Reaction Details Report a problem with these data
Target
Neurotensin
Ligand
BDBM82418
Substrate
n/a
Ki
1600±n/a nM
Comments
PDSP_1307
Citation
 Betancur, C; Canton, M; Gully, D; Vela, G; Pélaprat, D; Rostène, W Characterization and distribution of binding sites for a new neurotensin receptor antagonist ligand, [3H]SR 48692, in the guinea pig brain. J Pharmacol Exp Ther 273:1450-8 (1995) [PubMed] 
Target
Name:
Neurotensin
Synonyms:
NEUT_CAVPO | NT | NTS | Neurotensin
Type:
Enzyme Catalytic Domain
Mol. Mass.:
1681.93
Organism:
GUINEA PIG
Description:
NT 0 GUINEA PIG::P32560
Residue:
13
Sequence:
QLYENKSRRPYIL
  
Inhibitor
Name:
BDBM82418
Synonyms:
CAS_3025353 | NSC_3025353 | Neuromedin N
Type:
Small organic molecule
Emp. Form.:
C38H63N7O8
Mol. Mass.:
745.9489
SMILES:
CCC(C)C(N)C(=O)C(C)(CC(=O)C(N)CCCCN)C(C(=O)C(N)Cc1ccc(O)cc1)(C(=O)C1CCCN1)C(N)(C(O)=O)C(=O)C(N)C(C)CC
Structure:
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