Reaction Details Report a problem with these data
Target
Olfactory receptor
Ligand
BDBM81351
Substrate
n/a
Meas. Tech.
Inhibition Assay
IC50
3.7e+4± 1.2e+4 nM
Citation
Peterlin, Z; Li, Y; Sun, G; Shah, R; Firestein, S; Ryan, K The importance of odorant conformation to the binding and activation of a representative olfactory receptor. Chem Biol 15:1317-27 (2008) [PubMed] Article
More Info.:
Target
Name:
Olfactory receptor
Synonyms:
Olfactory receptor 17 | Olr17
Type:
Protein
Mol. Mass.:
35760.42
Organism:
Rattus norvegicus (Rat)
Description:
D3Z9H0
Residue:
346
Sequence:
MFVPVLITSHPRSPGCCSSPSGQRKRNMDVKNRTAVTEFIFLGFPGSSSLQLPLFMIFLIVYLLSLMGNTLIIFLILMDSTLQTPMYIFLGNLSFLEIWYTTATVPKLLATCVTKVVTIPVAGCITQYYFFFSLGATECILLAVMAYDRHVAVCRPLHYSLLMSVHICLRFAAASWIGGFIAPLLPTILVSQLNFCGPQKINHFFCDSDPIFKLSCSDTFLVEALGYTCTSVVILSSFLLTMSSYGNIVVTIIRLSSREARKKTFSTCASHLTVVTMYYGTIIFAYVRPPAKYNFTIGKVVSVFYCVITPLVNPLTYTLRNKDVMKAFQKFLSQKRFLSGKTMHAV