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Target
Trans-activator protein BZLF1
Ligand
BDBM50018
Substrate
n/a
Meas. Tech.
Counterscreen for inhibitors of EBNA-1: fluorescence polarization-based biochemical high throughput dose response assay to identify inhibitors of the Epstein-Barr virus-encoded protein, ZTA
IC50
111248±n/a nM
Citation
 PubChem, PC Counterscreen for inhibitors of EBNA-1: fluorescence polarization-based biochemical high throughput dose response assay to identify inhibitors of the Epstein-Barr virus-encoded protein, ZTA PubChem Bioassay (2010)[AID] 
Target
Name:
Trans-activator protein BZLF1
Synonyms:
BZLF1 | BZLF1_EBVB9 | PPP5C protein
Type:
Enzyme Catalytic Domain
Mol. Mass.:
26856.37
Organism:
Human herpesvirus 4
Description:
gi_82503229
Residue:
245
Sequence:
MMDPNSTSEDVKFTPDPYQVPFVQAFDQATRVYQDLGGPSQAPLPCVLWPVLPEPLPQGQLTAYHVSTAPTGSWFSAPQPAPENAYQAYAAPQLFPVSDITQNQQTNQAGGEAPQPGDNSTVQTAAAVVFACPGANQGQQLADIGVPQPAPVAAPARRTRKPQQPESLEECDSELEIKRYKNRVASRKCRAKFKQLLQHYREVAAAKSSENDRLRLLLKQMCPSLDVDSIIPRTPDVLHEDLLNF
  
Inhibitor
Name:
BDBM50018
Synonyms:
3-amino-6-(2-furanyl)-N-phenyl-2-thieno[2,3-b]pyridinecarboxamide | 3-amino-6-(2-furyl)-N-phenyl-thieno[2,3-b]pyridine-2-carboxamide | 3-amino-6-(furan-2-yl)-N-phenylthieno[2,3-b]pyridine-2-carboxamide | 3-azanyl-6-(furan-2-yl)-N-phenyl-thieno[2,3-b]pyridine-2-carboxamide | MLS000042179 | SMR000048500 | cid_667115
Type:
Small organic molecule
Emp. Form.:
C18H13N3O2S
Mol. Mass.:
335.38
SMILES:
Nc1c(sc2nc(ccc12)-c1ccco1)C(=O)Nc1ccccc1
Structure:
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