Reaction Details Report a problem with these data
Target
Similar to alpha-tubulin isoform 1
Ligand
BDBM50470020
Substrate
n/a
Meas. Tech.
ChEMBL_211352 (CHEMBL873906)
IC50
450±n/a nM
Citation
 Li, L; Wang, HK; Kuo, SC; Wu, TS; Mauger, A; Lin, CM; Hamel, E; Lee, KH Antitumor agents. 155. Synthesis and biological evaluation of 3',6,7-substituted 2-phenyl-4-quinolones as antimicrotubule agents. J Med Chem 37:3400-7 (1994) [PubMed]  Article 
Target
Name:
Similar to alpha-tubulin isoform 1
Synonyms:
Similar to alpha-tubulin isoform 1
Type:
PROTEIN
Mol. Mass.:
10383.05
Organism:
Bos taurus
Description:
ChEMBL_104716
Residue:
99
Sequence:
CVSASPSTLARLVSRSAMPAGSSTAWNTAFSPMARCQVTKTIGGGDDSFNTFFSETGAGKHVPRAVFVDLEPTVIDEVRTGTYRSSSTLSSSSQAKKMP
  
Inhibitor
Name:
BDBM50470020
Synonyms:
CHEMBL325260
Type:
Small organic molecule
Emp. Form.:
C23H17NO4
Mol. Mass.:
371.3854
SMILES:
Oc1cc(nc2cc3OCOc3cc12)-c1cccc(OCc2ccccc2)c1
Structure:
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