Reaction Details Report a problem with these data
Target
Cell division protein FtsZ
Ligand
BDBM81335
Substrate
n/a
Meas. Tech.
Fluorescent Coupled Assay
pH
7.5±0
IC50
6.02e+4± 8.8e+3 nM
Citation
Läppchen, T; Pinas, VA; Hartog, AF; Koomen, GJ; Schaffner-Barbero, C; Andreu, JM; Trambaiolo, D; Löwe, J; Juhem, A; Popov, AV; den Blaauwen, T Probing FtsZ and tubulin with C8-substituted GTP analogs reveals differences in their nucleotide binding sites. Chem Biol 15:189-99 (2008) [PubMed] Article
More Info.:
Target
Name:
Cell division protein FtsZ
Synonyms:
FTSZ_AQUAE | ftsZ
Type:
Protein
Mol. Mass.:
40146.54
Organism:
Aquifex aeolicus
Description:
O66809
Residue:
367
Sequence:
MEEFVNPCKIKVIGVGGGGSNAVNRMYEDGIEGVELYAINTDVQHLSTLKVPNKIQIGEKVTRGLGAGAKPEVGEEAALEDIDKIKEILRDTDMVFISAGLGGGTGTGAAPVIAKTAKEMGILTVAVATLPFRFEGPRKMEKALKGLEKLKESSDAYIVIHNDKIKELSNRTLTIKDAFKEVDSVLSKAVRGITSIVVTPAVINVDFADVRTTLEEGGLSIIGMGEGRGDEKADIAVEKAVTSPLLEGNTIEGARRLLVTIWTSEDIPYDIVDEVMERIHSKVHPEAEIIFGAVLEPQEQDFIRVAIVATDFPEEKFQVGEKEVKFKVIKKEEKEEPKEEPKPLSDTTYLEEEEIPAVIRRKNKRLL