Reaction Details Report a problem with these data
Target
Interleukin-6 receptor subunit alpha
Ligand
BDBM85330
Substrate
n/a
Meas. Tech.
ChEMBL_220771 (CHEMBL842047)
Ki
>10000±n/a nM
Citation
van Wijngaarden, I; Hamminga, D; van Hes, R; Standaar, PJ; Tipker, J; Tulp, MT; Mol, F; Olivier, B; de Jonge, A Development of high-affinity 5-HT3 receptor antagonists. Structure-affinity relationships of novel 1,7-annelated indole derivatives. J Med Chem 36:3693-9 (1994) [PubMed] Article
More Info.:
Target
Name:
Interleukin-6 receptor subunit alpha
Synonyms:
IL6RA_RAT | Il6r | Il6ra | Interleukin-6 receptor alpha chain
Type:
PROTEIN
Mol. Mass.:
50182.76
Organism:
Rattus norvegicus
Description:
ChEMBL_218510
Residue:
460
Sequence:
MLAVGCTLLVALLAAPAVALVLGSCRALEVANGTVTSLPGATVTLICPGKEAAGNATIHWVYSGSQSREWTTTGNTLVLRAVQVNDTGHYLCFLDDHLVGTVPLLVDVPPEEPKLSCFRKNPLVNAFCEWHPSSTPSPTTKAVMFAKKINTTNGKSDFQVPCQYSQQLKSFSCEVEILEGDKVYHIVSLCVANSVGSRSSHNVVFQSLKMVQPDPPANLVVSAIPGPRWLKVSWQDPESWDPSYYLLQFELRYRPVWSKFTVWPLQVAQHQCVIHDALRGVKHVVQVRGKEEFDIGQWSKWSPEVTGTPWLAEPRTTPAGIPGNPTQVSVEDYDNHEDQYGSSTEATSVLAPVQGSSPIPLPTFLVAGGSLAFGLLLCVFIILRLKKKWKSQAEKESKTTSPPPYPLGPLKPTFLLVPLLTPSGSHNSSGTDNTGSHSCLGVRDPQCPNDNSNRDYLFPR