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Target
Matrix metalloproteinase-14 [1-36]
Ligand
BDBM48240
Substrate
n/a
Meas. Tech.
Luminescent HTS for small molecule inhibitors of MT1-MMP transcription
EC50
540±n/a nM
Citation
 PubChem, PC Luminescent HTS for small molecule inhibitors of MT1-MMP transcription PubChem Bioassay (2008)[AID] 
Target
Name:
Matrix metalloproteinase-14 [1-36]
Synonyms:
MMP14 | MMP14_PONAB | matrix metalloproteinase 1
Type:
Enzyme Catalytic Domain
Mol. Mass.:
3658.23
Organism:
Homo sapiens (Human)
Description:
gi_6690534
Residue:
36
Sequence:
MSPAPRPSRCLLLPLLTLGTALASLGSAQSSSFSPE
  
Inhibitor
Name:
BDBM48240
Synonyms:
2-Phenyl-6,7,8,9-tetrahydro-benzo[e]imidazo[1,2-b][1,2,4]triazine | 2-phenyl-6,7,8,9-tetrahydroimidazo[1,2-b][1,2,4]benzotriazine | MLS000554665 | SMR000146782 | cid_619518
Type:
Small organic molecule
Emp. Form.:
C15H14N4
Mol. Mass.:
250.2985
SMILES:
C1CCc2nn3cc(nc3nc2C1)-c1ccccc1
Structure:
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