Reaction Details
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Report a problem with these dataTarget
Norepinephrine transporter
Ligand
BDBM82218
Substrate
n/a
Ki
380±n/a nM
Comments
PDSP_4198
Citation
Koe, BK; Weissman, A; Welch, WM; Browne, RG Sertraline, 1S,4S-N-methyl-4-(3,4-dichlorophenyl)-1,2,3,4-tetrahydro-1-naphthylamine, a new uptake inhibitor with selectivity for serotonin. J Pharmacol Exp Ther 226:686-700 (1983) [PubMed] More Info.:
Target
Name:
Norepinephrine transporter
Synonyms:
n/a
Type:
Enzyme Catalytic Domain
Mol. Mass.:
2082.45
Organism:
RAT
Description:
Norepinephrine transporter 0 RAT::Q9JIA2
Residue:
19
Sequence:
MLLARMKPQVQPELGGADQ
Inhibitor
Name:
BDBM82218
Synonyms:
CP-51973
Type:
n/a
Emp. Form.:
C17H17Cl2N
Mol. Mass.:
306.23
SMILES:
CN[C@@H]1CC[C@H](c2ccc(Cl)c(Cl)c2)c2ccccc12
Structure:
