Reaction Details Report a problem with these data
Target
Hrh3 protein
Ligand
BDBM7882
Substrate
n/a
Ki
>10000±n/a nM
Comments
PDSP_970
Citation
 West, RE; Zweig, A; Granzow, RT; Siegel, MI; Egan, RW Biexponential kinetics of (R)-alpha-[3H]methylhistamine binding to the rat brain H3 histamine receptor. J Neurochem 55:1612-6 (1990) [PubMed]  Article 
Target
Name:
Hrh3 protein
Synonyms:
HISTAMINE H3 | HRH3 | Hrh3 protein
Type:
Enzyme Catalytic Domain
Mol. Mass.:
37860.96
Organism:
RAT
Description:
Q5PPG3
Residue:
344
Sequence:
MERAPPDGLMNASGTLAGEAAAAGGARGFSAAWTAVLAALMALLIVATVLGNALVMLAFVADSSLRTQNNFFLLNLAISDFLVGAFCIPLYVPYVLTGRWTFGRGLCKLWLVVDYLLCASSVFNIVLISYDRFLSVTRAVSYRAQQGDTRRAVRKMALVWVLAFLLYGPAILSWEYLSGGSSIPEGHCYAEFFYNWYFLITASTLEFFTPFLSVTFFNLSIYLNIQRRTRLRLDGGREAGPEPPPDAQPSPPPAPPSCWGCWPKGHGEAMPLHRGSKPSASSASLEKRMKMVSQSITQRFRLSRDKKVAKSLAIIVSIFGLCWAPYTLLMIIRAACHGRCIPDY
  
Inhibitor
Name:
BDBM7882
Synonyms:
1H-imidazole | CHEMBL540 | Imidazole (Im) | US9138393, Imidazole | US9144538, Imidazole | imidazole
Type:
Small organic molecule
Emp. Form.:
C3H4N2
Mol. Mass.:
68.0773
SMILES:
c1c[nH]cn1
Structure:
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