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Target
Mu-type opioid receptor
Ligand
BDBM50068136
Substrate
n/a
Meas. Tech.
ChEMBL_76016 (CHEMBL685497)
EC50
1250±n/a nM
Citation
 Liao, S; Alfaro-Lopez, J; Shenderovich, MD; Hosohata, K; Lin, J; Li, X; Stropova, D; Davis, P; Jernigan, KA; Porreca, F; Yamamura, HI; Hruby, VJ De novo design, synthesis, and biological activities of high-affinity and selective non-peptide agonists of the delta-opioid receptor. J Med Chem 41:4767-76 (1998) [PubMed]  Article 
Target
Name:
Mu-type opioid receptor
Synonyms:
M-OR-1 | MOR-1 | Mu opioid receptor | Mu-type opioid receptor (Mu) | OPIATE Mu | OPRM1 | OPRM_CAVPO
Type:
Enzyme Catalytic Domain
Mol. Mass.:
11165.58
Organism:
GUINEA PIG
Description:
P97266
Residue:
98
Sequence:
YTKMKTATNIYIFNLALADALATSTLPFQSVNYLMGTWPFGTILCKIVISIDYYNMFTSIFTLCTMSVDRYIAVCHPVKALDFRTPRNAKTVNVCNWI
  
Inhibitor
Name:
BDBM50068136
Synonyms:
3-[(4-Benzyl-piperazin-1-yl)-phenyl-methyl]-phenol | CHEMBL356587
Type:
Small organic molecule
Emp. Form.:
C24H26N2O
Mol. Mass.:
358.476
SMILES:
Oc1cccc(c1)C(N1CCN(Cc2ccccc2)CC1)c1ccccc1
Structure:
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