Reaction Details Report a problem with these data
Target
Platelet-activating factor receptor
Ligand
BDBM50035266
Substrate
n/a
Meas. Tech.
ChEMBL_158194 (CHEMBL767884)
IC50
13500±n/a nM
Citation
Sawyer, DA; Beams, RM; Blackwell, GJ; Brockwell, MA; Cheesman, NJ; Demaine, DA; Garland, LG; Hodson, HF; Hyde, RM; Islip, PJ Development of a novel series of trialkoxyaryl derivatives as specific and competitive antagonists of platelet activating factor. J Med Chem 38:2130-7 (1995) [PubMed] Article
More Info.:
Target
Name:
Platelet-activating factor receptor
Synonyms:
PAF-R | PTAFR | PTAFR_CAVPO | Platelet activating factor receptor | Platelet-activating factor receptor
Type:
Protein
Mol. Mass.:
39005.63
Organism:
Cavia porcellus
Description:
n/a
Residue:
342
Sequence:
MELNSSSRVDSEFRYTLFPIVYSIIFVLGIIANGYVLWVFARLYPSKKLNEIKIFMVNLTVADLLFLITLPLWIVYYSNQGNWFLPKFLCNLAGCLFFINTYCSVAFLGVITYNRFQAVKYPIKTAQATTRKRGIALSLVIWVAIVAAASYFLVMDSTNVVSNKAGSGNITRCFEHYEKGSKPVLIIHICIVLGFFIVFLLILFCNLVIIHTLLRQPVKQQRNAEVRRRALWMVCTVLAVFVICFVPHHMVQLPWTLAELGMWPSSNHQAINDAHQVTLCLLSTNCVLDPVIYCFLTKKFRKHLSEKLNIMRSSQKCSRVTTDTGTEMAIPINHTPVNPIKN