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Target
Trans-activator protein BZLF1
Ligand
BDBM62440
Substrate
n/a
Meas. Tech.
Counterscreen for inhibitors of EBNA-1: fluorescence polarization-based biochemical high throughput dose response assay to identify inhibitors of the Epstein-Barr virus-encoded protein, ZTA
IC50
111183±n/a nM
Citation
 PubChem, PC Counterscreen for inhibitors of EBNA-1: fluorescence polarization-based biochemical high throughput dose response assay to identify inhibitors of the Epstein-Barr virus-encoded protein, ZTA PubChem Bioassay (2010)[AID] 
Target
Name:
Trans-activator protein BZLF1
Synonyms:
BZLF1 | BZLF1_EBVB9 | PPP5C protein
Type:
Enzyme Catalytic Domain
Mol. Mass.:
26856.37
Organism:
Human herpesvirus 4
Description:
gi_82503229
Residue:
245
Sequence:
MMDPNSTSEDVKFTPDPYQVPFVQAFDQATRVYQDLGGPSQAPLPCVLWPVLPEPLPQGQLTAYHVSTAPTGSWFSAPQPAPENAYQAYAAPQLFPVSDITQNQQTNQAGGEAPQPGDNSTVQTAAAVVFACPGANQGQQLADIGVPQPAPVAAPARRTRKPQQPESLEECDSELEIKRYKNRVASRKCRAKFKQLLQHYREVAAAKSSENDRLRLLLKQMCPSLDVDSIIPRTPDVLHEDLLNF
  
Inhibitor
Name:
BDBM62440
Synonyms:
MLS000578646 | N-[(E)-1-(1H-benzimidazol-2-yl)-2-(4-bromophenyl)ethenyl]-2-furancarboxamide | N-[(E)-1-(1H-benzimidazol-2-yl)-2-(4-bromophenyl)ethenyl]furan-2-carboxamide | N-[(E)-1-(1H-benzimidazol-2-yl)-2-(4-bromophenyl)vinyl]-2-furamide | N-[1-(1H-benzimidazol-2-yl)-2-(4-bromophenyl)vinyl]-2-furamide | SMR000186139 | cid_5340350
Type:
Small organic molecule
Emp. Form.:
C20H14BrN3O2
Mol. Mass.:
408.248
SMILES:
Brc1ccc(\C=C(\NC(=O)c2ccco2)c2nc3ccccc3[nH]2)cc1
Structure:
Search PDB for entries with ligand similarity: