC Dose Response Assay for Formylpeptide Receptor (FPR) Ligands and Dose Response Counter-Screen Assay for Formylpeptide-Like-1 (FPRL1) Ligands PubChem Bioassay (2007)[AID] 
Target
Name:
fMet-Leu-Phe receptor
Synonyms:
FPR | FPR1 | FPR1_HUMAN | Formyl peptide Receptor | N-formyl peptide receptor 1 | N-formylpeptide chemoattractant receptor | fMLP receptor | fMet-Leu-Phe receptor | formyl peptide receptor 1
Type:
Enzyme Catalytic Domain
Mol. Mass.:
38456.14
Organism:
Homo sapiens (Human)
Description:
gi_4503779
Residue:
350
Sequence:
METNSSLPTNISGGTPAVSAGYLFLDIITYLVFAVTFVLGVLGNGLVIWVAGFRMTHTVTTISYLNLAVADFCFTSTLPFFMVRKAMGGHWPFGWFLCKFVFTIVDINLFGSVFLIALIALDRCVCVLHPVWTQNHRTVSLAKKVIIGPWVMALLLTLPVIIRVTTVPGKTGTVACTFNFSPWTNDPKERINVAVAMLTVRGIIRFIIGFSAPMSIVAVSYGLIATKIHKQGLIKSSRPLRVLSFVAAAFFLCWSPYQVVALIATVRIRELLQGMYKEIGIAVDVTSALAFFNSCLNPMLYVFMGQDFRERLIHALPASLERALTEDSTQTSDTATNSTLPSAEVELQAK
  
Inhibitor
Name:
BDBM37754
Synonyms:
MLS000045942 | N-(5-imidazo[1,2-a]pyrimidin-2-yl-2-methoxy-phenyl)butanamide | N-(5-imidazo[1,2-a]pyrimidin-2-yl-2-methoxy-phenyl)butyramide | N-(5-imidazo[1,2-a]pyrimidin-2-yl-2-methoxyphenyl)butanamide | N-[5-(2-imidazo[1,2-a]pyrimidinyl)-2-methoxyphenyl]butanamide | SMR000028314 | cid_3245971
Type:
Small organic molecule
Emp. Form.:
C17H18N4O2
Mol. Mass.:
310.3504
SMILES:
CCCC(=O)Nc1cc(ccc1OC)-c1cn2cccnc2n1
Structure:
Search PDB for entries with ligand similarity: