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Target
Galanin receptor type 2
Ligand
BDBM42052
Substrate
n/a
Meas. Tech.
Dose Response cell-based high-throughput screening assay to identify antagonists of galanin receptor 2 (GALR2)
IC50
1289±n/a nM
Citation
 PubChem, PC Dose Response cell-based high-throughput screening assay to identify antagonists of galanin receptor 2 (GALR2) PubChem Bioassay (2008)[AID] 
Target
Name:
Galanin receptor type 2
Synonyms:
GALNR2 | GALR2 | GALR2_HUMAN | Galanin R2 | Galanin receptor 2 | Galanin receptor type 2 | Galanin receptor type 2 (GAL2-R) (GALR2).
Type:
Enzyme Catalytic Domain
Mol. Mass.:
41724.40
Organism:
Homo sapiens (Human)
Description:
Galanin R2 GALR2 HUMAN::O43603
Residue:
387
Sequence:
MNVSGCPGAGNASQAGGGGGWHPEAVIVPLLFALIFLVGTVGNTLVLAVLLRGGQAVSTTNLFILNLGVADLCFILCCVPFQATIYTLDGWVFGSLLCKAVHFLIFLTMHASSFTLAAVSLDRYLAIRYPLHSRELRTPRNALAAIGLIWGLSLLFSGPYLSYYRQSQLANLTVCHPAWSAPRRRAMDICTFVFSYLLPVLVLGLTYARTLRYLWRAVDPVAAGSGARRAKRKVTRMILIVAALFCLCWMPHHALILCVWFGQFPLTRATYALRILSHLVSYANSCVNPIVYALVSKHFRKGFRTICAGLLGRAPGRASGRVCAAARGTHSGSVLERESSDLLHMSEAAGALRPCPGASQPCILEPCPGPSWQGPKAGDSILTVDVA
  
Inhibitor
Name:
BDBM42052
Synonyms:
2-N,3-N-dimethyl-6,7-dinitroquinoxaline-2,3-diamine | MLS000579073 | N,N'-(6,7-dinitro-1,4-dihydroquinoxaline-2,3-diylidene)dimethanamine | N2,N3-dimethyl-6,7-dinitro-quinoxaline-2,3-diamine | N2,N3-dimethyl-6,7-dinitroquinoxaline-2,3-diamine | SMR000186662 | cid_4686258 | methyl-[3-(methylamino)-6,7-dinitro-quinoxalin-2-yl]amine
Type:
Small organic molecule
Emp. Form.:
C10H10N6O4
Mol. Mass.:
278.2242
SMILES:
CNc1nc2cc(c(cc2nc1NC)[N+]([O-])=O)[N+]([O-])=O
Structure:
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