Reaction Details Report a problem with these data
Target
Alpha-1A adrenergic receptor
Ligand
BDBM50118702
Substrate
n/a
Meas. Tech.
ChEMBL_911064 (CHEMBL3056711)
EC50
7079±n/a nM
Citation
  TBA Med Chem Res 13:134-148 (2004)    Article 
Target
Name:
Alpha-1A adrenergic receptor
Synonyms:
ADA1A_RABIT | ADRA1A | ADRA1C | adrenergic Alpha1
Type:
Enzyme Catalytic Domain
Mol. Mass.:
51390.87
Organism:
RABBIT
Description:
adrenergic Alpha1 0 RABBIT::O02824
Residue:
466
Sequence:
MVFLSGNASDSSNCTHPPAPVNISKAILLGVILGGLILFGVLGNILVILSVACHRHLHSVTHYYIVNLAVADLLLTSTVLPFSAIFEILGYWAFGRVFCNIWAAVDVLCCTASIISLCVISIDRYIGVSYPLRYPTIVTQRRGLRALLCVWAFSLVISVGPLFGWRQPAPDDETICQINEEPGYVLFSALGSFYVPLTIILAMYCRVYVVAKRESRGLKSGLKTDKSDSEQVTLRIHRKNAPAGGSGVASAKNKTHFSVRLLKFSREKKAAKTLGIVVGCFVLCWLPFFLVMPIGSFFPDFKPPETVFKIVFWLGYLNSCINPIIYPCSSQEFKKAFQNVLKIQCLRRKQSSKHALGYTLHAPSQALEGQHKDMVRIPVGSGETFYKISKTDGVCEWKFFSSMPRGSARITVPKDQSACTTARVRSKSFLQVCCCVGPSTPNPGENHQVPTIKIHTISLSENGEEV
  
Inhibitor
Name:
BDBM50118702
Synonyms:
2-Amino-1-(2,5-dimethoxy-phenyl)-ethanol | CHEMBL1076 | DESGLYMIDODRINE | Orvaten | Proamatine
Type:
Small organic molecule
Emp. Form.:
C10H15NO3
Mol. Mass.:
197.231
SMILES:
COc1ccc(OC)c(c1)C(O)CN
Structure:
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