Reaction Details
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Report a problem with these dataTarget
Norepinephrine transporter
Ligand
BDBM50021217
Substrate
n/a
Ki
0.79±n/a nM
Comments
PDSP_3888
Citation
Hyttel, J; Larsen, JJ Neurochemical profile of Lu 19-005, a potent inhibitor of uptake of dopamine, noradrenaline, and serotonin. J Neurochem 44:1615-22 (1985) [PubMed] Article More Info.:
Target
Name:
Norepinephrine transporter
Synonyms:
n/a
Type:
Enzyme Catalytic Domain
Mol. Mass.:
2082.45
Organism:
RAT
Description:
Norepinephrine transporter 0 RAT::Q9JIA2
Residue:
19
Sequence:
MLLARMKPQVQPELGGADQ
Inhibitor
Name:
BDBM50021217
Synonyms:
CHEMBL52247 | Talsupram | [3-(3,3-Dimethyl-1-phenyl-1,3-dihydro-benzo[c]thiophen-1-yl)-propyl]-methyl-amine(Talsupram)
Type:
Small organic molecule
Emp. Form.:
C20H25NS
Mol. Mass.:
311.484
SMILES:
CNCCCC1(SC(C)(C)c2ccccc12)c1ccccc1
Structure:
