Reaction Details
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Report a problem with these dataTarget
Thromboxane A2 receptor
Ligand
BDBM82227
Substrate
n/a
Ki
>10000±n/a nM
Comments
PDSP_4874
Citation
Armstrong, RA; Jones, RL; Wilson, NH Ligand binding to thromboxane receptors on human platelets: correlation with biological activity. Br J Pharmacol 79:953-64 (1983) [PubMed] Article More Info.:
Target
Name:
Thromboxane A2 receptor
Synonyms:
TA2R_MOUSE | Tbxa2r | Thromboxane A2
Type:
Enzyme Catalytic Domain
Mol. Mass.:
37114.77
Organism:
MOUSE
Description:
Thromboxane A2 TBXA2R MOUSE::P30987
Residue:
341
Sequence:
MWPNGTSLGACFRPVNITLQERRAIASPWFAASFCALGLGSNLLALSVLAGARPGAGPRSSFLALLCGLVLTDFLGLLVTGAIVASQHAALLDWRATDPSCRLCYFMGVAMVFFGLCPLLLGAAMASERFVGITRPFSRPTATSRRAWATVGLVWVAAGALGLLPLLGLGRYSVQYPGSWCFLTLGTQRGDVVFGLIFALLGSASVGLSLLLNTVSVATLCRVYHTREATQRPRDCEVEMMVQLVGIMVVATVCWMPLLVFIMQTLLQTPPVMSFSGQLLRATEHQLLIYLRVATWNQILDPWVYILFRRSVLRRLHPRFSSQLQAVSLRRPPAQAMLSGP
Inhibitor
Name:
BDBM82227
Synonyms:
15-methyl PGF2alpha | CAS_37255 | NSC_37255
Type:
Small organic molecule
Emp. Form.:
C21H36O5
Mol. Mass.:
368.5075
SMILES:
CCCCCC(C)(O)C=CC1C(O)CC(O)C1CC=CCCCC(O)=O |w:8.7,18.18|
Structure:
