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Target
Matrix metalloproteinase-14 [1-36]
Ligand
BDBM48174
Substrate
n/a
Meas. Tech.
Luminescent HTS for small molecule inhibitors of MT1-MMP transcription
EC50
5620±n/a nM
Citation
 PubChem, PC Luminescent HTS for small molecule inhibitors of MT1-MMP transcription PubChem Bioassay (2008)[AID] 
Target
Name:
Matrix metalloproteinase-14 [1-36]
Synonyms:
MMP14 | MMP14_PONAB | matrix metalloproteinase 1
Type:
Enzyme Catalytic Domain
Mol. Mass.:
3658.23
Organism:
Homo sapiens (Human)
Description:
gi_6690534
Residue:
36
Sequence:
MSPAPRPSRCLLLPLLTLGTALASLGSAQSSSFSPE
  
Inhibitor
Name:
BDBM48174
Synonyms:
2-methyl-N-[2-(4-methylphenyl)-1,3-benzoxazol-5-yl]propanamide | 2-methyl-N-[2-(p-tolyl)-1,3-benzoxazol-5-yl]propionamide | MLS000109481 | SMR000105424 | cid_1364012
Type:
Small organic molecule
Emp. Form.:
C18H18N2O2
Mol. Mass.:
294.3477
SMILES:
CC(C)C(=O)Nc1ccc2oc(nc2c1)-c1ccc(C)cc1
Structure:
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